Development of a Highly Efficient NIR-II Phototherapeutic Agent for Fluorescence Imaging-Guided Synergistic PTT/PDT/Chemotherapy of Colorectal Cancer DOI
Ji Liu, Lei Liang,

Ping Gan

и другие.

Journal of Medicinal Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Апрель 1, 2025

NIR-II-triggered phototherapy presents a noninvasive, resistance-free alternative therapeutic approach with deeper tissue penetration and improved imaging of deep tumors. However, many NIR-II phototherapeutic agents suffer from low fluorescence quantum yields, poor photothermal conversion efficiency (PCE), reduced efficacy due to the upregulation heat shock protein HSP70. This study develops small-molecule agent (IRF) high yield (17.4%), excellent PCE (96.8%) for therapy (PTT), photodynamic (PDT) activity. To decrease thermal resistance during phototherapy, IRF evodiamine (EVO) were loaded onto hyaluronic acid (HA)-modified nanoparticles, creating multifunctional nanoplatform termed EVO/IRF@HA NPs. NPs can actively target tumors via HA moiety. Upon 980 nm laser irradiation, increases temperature content reactive oxygen species synergistic PTT/PDT. Importantly, EVO effectively inhibits overexpression HSP70, enabling combined PTT/PDT/chemotherapy effective colorectal cancer (CRC) treatment.

Язык: Английский

Electrostatic Co‐Assembly of Cyanine Pair for Augmented Photoacoustic Imaging and Photothermal Therapy DOI Creative Commons

Haiqiao Huang,

Yingnan Wu,

Xin He

и другие.

Advanced Science, Год журнала: 2025, Номер unknown

Опубликована: Фев. 14, 2025

Abstract Molecular phototheranostic dyes are of eminent interest for oncological diagnosis and imaging‐guided phototherapy. However, it remains challenging to develop photosensitizers (PSs) that simultaneously integrate high‐contrast photoacoustic imaging efficient therapeutic capabilities. In this work, a supramolecular strategy is employed construct molecular pair agent via the direct self‐assembly two cyanines, C5TNa (anionic) Cy‐Et (cationic). The Coulombic interactions between facilitate formation complementary cyanine (C5T‐ET) creation CT‐J‐type aggregates in water. This results completely quenched fluorescence significantly enhances nonradiative deactivation (≈22 ps), leading 3.3‐fold increase photothermal conversion efficiency 7.1‐fold enhancement response compared indocyanine green (ICG). As result, J‐type aggregate demonstrates high capability remarkable antitumor efficacy vivo, highlighting its potential clinical applications. work provides strong experimental evidence superior performance enhancing photosensitization response. It believed will propel advancement controllable dye J‐aggregates contribute practical implementation phototherapy vivo.

Язык: Английский

Процитировано

1

Structure–Activity Relationship of Hemicyanine Molecules: Mitochondrion-Targeting Hemicyanine Fluorescent Molecular Probes for HSO3 Recognition and Near-Infrared Image-Guided Photothermal/Photodynamic Synergetic Therapy DOI
Lu Zhang, Ke Yan,

Shuang Min

и другие.

The Journal of Physical Chemistry Letters, Год журнала: 2025, Номер unknown, С. 1746 - 1752

Опубликована: Фев. 10, 2025

Hemicyanine molecules have unparalleled potential in the fields of fluorescence sensing, bioimaging, and disease therapeutics due to their excellent optical properties, cell penetration, mitochondrial targeting, photosensitivity. Herein, three dual-cation hemicyanine molecular probes named DCy, PDCy, TDCy were developed. All them could detect HSO3-, PDCy recognize HSO3- under 365 nm ultraviolet light or sunlight. In addition, is a multifunctional molecule, which has following advantages: simple synthesis, red near-infrared dual-channel imaging, photothermal/photodynamic synergistic therapy capabilities. Upon analysis correlation between structures recognition, photosensitivity, photothermal activity, cytotoxicity, structure-activity relationship be summarized, provide guidance for subsequent research development.

Язык: Английский

Процитировано

0

Tuning the Near-Infrared J-Aggregate of a Multicationic Photosensitizer through Molecular Coassembly for Symbiotic Photothermal Therapy and Chemotherapy DOI
Zhenyan He, Yuting Gao, Zhen Huang

и другие.

ACS Nano, Год журнала: 2025, Номер unknown

Опубликована: Март 7, 2025

Cationic photosensitizers (PSs) offer many intriguing advantages, in addition to generating heat or reactive oxygen species for cancer phototherapy. However, the preparation of cationic PSs with enhanced near-infrared (NIR) absorption remains a significant challenge. In this work, we have synthesized PS TPBBT, which incorporates strong electron-withdrawing unit, benzobisthiadiazole, and four terminal pyridinium groups. It self-assembles into mixed H/J aggregated state maximal peak at 620 nm but coassembles negatively charged planar small molecules form sole J-aggregates. Following strategy, coassemble TPBBT rhein, planar, anionic traditional Chinese medicine an anticancer activity, allows near 100 bathochromic shift improves photothermal conversion efficiency (PCE) from 6.4 60.4% under 808 laser irradiation. Additionally, coassembling significantly enhances cellular uptake rhein through effect. The coassembly (TPBBTein) can completely eliminate 4T1 tumors on mouse models, validating that facile strategy not only tune NIR J-aggregate molecular also promotes efficient, symbiotic combination therapy chemotherapy.

Язык: Английский

Процитировано

0

In-situ injectable hydrogel for near-infrared-regulated hyperthermic perfusion therapy of triple-negative breast cancer DOI
Lijie Zhai, Linwei Li, Tao Liao

и другие.

Journal of Colloid and Interface Science, Год журнала: 2025, Номер unknown

Опубликована: Март 1, 2025

Язык: Английский

Процитировано

0

Development of a Highly Efficient NIR-II Phototherapeutic Agent for Fluorescence Imaging-Guided Synergistic PTT/PDT/Chemotherapy of Colorectal Cancer DOI
Ji Liu, Lei Liang,

Ping Gan

и другие.

Journal of Medicinal Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Апрель 1, 2025

NIR-II-triggered phototherapy presents a noninvasive, resistance-free alternative therapeutic approach with deeper tissue penetration and improved imaging of deep tumors. However, many NIR-II phototherapeutic agents suffer from low fluorescence quantum yields, poor photothermal conversion efficiency (PCE), reduced efficacy due to the upregulation heat shock protein HSP70. This study develops small-molecule agent (IRF) high yield (17.4%), excellent PCE (96.8%) for therapy (PTT), photodynamic (PDT) activity. To decrease thermal resistance during phototherapy, IRF evodiamine (EVO) were loaded onto hyaluronic acid (HA)-modified nanoparticles, creating multifunctional nanoplatform termed EVO/IRF@HA NPs. NPs can actively target tumors via HA moiety. Upon 980 nm laser irradiation, increases temperature content reactive oxygen species synergistic PTT/PDT. Importantly, EVO effectively inhibits overexpression HSP70, enabling combined PTT/PDT/chemotherapy effective colorectal cancer (CRC) treatment.

Язык: Английский

Процитировано

0