Three‐component allylic alkylation reaction of α‐diazo ketones with water and allyl carbonates for construction of homoallylic alcohols DOI

Liping Yin,

Xinyi Zhang,

B. D. Wang

и другие.

Advanced Synthesis & Catalysis, Год журнала: 2024, Номер 366(17), С. 3616 - 3623

Опубликована: Июнь 20, 2024

Abstract A three‐component allylic alkylation reaction of α‐diazo ketones, water and allyl carbonate under the cooperative catalysis Rh 2 (OAc) 4 , Pd (dba) 3 Brønsted acid was disclosed. This method provides an expeditious access to α‐keto homoallylic alcohols in good high yields. Controlled experiments support that transformations proceed through cross‐interception two active intermediates Pd‐allyl species enol derived from oxonium ylides. Moreover, synthetic generated products enable creation motifs enriched with dense functional groups, underscoring their potential as valuable building blocks.

Язык: Английский

Overview of Transition Metal Catalyzed Multicomponent Reactions Based on Trapping of Allylic Electrophiles DOI

Kriti Gupta,

Mahesh Singh Harariya,

Arushi Tyagi

и другие.

ChemCatChem, Год журнала: 2024, Номер 16(4)

Опубликована: Янв. 11, 2024

Abstract Multicomponent reactions provide an excellent approach toward quaternary carbon centres utilizing convergent chemical in a highly selective manner under one‐pot conditions. The reactivity of substrates and metal catalysts is carefully controlled, precluding the formation side‐products. In this context, transition catalyzed onium ylides generated via diazo precursors nucleophiles with third component (an electrophile) have garnered significant attention. Using allylic precursor as electrophilic partner provides opportunities to construct all‐carbon centres. Furthermore, presence allyl fragment multicomponent product serves pivotal handle for carrying out subsequent modifications. Several recent studies employed Rh, Pd, dual Rh/Pd catalytic systems involving alkylation that proceed synergistic or relay pathway. Although not significantly successful, few cases, asymmetric induction achieved through chiral phosphoric acids phosphine ligands. Limited substrate catalyst scope underlying mechanistic complexities posed formidable challenges, slowing advancement reactions. This review details using readily available like compounds, carbonates, (R‐OH, R‐NH 2 , etc .) forming complex organic compounds. Our primary objective discuss issues may facilitate progress field.

Язык: Английский

Процитировано

6

A combined experimental and computational study reveals a crossover between conventional cross-coupling and carbene insertion pathways in a Pd catalyzed C(sp2)–H insertion DOI Creative Commons

Arushi Tyagi,

Kritika Gaur,

Anubhav Goswami

и другие.

Chemical Science, Год журнала: 2025, Номер unknown

Опубликована: Янв. 1, 2025

Computational (DFT and DLPNO-CCSD(T)) calculations along with experimental tools (deuterium labelling, kinetic studies using VTNA, ESI-HRMS UV) are used to probe the mechanism of a Pd(ii)-catalyzed enantioselective carbene insertion into C(sp2)-H indole. Using deuterium labelling studies, we demonstrate intermediacy metal-hydride species, which contrasts mechanistic routes for other transition metals (Rh, Fe, Au, Cu, etc.). Our VTNA study reveals order be one in both diazo indole, microkinetic modelling aligns well computationally predicted mechanism. The is further supported by detection most stable intermediate catalytic cycle ESI-HRMS. An investigation origin stereoselectivity DLPNO-CCSD(T) presents new paradigm, wherein stereocontrol arises during formation Pd itself as opposed proton transfer steps found all metal catalysts.

Язык: Английский

Процитировано

0

Advances in catalysis using Xantphos-like ligands; simplicity goes a long way DOI
Piet W. N. M. van Leeuwen, Israel Cano, Zoraida Freixa

и другие.

Coordination Chemistry Reviews, Год журнала: 2025, Номер 537, С. 216636 - 216636

Опубликована: Апрель 11, 2025

Язык: Английский

Процитировано

0

Divergent Reactions of α-Diazo 1,3-Dicarbonyl Compounds with Allylic Carbonates Involving Ketene versus Carbene Intermediates Enabled by Cooperative Rh(II)/Pd(0) Dual Catalysis DOI

De-Xin Song,

Yuhua Song,

Heng-Hua Huang

и другие.

Organic Letters, Год журнала: 2024, Номер 26(37), С. 7920 - 7925

Опубликована: Сен. 9, 2024

A cooperative Rh(II)/Pd(0) dual-catalysis strategy that enabled divergent reactions of α-diazo 1,3-dicarbonyl compounds with allylic carbonates involving ketene versus carbene intermediates is described. The efficient synthesis α-quaternary allylated β-keto-esters was accomplished by the alkylation compounds. Alternatively, an unprecedented (1+4) annulation 2-(hydroxymethyl)allyl via dual catalysis also successfully developed, affording a wide variety tetrahydrofurans in good to high yields.

Язык: Английский

Процитировано

2

Rh(II)-Catalyzed Chemoselective Oxy-alkynylation of Acceptor–Acceptor Carbenes: Synthesis of C2-Quaternary Alkyne-Substituted 3(2H)-Furanones DOI
Qing Liu,

Yang‐Ting Ma,

Xiaoyan Huang

и другие.

Organic Letters, Год журнала: 2023, Номер 25(22), С. 4044 - 4049

Опубликована: Май 31, 2023

A Rh(II)-catalyzed oxy-alkynylation of acceptor-acceptor carbenes using EBX reagents was successfully developed. The key alkyne-transfer step is likely to occur through a tandem process involving β-addition, an α-elimination, and 1,2-shift, which supported by the formation alkylidene carbene. Various diverse C2-quaternary alkyne-substituted benzofuran-3-ones 2,2,4,5-tetrasubstituted 3(2H)-furanones can be synthesized smoothly, depending on choice diazo compounds base additives. Furthermore, this reaction characterized mild conditions, high functional group compatibility, broad substrate scope.

Язык: Английский

Процитировано

2

Three‐component allylic alkylation reaction of α‐diazo ketones with water and allyl carbonates for construction of homoallylic alcohols DOI

Liping Yin,

Xinyi Zhang,

B. D. Wang

и другие.

Advanced Synthesis & Catalysis, Год журнала: 2024, Номер 366(17), С. 3616 - 3623

Опубликована: Июнь 20, 2024

Abstract A three‐component allylic alkylation reaction of α‐diazo ketones, water and allyl carbonate under the cooperative catalysis Rh 2 (OAc) 4 , Pd (dba) 3 Brønsted acid was disclosed. This method provides an expeditious access to α‐keto homoallylic alcohols in good high yields. Controlled experiments support that transformations proceed through cross‐interception two active intermediates Pd‐allyl species enol derived from oxonium ylides. Moreover, synthetic generated products enable creation motifs enriched with dense functional groups, underscoring their potential as valuable building blocks.

Язык: Английский

Процитировано

0