Formulation of Felodipine lipid nanoparticle-loaded oral fast-dissolving films DOI

Suparna Anand Naik,

Cleona Elizabeth Mary DCruz,

Lalit Kumar

и другие.

Tenside Surfactants Detergents, Год журнала: 2024, Номер 61(6), С. 568 - 583

Опубликована: Окт. 8, 2024

Abstract Felodipine, a calcium channel blocker used to treat hypertension, is BCS Class II drug characterized by low solubility, high permeability and significant hepatic metabolism, which limits its bioavailability 15 %. This study focuses on improving the of Felodipine developing oral fast-dissolving films (OFDFs) incorporating lipid nanoparticles. loaded nanoparticles were prepared using glyceryl monooleate (GMO) as Poloxamer 407 surfactant, then incorporated into OFDFs solvent casting technique. A Box-Behnken design with Design Expert Stat-Ease ® 360 was evaluate impact GMO, concentration, sonication time particle size entrapment efficiency. The resulting nanoparticle dispersions had sizes ranging from 74.92 nm 112.1 efficiencies between 80.43 % 95.23 Differential scanning calorimetry (DSC), Fourier transform infrared spectroscopy (FTIR), X-ray diffraction (XRD) confirmed successful encapsulation. OFDF showed optimal mechanical properties, disintegration within (41.33 ± 3.51) s, an in-vitro release (89.82 2.75) in 6 min. Scanning electron microscopy (SEM) revealed smooth, uniform, porous surface remained stable for three months. concludes that improve permeability, dissolution, onset action, making them promising approach antihypertensive therapy.

Язык: Английский

Polymeric nanoparticles as delivery vehicles for targeted delivery of chemotherapy drug fludarabine to treat hematological cancers DOI

Mehrab Pourmadadi,

Hamed Mirzaei Dehaghi,

Amirhossein Ghaemi

и другие.

Inorganic Chemistry Communications, Год журнала: 2024, Номер 167, С. 112819 - 112819

Опубликована: Июль 6, 2024

Язык: Английский

Процитировано

11

Advancing cancer therapy: Unveiling the cutting-edge potential of carmustine nano carriers for targeted treatment DOI

Amirhossein Khanizadeh,

Amirhossein Ghaemi, Mehrab Pourmadadi

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2024, Номер 99, С. 105943 - 105943

Опубликована: Июль 4, 2024

Язык: Английский

Процитировано

6

Understanding the journey of biopolymeric nanoformulations for oral drug delivery: Conventional to advanced treatment approaches DOI
Ameya Sharma,

Nitin Jangra,

Divya Dheer

и другие.

European Polymer Journal, Год журнала: 2024, Номер 218, С. 113338 - 113338

Опубликована: Июль 26, 2024

Язык: Английский

Процитировано

6

Advancements in Nanocarrier-Mediated Sunitinib Delivery: Addressing Obstacles and Revealing its Therapeutic Promise in Oncological Treatment DOI

Mohammad Javad Javid‐Naderi,

Zohreh Abbasi,

Sonia Fathi‐karkan

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2024, Номер 100, С. 106107 - 106107

Опубликована: Авг. 25, 2024

Язык: Английский

Процитировано

2

Advances in polymeric and non-polymeric nanocarriers for the magnified delivery of levofloxacin against bacterial infection DOI Creative Commons

Negar Safaran,

Shohreh Javadi,

Mehrab Pourmadadi

и другие.

Journal of Nanoparticle Research, Год журнала: 2024, Номер 26(8)

Опубликована: Авг. 1, 2024

Abstract This review examines the latest developments in nanoscopic antibiotic formulations used to treat infections caused by bacteria. A wide range of nanocarrier platforms are discussed, including polymer-based nanoparticles (NPs), lipid-based vesicles, mesoporous silica, and other inorganic materials. The levofloxacin (LVF) is predominantly as a model drug given its broad-spectrum activity. Studies this regard have evaluated loading encapsulation efficiency (EE) using analytical techniques such FTIR, DLS, TEM. In vitro release kinetics was characterized through dialysis fluorescence-based assays. Zone inhibition viability studies provided insights into antibacterial efficacy. Some approaches incorporated stimuli-responsive polymers or targeting ligands facilitate controlled targeted release. Overall, nanocarriers demonstrated potential for sustained levels, reduced dosing, improved treatment biofilms intracellular compared free administration. offers comprehensive analysis promising field with implications combating resistance.

Язык: Английский

Процитировано

1

Revolutionizing Cancer Treatment: Exploring the Latest Breakthroughs in Bicalutamide Delivery and Co-Delivery Nanoformulations for Cancer Therapy DOI
Mehrab Pourmadadi,

Nazanin Askari,

Amirhossein Ghaemi

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2024, Номер unknown, С. 106201 - 106201

Опубликована: Сен. 1, 2024

Язык: Английский

Процитировано

0

Formulation of Felodipine lipid nanoparticle-loaded oral fast-dissolving films DOI

Suparna Anand Naik,

Cleona Elizabeth Mary DCruz,

Lalit Kumar

и другие.

Tenside Surfactants Detergents, Год журнала: 2024, Номер 61(6), С. 568 - 583

Опубликована: Окт. 8, 2024

Abstract Felodipine, a calcium channel blocker used to treat hypertension, is BCS Class II drug characterized by low solubility, high permeability and significant hepatic metabolism, which limits its bioavailability 15 %. This study focuses on improving the of Felodipine developing oral fast-dissolving films (OFDFs) incorporating lipid nanoparticles. loaded nanoparticles were prepared using glyceryl monooleate (GMO) as Poloxamer 407 surfactant, then incorporated into OFDFs solvent casting technique. A Box-Behnken design with Design Expert Stat-Ease ® 360 was evaluate impact GMO, concentration, sonication time particle size entrapment efficiency. The resulting nanoparticle dispersions had sizes ranging from 74.92 nm 112.1 efficiencies between 80.43 % 95.23 Differential scanning calorimetry (DSC), Fourier transform infrared spectroscopy (FTIR), X-ray diffraction (XRD) confirmed successful encapsulation. OFDF showed optimal mechanical properties, disintegration within (41.33 ± 3.51) s, an in-vitro release (89.82 2.75) in 6 min. Scanning electron microscopy (SEM) revealed smooth, uniform, porous surface remained stable for three months. concludes that improve permeability, dissolution, onset action, making them promising approach antihypertensive therapy.

Язык: Английский

Процитировано

0