Synthesis of spiroindolenines through a one-pot multistep process mediated by visible light DOI Creative Commons

Francesco Gambuti,

Jacopo Pizzorno,

Chiara Lambruschini

и другие.

Beilstein Journal of Organic Chemistry, Год журнала: 2024, Номер 20, С. 2722 - 2731

Опубликована: Окт. 29, 2024

Spiro-heterocyclic indolenines are privileged scaffolds widely present in numerous indole alkaloids. Here, we develop a novel approach for the one-pot multistep synthesis of different spiro[indole-isoquinolines]. The protocol proposed involves visible light mediated oxidation N -aryl tertiary amines using bromochloroform with generation reactive iminium species, which reacts an isocyanide and electron-rich aniline three-component Ugi-type reaction to give α-aminoamidine. This compound might undergo additional light-mediated furnish second intermediate, acts as electrophile intramolecular electrophilic aromatic substitution giving final spiro-indolenine. scope process has been investigated respect all three components. Simple operations, mild conditions, good yields make this strategy convenient sustainable way obtain spiro-indolenine derivatives.

Язык: Английский

Advances in gold catalyzed synthesis of quinoid heteroaryls DOI Creative Commons
Adnan Majeed, Ayesha Zafar,

Zanira Mushtaq

и другие.

RSC Advances, Год журнала: 2024, Номер 14(29), С. 21047 - 21064

Опубликована: Янв. 1, 2024

Synthesis of quinoid heteroaryls via gold-catalyzed cascade protocols: recent advances and methodologies.

Язык: Английский

Процитировано

8

Fluorination of α-Imino Gold Carbenes to Access C3-Fluorinated Aza-Heterocycles DOI
Shashank P. Sancheti, Dibya Jyoti Mondal, Nitin T. Patil

и другие.

ACS Catalysis, Год журнала: 2023, Номер 13(7), С. 4391 - 4397

Опубликована: Март 16, 2023

Reported herein is the fluorination of α-imino gold carbenes, generated in situ from azidoalkynes, to access substituted C3-fluorinated quinolones and indoles. The methodology has been applied for synthesizing quinolone- quinoline-based natural products, including pseudanes (4 representative examples), chimanine A, graveolinine. Mechanistic investigations, NMR SC-XRD analysis, reveal that NEt3·3HF reacts with catalyst generate a phosphine-ligated fluoride-bridged binuclear complex which then generates active this reaction.

Язык: Английский

Процитировано

10

Construction of the quinobenzoxazine coreviagold-catalyzed dual annulation of azide-tethered alkynones with anthranils DOI
Swapnil V. Halnor, Pawan S. Dhote, Chepuri V. Ramana

и другие.

Organic & Biomolecular Chemistry, Год журнала: 2023, Номер 21(10), С. 2127 - 2137

Опубликована: Янв. 1, 2023

A new catalytic method for the construction of quinobenzoxazine core has been developed employing gold-catalyzed cyclization o-azidoacetylenic ketones in presence anthranils. The overall process comprises a 6-endo-dig cyclisation ketone leading to α-imino gold carbene and subsequent transfer anthranil 3-aryl-imino-quinoline-4-one intermediate, which undergoes 6π-electrocyclization aromatization form central core. This transformation provides approach diverse array structures, addition being scalable having mild reaction conditions.

Язык: Английский

Процитировано

4

Synthesis of acridinesviacopper-catalyzed amination/annulation cascades between arylboronic acids and anthranils DOI
Yuge Li, Liang Xu, Yu Wei

и другие.

Organic & Biomolecular Chemistry, Год журнала: 2022, Номер 20(48), С. 9742 - 9745

Опубликована: Янв. 1, 2022

The direct conversion of aryl boronic acids and anthranils to acridines has been realized herein, via the catalysis copper species under acidic conditions.

Язык: Английский

Процитировано

4

Synthesis, characterization, and crystal structure of 2-(2-azidophenyl)-3-oxo-3H-indole 1-oxide DOI Creative Commons
Pawan S. Dhote, Srinu Tothadi, Chepuri V. Ramana

и другие.

Acta Crystallographica Section E Crystallographic Communications, Год журнала: 2024, Номер 80(3), С. 310 - 313

Опубликована: Фев. 20, 2024

An attempt to explore the reactivity of nitro group in presence gold catalysis comparison azide yielded intriguing results. Surprisingly, only exhibited reactivity, ultimately giving rise formation title isatogen, C 14 H 8 N 4 O 2 . In crystal structure, weak C—H...O hydrogen bonds and π–π stacking interactions link molecules. The structure exhibits disorder molecule.

Язык: Английский

Процитировано

0

Synthesis of spiroindolenines through a one-pot multistep process mediated by visible light DOI Creative Commons

Francesco Gambuti,

Jacopo Pizzorno,

Chiara Lambruschini

и другие.

Beilstein Journal of Organic Chemistry, Год журнала: 2024, Номер 20, С. 2722 - 2731

Опубликована: Окт. 29, 2024

Spiro-heterocyclic indolenines are privileged scaffolds widely present in numerous indole alkaloids. Here, we develop a novel approach for the one-pot multistep synthesis of different spiro[indole-isoquinolines]. The protocol proposed involves visible light mediated oxidation N -aryl tertiary amines using bromochloroform with generation reactive iminium species, which reacts an isocyanide and electron-rich aniline three-component Ugi-type reaction to give α-aminoamidine. This compound might undergo additional light-mediated furnish second intermediate, acts as electrophile intramolecular electrophilic aromatic substitution giving final spiro-indolenine. scope process has been investigated respect all three components. Simple operations, mild conditions, good yields make this strategy convenient sustainable way obtain spiro-indolenine derivatives.

Язык: Английский

Процитировано

0