Organic Letters, Год журнала: 2025, Номер unknown
Опубликована: Фев. 20, 2025
The trifluoroethoxy group (OCH2CF3) is a valuable motif prevalent in pharmaceuticals and agrichemicals. Herein, we present simple radical trifluoroethoxylation method that enables nondirected functionalization of C-H bonds broad array substrates, providing access to (hetero)aryl trifluoroethyl ethers. current protocol tolerates variety synthetically pharmacologically relevant functional groups. Applicability also demonstrated through the late-stage biorelevant molecules marketing drugs.
Язык: Английский