Unraveling the Protective Role of Oleocanthal and Its Oxidation Product, Oleocanthalic Acid, against Neuroinflammation DOI Creative Commons
Maria Cristina Barbalace, Michela Freschi, Irene Rinaldi

и другие.

Antioxidants, Год журнала: 2024, Номер 13(9), С. 1074 - 1074

Опубликована: Сен. 3, 2024

Neuroinflammation is a critical aspect of various neurodegenerative diseases, such as Alzheimer's and Parkinson's diseases. This study investigates the anti-neuroinflammatory properties oleocanthal its oxidation product, oleocanthalic acid, using BV-2 cell line activated with lipopolysaccharide. Our findings revealed that significantly inhibited production pro-inflammatory cytokines reduced expression inflammatory genes, counteracted oxidative stress induced by lipopolysaccharide, increased phagocytic activity. Conversely, acid was not able to counteract lipopolysaccharide-induced activation. The docking analysis plausible interaction oleocanthal, both CD14 MD-2 leading potential interference TLR4 signaling. Since our data show only partially reduces activation NF-kB, action antagonist alone cannot explain remarkable effect against neuroinflammation. Proteomic counteracts LPS modulation 31 proteins, including significant targets gelsolin, clathrin, ACOD1, four different isoforms 14-3-3 protein, indicating new molecular compound. In conclusion, but mitigates neuroinflammation through multiple mechanisms, highlighting pleiotropic particularly important in context neurodegeneration.

Язык: Английский

Modulating Neuroinflammation as a Prospective Therapeutic Target in Alzheimer’s Disease DOI Creative Commons

Eunshil Lee,

Yongmin Chang

Cells, Год журнала: 2025, Номер 14(3), С. 168 - 168

Опубликована: Янв. 22, 2025

The recent approval of lecanemab highlights that the amyloid beta (Aβ) protein is an important pathological target in Alzheimer’s disease (AD) and further emphasizes significance neuroinflammatory pathways regulating Aβ accumulation. Indeed, accumulation triggers microglia activation, which are key mediators neuroinflammation. inflammatory responses this process can lead to neuronal damage functional decline. Microglia secrete proinflammatory cytokines accelerate death release anti-inflammatory growth factors contributing recovery protection. Thus, play a dual role neurodegeneration neuroprotection, complicating their function AD. Therefore, elucidating complex interactions between protein, microglia, neuroinflammation essential for developing new strategies treating This review investigates receptors involved activating aims enhance understanding how these processes impact AD, as well they be regulated. also analyzed studies reported existing literature ongoing clinical trials. Overall, will contribute regulatory mechanisms therapies slow progression

Язык: Английский

Процитировано

1

Unraveling the Protective Role of Oleocanthal and Its Oxidation Product, Oleocanthalic Acid, against Neuroinflammation DOI Creative Commons
Maria Cristina Barbalace, Michela Freschi, Irene Rinaldi

и другие.

Antioxidants, Год журнала: 2024, Номер 13(9), С. 1074 - 1074

Опубликована: Сен. 3, 2024

Neuroinflammation is a critical aspect of various neurodegenerative diseases, such as Alzheimer's and Parkinson's diseases. This study investigates the anti-neuroinflammatory properties oleocanthal its oxidation product, oleocanthalic acid, using BV-2 cell line activated with lipopolysaccharide. Our findings revealed that significantly inhibited production pro-inflammatory cytokines reduced expression inflammatory genes, counteracted oxidative stress induced by lipopolysaccharide, increased phagocytic activity. Conversely, acid was not able to counteract lipopolysaccharide-induced activation. The docking analysis plausible interaction oleocanthal, both CD14 MD-2 leading potential interference TLR4 signaling. Since our data show only partially reduces activation NF-kB, action antagonist alone cannot explain remarkable effect against neuroinflammation. Proteomic counteracts LPS modulation 31 proteins, including significant targets gelsolin, clathrin, ACOD1, four different isoforms 14-3-3 protein, indicating new molecular compound. In conclusion, but mitigates neuroinflammation through multiple mechanisms, highlighting pleiotropic particularly important in context neurodegeneration.

Язык: Английский

Процитировано

2