Catalytic regioselective construction of phenylthio- and phenoxyldifluoroalkyl tetrazoles from difluorodiazoketones DOI

Hong‐Song Shi,

Shuo-Han Li,

Fa‐Guang Zhang

и другие.

Chemical Communications, Год журнала: 2021, Номер 57(100), С. 13744 - 13747

Опубликована: Янв. 1, 2021

Here we report the design and synthesis of two new difluoro-diazoketone reagents (difluorophenylthiol diazoketone difluorophenoxyl diazoketone) their [3+2] cycloaddition reactions with aryldiazonium salts under silver catalysis conditions. This protocol enables regioselective access to a broad scope difluorophenylthiol- difluorophenoxyl-substituted tetrazole-carbinols in one-pot operation. Further synthetic derivatizations including dephenylthiolation unexpected phenylthiol group migration/fluorination allow efficient preparation α-difluoromethyl α-trifluoromethyl tetrazole-thioethers.

Язык: Английский

Recent Progress in Synthetic Applications of Hypervalent Iodine(III) Reagents DOI Creative Commons
Akira Yoshimura, Viktor V. Zhdankin

Chemical Reviews, Год журнала: 2024, Номер unknown

Опубликована: Сен. 13, 2024

Hypervalent iodine(III) compounds have found wide application in modern organic chemistry as environmentally friendly reagents and catalysts. iodine are commonly used synthetically important halogenations, oxidations, aminations, heterocyclizations, various oxidative functionalizations of substrates. Iodonium salts arylating reagents, while iodonium ylides imides excellent carbene nitrene precursors. Various derivatives benziodoxoles, such azidobenziodoxoles, trifluoromethylbenziodoxoles, alkynylbenziodoxoles, alkenylbenziodoxoles group transfer the presence transition metal catalysts, under metal-free conditions, or using photocatalysts photoirradiation conditions. Development hypervalent catalytic systems discovery highly enantioselective reactions chiral represent a particularly recent achievement field chemistry. Chemical transformations promoted by many cases unique cannot be performed any other common, non-iodine-based reagent. This review covers literature published mainly last 7-8 years, between 2016 2024.

Язык: Английский

Процитировано

37

Nitrogen-Based Organofluorine Functional Molecules: Synthesis and Applications DOI
Shuai Liu, Jun Zhou, Lu Yu

и другие.

Chemical Reviews, Год журнала: 2025, Номер unknown

Опубликована: Апрель 22, 2025

Fluorine and nitrogen form a successful partnership in organic synthesis, medicinal chemistry, material sciences. Although fluorine-nitrogen chemistry has long rich history, this field received increasing interest made remarkable progress over the past two decades, driven by recent advancements transition metal organocatalysis photochemistry. This review, emphasizing contributions from 2015 to 2023, aims update state of art synthesis applications nitrogen-based organofluorine functional molecules chemistry. In dedicated sections, we first focus on fluorine-containing reagents organized according type groups attached nitrogen, including N-F, N-RF, N-SRF, N-ORF. review also covers nitrogen-linked building blocks, catalysts, pharmaceuticals, agrochemicals, underlining these components' broad applicability growing importance modern

Язык: Английский

Процитировано

1

One‐Pot Reaction of (β‐Amino‐α,α‐difluoroethyl)phosphonates with Trifluoromethylated Ketones via Aza‐Wittig Reagents DOI
Qian Wang, Jiang Liu, Nana Wang

и другие.

Advanced Synthesis & Catalysis, Год журнала: 2022, Номер 364(12), С. 1969 - 1974

Опубликована: Апрель 30, 2022

Abstract We report a one‐pot reaction of (β‐amino‐α,α‐difluoroethyl)phosphonates involving aza‐Wittig reagents, in which, difluoromethylphosphonate‐containing diazo and trifluoromethylated ketones assemble to furnish azo‐containing α‐fluorovinylphosphonates. Mechanism studies disclose pathway, which contains an reaction, water addition hydrazone, C−F bond cleavage with reagent as key intermediate. This is conducted at 60 °C affording series α‐fluorovinylphosphonate compounds 42–94% yields Z ‐stereoselectivity. work opens vision for the difluoroalkyl‐substituted diazos, provides strategy synthesis derivatives. magnified image

Язык: Английский

Процитировано

11

Aza-Wittig reaction of (β-diazo-α,α-difluoroethyl)phosphonates with aldehydes for the synthesis of difluoromethylphosphonate-containing arylidene hydrazones DOI Open Access
Qian Wang, Romana Pajkert, Haibo Mei

и другие.

Journal of Fluorine Chemistry, Год журнала: 2023, Номер 273, С. 110226 - 110226

Опубликована: Ноя. 29, 2023

Язык: Английский

Процитировано

2

Catalytic regioselective construction of phenylthio- and phenoxyldifluoroalkyl tetrazoles from difluorodiazoketones DOI

Hong‐Song Shi,

Shuo-Han Li,

Fa‐Guang Zhang

и другие.

Chemical Communications, Год журнала: 2021, Номер 57(100), С. 13744 - 13747

Опубликована: Янв. 1, 2021

Here we report the design and synthesis of two new difluoro-diazoketone reagents (difluorophenylthiol diazoketone difluorophenoxyl diazoketone) their [3+2] cycloaddition reactions with aryldiazonium salts under silver catalysis conditions. This protocol enables regioselective access to a broad scope difluorophenylthiol- difluorophenoxyl-substituted tetrazole-carbinols in one-pot operation. Further synthetic derivatizations including dephenylthiolation unexpected phenylthiol group migration/fluorination allow efficient preparation α-difluoromethyl α-trifluoromethyl tetrazole-thioethers.

Язык: Английский

Процитировано

4