Therapeutic Significance of NLRP3 Inflammasome in Cancer: Friend or Foe? DOI Open Access
Aliea M. Jalali, Keith Mitchell, Christian Pompoco

и другие.

International Journal of Molecular Sciences, Год журнала: 2024, Номер 25(24), С. 13689 - 13689

Опубликована: Дек. 21, 2024

Besides various infectious and inflammatory complications, recent studies also indicated the significance of NLRP3 inflammasome in cancer progression therapy. NLRP3-mediated immune response pyroptosis could be helpful or harmful cancer, depend on nature tumor microenvironment. The activation increase surveillance efficacy immunotherapy. It can lead to removal cells by recruitment phagocytic macrophages, T-lymphocytes, other site. On hand, harmful, as chronic inflammation driven supports creating an environment that facilitates cell proliferation, migration, invasion, metastasis. release pro-inflammatory cytokines such IL-1β IL-18 promote growth angiogenesis, while sustained may suppression, hindering effective anti-tumor responses. In this review article, we discuss role inflammasome-mediated pathophysiology types; understanding is essential for development innovative therapeutic strategies spread.

Язык: Английский

Liquid Biopsy in Cancer Management: Integrating Diagnostics and Clinical Applications DOI Creative Commons

Shashwat Pandey,

Preeti Kumari Yadav

Practical Laboratory Medicine, Год журнала: 2024, Номер unknown, С. e00446 - e00446

Опубликована: Дек. 1, 2024

Liquid biopsy is an innovative, minimally invasive diagnostic tool revolutionizing cancer management by enabling the detection and analysis of cancer-related biomarkers from bodily fluids such as blood, urine, or cerebrospinal fluid. Unlike traditional tissue biopsies, which require procedures, liquid offers a more accessible repeatable method for tracking progression, detecting early-stage cancers, monitoring therapeutic responses. The technology primarily focuses on analyzing circulating tumor cells (CTCs), DNA (ctDNA), other cancer-derived genetic materials. These provide critical information heterogeneity, mutation profiles, potential drug resistance. In clinical practice, has demonstrated its utility in identifying actionable mutations, guiding personalized treatment strategies, assessing minimal residual disease (MRD). While holds immense promise, challenges related to sensitivity, specificity, standardization remain. Efforts optimize pre-analytical analytical processes, along with establishment robust regulatory frameworks, are crucial widespread adoption. This abstract highlights transformative diagnosis, prognosis, monitoring, emphasizing role advancing oncology. Further research, trials, harmonization will be vital realizing full precision care.

Язык: Английский

Процитировано

5

An innovative approach to development of new pyrazolylquinolin-2-one hybrids as dual EGFR and BRAFV600E inhibitors DOI Creative Commons

Mohamed M. Hawwas,

Ahmed S. Mancy,

Mohamed Ramadan

и другие.

Molecular Diversity, Год журнала: 2025, Номер unknown

Опубликована: Март 8, 2025

Novel quinoline-based derivatives 2a-e and 4a-j have been designed synthesized as potential antiproliferative agents. The compounds were screened for their activity against sixty cell lines according to NCI protocol. promising hybrids 4d-g are by MTT assays on three cancer lines: leukemia (MOLT-4), lung (HOP-92), breast (T47D), with IC50 values ranging from 4.982 ± 0.2 36.52 1.46 µM compared Staurosporine, compound 4e being the most effective. Derivatives evaluated inhibitory EGFR BRAFV600E. Compound exhibited highest activities, of 0.055 0.002 μM 0.068 0.003 BRAFV600E, reference drugs erlotinib (IC50 0.06 μM) vemurafenib 0.035 0.001 μM), respectively. Cell cycle analysis HOP-92 manifested that pre-G1 apoptosis signaling took place after treatment. Docking simulations employed analyze modes scores respect results revealed strong affinity both BRAFV600E - 3.226 3.474 kcal/mol,

Язык: Английский

Процитировано

0

Oral Melanoma in Older Adults: Epidemiology, Molecular Landscape, and Treatment Strategies DOI
José Alcides Almeida de Arruda, Victor Zanetti Drumond, Jefferson da Rocha Tenório

и другие.

Pigment Cell & Melanoma Research, Год журнала: 2025, Номер 38(3)

Опубликована: Апрель 14, 2025

ABSTRACT Oral melanoma is an aggressive neoplasm arising from melanocytes in the mucosal epithelium, accounting for 0.2%–0.8% of all melanomas. Unlike cutaneous melanoma, it not associated with UV exposure, and its pathogenesis involves complex genetic molecular alterations. This predominantly affects older adults (≥ 60 years). Clinically, lesions often present as macular or nodular exophytic growth pattern, sometimes ulcerated, exhibit varied pigmentation. Diagnosis further complicated by non‐pigmented (amelanotic) variants that can resemble other oral pigmentations. Wide surgical excision remains mainstay treatment, combined chemotherapy; however, recurrence distant metastasis remain high. While immunotherapy has shown promise subtypes, efficacy uncertain. Treatment particularly challenging due to comorbidities treatment‐related morbidity. review summarizes epidemiology, clinical features, current treatment strategies adults. Key advances mechanisms underlying this are also outlined. As a strategic approach, integrating screening into routine geriatric dental care, supported diagnostic algorithms, may improve early detection, prognosis, survival outcomes vulnerable population.

Язык: Английский

Процитировано

0

In Silico Analysis of Novel circRNA‐miRNA‐mRNA Axis in BRAFV600E Melanoma: Implications for Primary to Metastasis Transformation and TIME Modulation DOI
Himanshu Naik, Rajat Choudhary, V. Badireenath Konkimalla

и другие.

The Journal of Gene Medicine, Год журнала: 2025, Номер 27(6)

Опубликована: Май 28, 2025

ABSTRACT Background The BRAF V600E mutation drives metastatic transition by altering the tumor immune microenvironment (TIME) through transcriptional and post‐transcriptional regulation. Recent studies identify circular RNA (circRNA) micro‐RNA (miRNA) as key regulators in melanoma. This study uses silico analysis to explore circRNA‐miRNA‐mRNA axis melanoma progression. Methods We analyzed primary ( n = 42) 89) samples from TCGA (SKCM), including their status, markers both types explored association with cells within TIME. regulatory were verified using ROC curve analysis, IHC data HPA database, an external dataset. Further, was established Cytoscape. Results Our comprehensive identifies SYK, HMOX1, IL33, CFH, FGF1, COL8A1, ADAMTS3 gene signatures, while VCAM‐1 SNAI2 dominate prominent associated subtype. Among infiltrating group, macrophages M1 M2, CD8 + T‐cells, T regs show a positive correlation significant infiltration screened miRNA targets sponges, built network involving two circRNAs (hsa‐circ‐0011617 hsa‐circ‐0011623) three miRNAs (hsa‐miR‐1246, hsa‐miR‐346, hsa‐miR‐1197) connected identified signature. Conclusion Overall, our reveals that might have potential role metastasis BRAF‐mutated TIME via circRNA–miRNA–mRNA axis.

Язык: Английский

Процитировано

0

Withaferin-A induced Vimentin S56 phosphorylation dissociates NEDD9 signaling loop to regress progressive metastatic melanoma into lung adenocarcinoma. DOI

Ankith Sherapura,

Bayram Kıran,

G.S. Pavan Kumar

и другие.

Chemico-Biological Interactions, Год журнала: 2024, Номер unknown, С. 111319 - 111319

Опубликована: Ноя. 1, 2024

Язык: Английский

Процитировано

1

Prognostic Role of Clinicopathological Characteristics and Serum Markers in Metastatic Melanoma Patients Treated with BRAF and MEK Inhibitors DOI Open Access
Eszter Anna Janka, Imre Szabó,

Sándor Kollár

и другие.

Cancers, Год журнала: 2024, Номер 16(17), С. 2981 - 2981

Опубликована: Авг. 27, 2024

Prognostic studies can provide important information about disease biology and improve the use of biomarkers to optimize treatment decisions.

Язык: Английский

Процитировано

0

Therapeutic Significance of NLRP3 Inflammasome in Cancer: Friend or Foe? DOI Open Access
Aliea M. Jalali, Keith Mitchell, Christian Pompoco

и другие.

International Journal of Molecular Sciences, Год журнала: 2024, Номер 25(24), С. 13689 - 13689

Опубликована: Дек. 21, 2024

Besides various infectious and inflammatory complications, recent studies also indicated the significance of NLRP3 inflammasome in cancer progression therapy. NLRP3-mediated immune response pyroptosis could be helpful or harmful cancer, depend on nature tumor microenvironment. The activation increase surveillance efficacy immunotherapy. It can lead to removal cells by recruitment phagocytic macrophages, T-lymphocytes, other site. On hand, harmful, as chronic inflammation driven supports creating an environment that facilitates cell proliferation, migration, invasion, metastasis. release pro-inflammatory cytokines such IL-1β IL-18 promote growth angiogenesis, while sustained may suppression, hindering effective anti-tumor responses. In this review article, we discuss role inflammasome-mediated pathophysiology types; understanding is essential for development innovative therapeutic strategies spread.

Язык: Английский

Процитировано

0