N-Unsubstituted 1,2-benzothiazine 1,1-dioxides: Pd-catalyzed one-pot sonochemical access and in silico / in vitro evaluation against MtbCM DOI

Narender Addu,

Hinuja Miriyala,

Ravikumar Kapavarapu

и другие.

Journal of Molecular Structure, Год журнала: 2023, Номер 1301, С. 137345 - 137345

Опубликована: Дек. 20, 2023

Язык: Английский

Convergent Synthesis of 2-Oxazolone-4-carboxylates Esters by Reaction of Aldehydes with Ambivalent N-Cbz-α-Tosylglycinate Ester DOI
Masahiro Abe, Baptiste Picard, Michaël De Paolis

и другие.

Organic Letters, Год журнала: 2020, Номер 22(12), С. 4864 - 4867

Опубликована: Июнь 10, 2020

N-Cbz-α-tosylglycinate ester was combined with aldehydes in a redox-neutral sequence leading to 2-oxazolone-4-carboxylates high functional group tolerance. While the scope of method delineated primary and secondary aliphatic as well aromatics, no racemization occurred chiral such Garner's. Hitherto unknown, this process relies on ambivalent role acting pronucleophile.

Язык: Английский

Процитировано

1
N-Unsubstituted 1,2-benzothiazine 1,1-dioxides: Pd-catalyzed one-pot sonochemical access and in silico / in vitro evaluation against MtbCM DOI

Narender Addu,

Hinuja Miriyala,

Ravikumar Kapavarapu

и другие.

Journal of Molecular Structure, Год журнала: 2023, Номер 1301, С. 137345 - 137345

Опубликована: Дек. 20, 2023

Язык: Английский

Процитировано

0