Synthesis of Sulfo(xo)nium Diacylmethylides DOI

Duo Fu,

Jiaxi Xu

European Journal of Organic Chemistry, Год журнала: 2024, Номер 27(27)

Опубликована: Апрель 29, 2024

Abstract Sulfo(xo)nium diacylmethylides (sulfur ylides) are simple, stable, readily prepared, and versatile synthons. Compared with the sulfo(xo)nium monoacylmethylides, they can be compatible more rigorous reaction conditions showcase unique characteristics due to their excellent stability. This concept article provides an account for syntheses of diacylmethylides, including utilization active methylene compounds, carbene precursors, electron‐deficient alkynes as substrates, discussions on substrate scopes, proposed mechanisms, selected product examples, applications. Challenges further exploration prospect in future also suggested.

Язык: Английский

Photoredox/Sulfide Dual Catalysis for Modular Synthesis of Multi‐Substituted Furan Rings via Catalytic Indirect Reductive Quenching DOI Open Access
Kakeru Matsukuma, Masanori Tayu,

Takumi Ogino

и другие.

Chemistry - An Asian Journal, Год журнала: 2025, Номер unknown

Опубликована: Янв. 7, 2025

The catalytic indirect reductive quenching method is facilitated by a combination of Ir(III) photoredox and sulfide dual-catalysis system. This study demonstrated for synthesizing multi-substituted furans using photoredox/sulfide enables the synthesis various furan derivatives, including spirofurans phthalans. utility this system was through gram-scale pharmaceutical molecule talopram. Mechanistic studies density functional theory calculations suggested formation sulfonium species via radical cations, followed intramolecular cyclization to produce desired derivatives.

Язык: Английский

Процитировано

0

Electrosynthesis of 1,4-diene derivatives bearing cyclopentene skeleton DOI Creative Commons

Yaqi Qiao,

Xiaoqing Fan,

Chengcheng Yuan

и другие.

iScience, Год журнала: 2025, Номер 28(3), С. 111976 - 111976

Опубликована: Фев. 10, 2025

1,n-Dual Π systems including 1,4-diene derivatives have been widely used as the elegant radical receptors to promote cascade additions give highly functionalized polycyclic scaffolds. However, tedious and complicated preparation of former deters broad utilization compromises practical value. Herein, a straightforward was developed from easily accessible alkynes γ,δ-unsaturated carboxylic acids via electrochemical oxidation cyclization Hofmann elimination. This transformation features with good excellent yields, functional group compatibility, selectivity without any Zaitsev elimination product detected.

Язык: Английский

Процитировано

0

Synthesis of Sulfo(xo)nium Diacylmethylides DOI

Duo Fu,

Jiaxi Xu

European Journal of Organic Chemistry, Год журнала: 2024, Номер 27(27)

Опубликована: Апрель 29, 2024

Abstract Sulfo(xo)nium diacylmethylides (sulfur ylides) are simple, stable, readily prepared, and versatile synthons. Compared with the sulfo(xo)nium monoacylmethylides, they can be compatible more rigorous reaction conditions showcase unique characteristics due to their excellent stability. This concept article provides an account for syntheses of diacylmethylides, including utilization active methylene compounds, carbene precursors, electron‐deficient alkynes as substrates, discussions on substrate scopes, proposed mechanisms, selected product examples, applications. Challenges further exploration prospect in future also suggested.

Язык: Английский

Процитировано

1