GABA Type A receptors expressed in triple negative breast cancer cells mediate chloride ion flux DOI Creative Commons

J Bundy,

Yasar Ahmed, Sandra Weller

и другие.

Frontiers in Pharmacology, Год журнала: 2024, Номер 15

Опубликована: Окт. 14, 2024

Triple negative breast cancer (TNBC) is known for its heterogeneous nature and aggressive onset, limited unresponsiveness to hormone therapies immunotherapy as well high likelihood of metastasis recurrence. Since no targeted standard treatment options are available TNBC, novel effective therapeutic targets urgently needed. Ion channels have emerged possible candidates therapy. We previously showed that GABA A β3 subunit expressed at higher levels in TNBC cell lines than non-tumorigenic MCF10A cells. knockdown causes cycle arrest via decreased cyclin D1 increased p21 expression. However, it not if the upregulated R express cell-surface mediate Cl − flux. ions play a role cell-cycle progression other cancers such gastric cancer. Here, using surface biotinylation (N-(Ethoxycarbonylmethyl)-6-Methoxyquinolinium Bromide) MQAE-dye based fluorescence quenching, we show on significantly chloride (Cl ) flux compared Moreover, this mediated can be modulated by pharmacological agents cells with knockdown. Further, bicuculline, antagonist reduced viability Overall, these results point an unexplored TNBC.

Язык: Английский

The epipliancy journey: Tumor initiation at the mercy of identity crisis and epigenetic drift DOI Creative Commons
Rahma Benhassoun,

Anne-Pierre Morel,

Victoria Jacquot

и другие.

Biochimica et Biophysica Acta (BBA) - Reviews on Cancer, Год журнала: 2025, Номер 1880(3), С. 189307 - 189307

Опубликована: Апрель 2, 2025

Cellular pliancy refers to the unique disposition of different stages cellular differentiation transform when exposed specific oncogenic insults. This concept highlights a strong interconnection between identity and tumorigenesis, implies overcoming epigenetic barriers defining states. Emerging evidence suggests that cell-type-specific response intrinsic extrinsic stresses is modulated by accessibility certain areas genome. Understanding interplay mechanisms, differentiation, insults crucial for deciphering complex nature tumorigenesis developing targeted therapies. Hence, relies on dynamic cooperation context through control, including reactivation such as epithelial-to-mesenchymal transition (EMT). Such mechanisms pathways confer plasticity cell allowing it adapt hostile environment in tumor initiation, thus changing its identity. Indeed, growing cancer disease crisis, whereby differentiated cells lose their defined gain progenitor characteristics. The loss fate commitment central feature appears be prerequisite neoplastic transformation. In this context, EMT-inducing transcription factors (EMT-TFs) cooperate with mitogenic oncoproteins foster malignant aberrant activation EMT-TFs plays an active role initiation alleviating key oncosuppressive endowing stem cell-like properties, ability self-renew, course tumorigenesis. highly phenotypic change occurs concomitantly major epigenome reorganization, component regulation. was initially proposed address fundamental question biology: why are some more likely become cancerous events at particular developmental stages? We propose epipliancy, difference configuration leads transformation following insult. Here, we present recent studies furthering our understanding how landscape may impact modulation during early initiation.

Язык: Английский

Процитировано

0

The Clinical Relevance of Epithelial-to-Mesenchymal Transition Hallmarks: A Cut-Off-Based Approach in Healthy and Cancerous Cell Lines DOI Open Access

Maria Cristina Rapanotti,

Elisa Cugini,

Maria Giovanna Scioli

и другие.

International Journal of Molecular Sciences, Год журнала: 2025, Номер 26(8), С. 3617 - 3617

Опубликована: Апрель 11, 2025

The atypical activation of the epithelial-to-mesenchymal transition represents one main mechanisms driving cancer cell dissemination. It enables epithelial cells to detach from primary tumor mass and gain survival advantages in bloodstream, significantly contributing spread circulating cells. Notably, is not a binary process but rather leads formation wide range subpopulations characterized by simultaneous expression both mesenchymal markers. Therefore, analyzing modulation EMT hallmarks during conversion healthy metastatic cells, which acquire stem characteristics, particular interest. This study investigates panel transition-related genes lines, derived various tissues, including lung, colon, pancreas, skin, neuro-ectoderm, with aim identifying potential cut-off values for assessing aggressiveness. Interestingly, we found that levels CDH1, encodes marker E-cadherin, CDH5, encoding vascular endothelial cadherin, transition-transcription factor ZEB1, effectively distinguished Additionally, our data suggest tissue-specific signature markers progression. Overall, results underscore importance investigating as identify most suitable acting indicators disease aggressiveness therapeutic responsiveness.

Язык: Английский

Процитировано

0

Recurring cycles of deprivation of serum and migration in confined spaces augments ganglioside SSEA-4 expression, boosting clonogenicity and cisplatin resistance in TNBC cell line DOI Creative Commons
Zain Nofal, Philipp Malakhov, Маргарита Пустовалова

и другие.

Scientific Reports, Год журнала: 2025, Номер 15(1)

Опубликована: Май 14, 2025

Abstract The remarkable biophysical properties of metastatic migrating cells, such as their exceptional motility and deformability, enable them to migrate through physical confinements created by neighboring cells or extracellular matrix. This study explores the adaptive responses breast cancer (BC) cell sublines derived from highly aggressive, triple-negative MDA-MB-231 non-metastatic MCF7 human BC lines, after undergoing three rounds confined migration (CM) stress. Our findings demonstrate that CM elicits common cell-type specific in sublines. In particular, both exhibit a similar enhancement clonogenicity nanoparticle (NP) uptake activity, indicating tumorigenic potential. We have, for first time, shown stimulation with induces hybrid epithelial-to-mesenchymal transition (EMT) phenotype cells. is characterized significant rise expression stage-specific embryonic antigen-4 (SSEA4), alongside substantial decline population CD133+ marked reduction Ki67 MDA-MB-231-derived subline following Cis-Platin treatment. These changes are likely associated heightened resistance this cisplatin. contrast, far fewer alterations MCF7-derived counterpart notable increase population, which seems be insufficient change susceptibility cisplatin exposure. contributes our understanding mechanisms underlying metastasis drug cancer, emphasizing need personalized approaches treatment consider heterogeneous different subtypes environmental stresses.

Язык: Английский

Процитировано

0

Gene regulatory network transitions reveal the central transcription factors in lung adenocarcinoma progression DOI Creative Commons
Upasana Ray, Ajay P. Singh, Debabrata Samanta

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2025, Номер unknown

Опубликована: Май 14, 2025

Abstract Transcription factors play a central role in cancer growth, progression, and metastasis, contribute to intratumor phenotypic plasticity which enable drug tolerance relapse. Changes the regulatory activities of transcription may not always be detected by investigating mutational signatures or differential expression factor, as done traditional analysis. In addition, past studies have focused on tumors whole thus, fully captured heterogeneity gene regulation among different cell types within tumor microenvironment. this work, through an analysis transitions network architecture dynamics, we identify associated with lung adenocarcinoma progression. The NR2F1 , neurodevelopment dormancy, emerge key factor progression adenocarcinoma. We further that are only active samples uncover how changes dynamics influence heterogeneity. Taken together, our work elucidates during identifies process, reveals complex cooccurring

Язык: Английский

Процитировано

0

Prognostic Significance of Combining Cytokeratin-19, E-Cadherin and Ki-67 Analysis in Triple-Negative Breast Cancer with Basal-Like and Non-Basal-Like Phenotype DOI

Zahra Klayech,

A. Moussa,

Moufida Souid

и другие.

Cancer Investigation, Год журнала: 2024, Номер 42(9), С. 769 - 781

Опубликована: Окт. 20, 2024

Triple-negative breast cancer (TNBC) is known to have the worst outcome compared other forms of cancer. Moreover, molecular markers identified basal-like (BLBC) phenotypes be also related a worse prognosis. In this study, we evaluated by immunohistochemistry (IHC) prognostic significance combining Cytokeratin-19 (CK19), E-cadherin, and Ki-67 tissue expression in triple-negative cases presenting or non-basal-like (n-BLBC) phenotype improve selection monitoring BC patients with more aggressive outcome. Herein, when n-BLBC, BLBC showed positive correlation lymph node metastasis occurrence lower survival rates. Immunohistochemistry analysis revealed significantly E-cadherin prevalence higher both CK19 n-BLBC. Spearman that negatively correlated expressions. BLBC, expressing combined loss was associated relapse-free overall survival. conclusion, TNBC/BLBC simultaneously losing overexpressing are most forms. This could predictive marker poor

Язык: Английский

Процитировано

1

GABA Type A receptors expressed in triple negative breast cancer cells mediate chloride ion flux DOI Creative Commons

J Bundy,

Yasar Ahmed, Sandra Weller

и другие.

Frontiers in Pharmacology, Год журнала: 2024, Номер 15

Опубликована: Окт. 14, 2024

Triple negative breast cancer (TNBC) is known for its heterogeneous nature and aggressive onset, limited unresponsiveness to hormone therapies immunotherapy as well high likelihood of metastasis recurrence. Since no targeted standard treatment options are available TNBC, novel effective therapeutic targets urgently needed. Ion channels have emerged possible candidates therapy. We previously showed that GABA A β3 subunit expressed at higher levels in TNBC cell lines than non-tumorigenic MCF10A cells. knockdown causes cycle arrest via decreased cyclin D1 increased p21 expression. However, it not if the upregulated R express cell-surface mediate Cl − flux. ions play a role cell-cycle progression other cancers such gastric cancer. Here, using surface biotinylation (N-(Ethoxycarbonylmethyl)-6-Methoxyquinolinium Bromide) MQAE-dye based fluorescence quenching, we show on significantly chloride (Cl ) flux compared Moreover, this mediated can be modulated by pharmacological agents cells with knockdown. Further, bicuculline, antagonist reduced viability Overall, these results point an unexplored TNBC.

Язык: Английский

Процитировано

0