Anticancer Ribosomally Synthesized and Post-Translationally Modified Peptides from Plants: Structures, Therapeutic Potential, and Future Directions DOI Creative Commons
Hye Jin Hwang,

Youngsang Nam,

Chanhee Jang

и другие.

Current Issues in Molecular Biology, Год журнала: 2024, Номер 47(1), С. 6 - 6

Опубликована: Дек. 26, 2024

Cancer remains a significant medical challenge, necessitating the discovery of novel therapeutic agents. Ribosomally synthesized and post-translationally modified peptides (RiPPs) from plants have emerged as promising source anticancer compounds, offering unique structural diversity potent biological activity. This review identifies discusses cytotoxic RiPPs across various plant families, focusing on their absolute chemical structures reported activities against cancer cell lines. Notably, plant-derived such rubipodanin A mallotumides A-C demonstrated low nanomolar IC50 values multiple types, highlighting potential. By integrating traditional ethnobotanical knowledge with modern genomic bioinformatic approaches, this study underscores importance resource for developing innovative treatments. These findings pave way further exploration RiPPs, emphasizing role in addressing ongoing challenges oncology enhancing repertoire effective therapies.

Язык: Английский

Review of plants as a promising source of bioactive peptides for the treatment of diabetes DOI
Quratulain Maqsood, Tahir Mehmood,

Fareeha Nadeem

и другие.

CABI Reviews, Год журнала: 2025, Номер unknown

Опубликована: Март 17, 2025

Abstract The bioactive compounds found in plants offer numerous therapeutic properties through protein and peptide molecules. occurrence of diabetes has developed into a significant worldwide healthcare crisis because this metabolic disease continues to affect millions individuals throughout the world while growing numbers annually. uncontrolled nature produces serious complications which include microangiopathy together with ketoacidosis followed by cardiovascular diseases. Drugs used treatment exist yet their marketplace costs combined side effects make researchers seek new techniques. use peptides extracted from attracts they show proven ability regulate diabetes-related pathways insulin sensitivity enhancement blood glucose control along weight management activities, anti-inflammatory processes, antioxidant properties. This review investigates plant-derived antidiabetic potential detailed research on biological mechanisms. current developments screening process, uses killing methods.

Язык: Английский

Процитировано

0

The emergence and loss of cyclic peptides in Nicotiana illuminate dynamics and mechanisms of plant metabolic evolution DOI Creative Commons

Elliot M. Suh,

Jakob K. Reinhardt, Jing‐Ke Weng

и другие.

Proceedings of the National Academy of Sciences, Год журнала: 2025, Номер 122(16)

Опубликована: Апрель 14, 2025

Specialized metabolism plays a central role in how plants cope with both biotic and abiotic stresses order to survive reproduce within dynamic challenging environments. One recently described class of plant-specific, ribosomally synthesized, posttranslationally modified peptides are the burpitides, which characterized by installation distinct sidechain macrocycles enzymes known as burpitide cyclases. While they found across many plant families exhibit diverse bioactivities, little is about their evolution or new variants arise. Here, we present identification cyclase, resurrected from defunct pseudogene model organism Nicotiana attenuata , coyote tobacco. By repairing ΨNatBURP2 expressing it heterologously benthamiana successfully reconstituted its original enzymatic activity. As an autocatalytic peptide installs unique C–C bond between tyrosine side chain specific backbone α-carbon heptapeptide core motif, resulting burpitides dubbed “nanamins.” Despite pseudogenization N. that closely related species, clevelandii retains wild-type gene produces nanamins. Phylogenetic analyses targeted mutagenesis experiments reveal this chemotype must have evolved duplication neofunctionalization more promiscuous ancestral gene. This work highlights novel chemotypes may rapidly emerge disappear plants, while expanding molecular toolkit for engineering applications agriculture drug discovery.

Язык: Английский

Процитировано

0

The emergence and loss of cyclic peptides in Nicotiana illuminate dynamics and mechanisms of plant metabolic evolution DOI Open Access

Elliot M. Suh,

Jakob K. Reinhardt, Jing‐Ke Weng

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2024, Номер unknown

Опубликована: Дек. 1, 2024

Specialized metabolism plays a central role in how plants cope with both biotic and abiotic stresses order to survive reproduce within dynamic challenging environments. One recently circumscribed class of plant-specific, ribosomally synthesized post-translationally modified peptides are the burpitides, which characterized by installation distinct sidechain macrocycles enzymes known as burpitide cyclases. While they found across many plant families exhibit diverse bioactivities, little is about their evolution or new variants arise. Here we present discovery cyclase, resurrected from defunct pseudogene model organism Nicotiana attenuata, coyote tobacco. By repairing ΨNatBURP2 expressing it heterologously benthamiana, successfully reconstituted its original enzymatic activity. As an autocatalytic peptide installs unique C-C bond between tyrosine side chain specific backbone a-carbon heptapeptide core motif, resulting dubbed "nanamin." Despite pseudogenization N. that closely related species, clevelandii, retains wild-type gene produces nanamins. Phylogenetic analyses targeted mutagenesis experiments reveal this chemotype must have evolved duplication neofunctionalization more promiscuous ancestral gene. This work highlights novel chemotypes may rapidly emerge disappear plants, while expanding molecular toolkit for engineering applications agriculture drug discovery.

Язык: Английский

Процитировано

0

Anticancer Ribosomally Synthesized and Post-Translationally Modified Peptides from Plants: Structures, Therapeutic Potential, and Future Directions DOI Creative Commons
Hye Jin Hwang,

Youngsang Nam,

Chanhee Jang

и другие.

Current Issues in Molecular Biology, Год журнала: 2024, Номер 47(1), С. 6 - 6

Опубликована: Дек. 26, 2024

Cancer remains a significant medical challenge, necessitating the discovery of novel therapeutic agents. Ribosomally synthesized and post-translationally modified peptides (RiPPs) from plants have emerged as promising source anticancer compounds, offering unique structural diversity potent biological activity. This review identifies discusses cytotoxic RiPPs across various plant families, focusing on their absolute chemical structures reported activities against cancer cell lines. Notably, plant-derived such rubipodanin A mallotumides A-C demonstrated low nanomolar IC50 values multiple types, highlighting potential. By integrating traditional ethnobotanical knowledge with modern genomic bioinformatic approaches, this study underscores importance resource for developing innovative treatments. These findings pave way further exploration RiPPs, emphasizing role in addressing ongoing challenges oncology enhancing repertoire effective therapies.

Язык: Английский

Процитировано

0