Fabrication and In Vivo Evaluation of In Situ pH-Sensitive Hydrogel of Sonidegib–Invasomes via Intratumoral Delivery for Basal Cell Skin Cancer Management DOI Creative Commons

Maha M. Ghalwash,

Amr Gamal,

Nada H. Mohammed

и другие.

Pharmaceuticals, Год журнала: 2024, Номер 18(1), С. 31 - 31

Опубликована: Дек. 30, 2024

Basal cell skin cancer (BCSC) develops when cells proliferate uncontrollably. Sonidegib (SDB) is a therapeutic option for the treatment of BCSC by inhibiting hedgehog signaling. The problems with SDB's low solubility, poor bioavailability, resistance, targeting, and first-pass action make it less effective taken orally. This investigation set out to design an intratumoral in situ pH-sensitive hydrogel SDB-invasomes (IPHS-INV) that can effectively treat improving sustainability, efficacy while also reducing its resistance undesirable side effects. Numerous S-INV formulations were developed using Box-Behnken Design Expert tested before settling on optimum formulation. An experimental 7, 12-dimethylbenzanthracene (DMBA) carcinoma rat model was used vivo studies IPHS-INV formulation after combined chitosan. Phospholipids (1.72% w/w), cholesterol (0.15% ethanol (1% v/v), cineole (1.5% v/v) shown be optimal components SDB-invasome outperformed permeation bioavailability free SDB 7.14 6 times, respectively, sustained release 57.41%. showed decrease tumor volume 99.05% reduction hypercellular tumors, indicating anti-cancer activity. maintained higher concentration targeting These findings support use as strategy BCSC.

Язык: Английский

Improved wound care via novel dextran and boric acid loaded wound healing gel in excision mice wound model DOI

Nosheen Maqbool,

Zakir Ali,

Sibgha Batool

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2025, Номер unknown, С. 106586 - 106586

Опубликована: Янв. 1, 2025

Язык: Английский

Процитировано

4

Fabrication of oral sustained release capecitabine loaded nanostructured lipid carriers with improved bioavailability and prolonged anticancer effects DOI

Mohsin Fawad,

Zakir Ali, Fatima Zahid

и другие.

Journal of Molecular Liquids, Год журнала: 2025, Номер 421, С. 126852 - 126852

Опубликована: Янв. 5, 2025

Язык: Английский

Процитировано

4

Development of Paroxetine Loaded Nanotransferosomal Gel for Intranasal Delivery with Enhanced Antidepressant Activity in Rats DOI
Akbar Tahir, Sidra Aslam, Saba Sohail

и другие.

Colloids and Surfaces B Biointerfaces, Год журнала: 2024, Номер 246, С. 114351 - 114351

Опубликована: Ноя. 7, 2024

Язык: Английский

Процитировано

6

Physicochemical characterization and in vivo assessment of novel apixaban-loaded polymeric nano-aggregates DOI
Fakhar ud Din, Hye In Lee, Jung Suk Kim

и другие.

Journal of Pharmaceutical Investigation, Год журнала: 2024, Номер unknown

Опубликована: Окт. 31, 2024

Язык: Английский

Процитировано

5

A thermoresponsive system of niclosamide for colon specific delivery in ulcerative colitis: Bioavailability and safety investigation DOI
Ali H. Alamri, Adel Al Fatease, Zakir Ali

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2025, Номер unknown, С. 106641 - 106641

Опубликована: Янв. 1, 2025

Язык: Английский

Процитировано

0

Improved biopharmaceutical performance of chlorpromazine-nanostructured lipid carriers: In vitro release, pharmacokinetics and toxicity testing DOI
Khushi Muhammad,

Uswa Shafique,

Abad Khan

и другие.

Journal of Drug Delivery Science and Technology, Год журнала: 2025, Номер unknown, С. 106885 - 106885

Опубликована: Апрель 1, 2025

Язык: Английский

Процитировано

0

Comparative analysis of novel modified drug delivery systems for improving the oral bioavailability of water-insoluble tadalafil using copovidone, TPGS and hydroxypropyl-β-cyclodextrin DOI
Fakhar ud Din, Dong Shik Kim, Jung Suk Kim

и другие.

Biomedicine & Pharmacotherapy, Год журнала: 2025, Номер 186, С. 118039 - 118039

Опубликована: Апрель 8, 2025

Язык: Английский

Процитировано

0

Thermoresponsive biomaterial system of Irinotecan and Curcumin for the treatment of colorectal cancer: In-vitro and in-vivo investigations DOI

Aleena Maryiam,

Sibgha Batool,

Zakir Ali

и другие.

Pharmaceutical Development and Technology, Год журнала: 2024, Номер 30(1), С. 37 - 56

Опубликована: Дек. 27, 2024

This study aims to develop a thermoresponsive biomaterial system of irinotecan (IRT) and curcumin (CUR) nano-transferosomal gel (IRT-CUR-NTG) for targeting colorectal cancer (CRC). The IRT-CUR-NTs were statistically optimized loaded into poloxamer-based thermosensitive gel. Transmission electron microscopy (TEM), Differential scanning calorimetry (DSC) Fourier-transform infrared spectroscopy (FTIR) the performed, whereas pH, gelation time, temperature, mucoadhesive strength IRT-CUR-NTG investigated. In-vitro release anticancer analyses explored using HT29 cells. Additionally, in-vivo pharmacokinetics was investigated followed by histopathological examination analysis. PS, PDI, ZP, %EE IRT CUR found be 136.15 nm, 0.143, -15.5 mV, 95.05% 85.12%, respectively. exhibited spherical shape with no chemical interactions among constituents. Similarly, homogenous suitable rectal administration. manifested prolonged profiles CUR. Moreover, significantly enhanced (4-fold) bioavailability toxicity observed when compared conventional more effective against cell lines. In-vivo antitumor analysis demonstrated reduced tumor volume mass after treatment IRT-CUT-NTG, indicating improved effect. It can concluded that is cancer.

Язык: Английский

Процитировано

1

Fabrication and In Vivo Evaluation of In Situ pH-Sensitive Hydrogel of Sonidegib–Invasomes via Intratumoral Delivery for Basal Cell Skin Cancer Management DOI Creative Commons

Maha M. Ghalwash,

Amr Gamal,

Nada H. Mohammed

и другие.

Pharmaceuticals, Год журнала: 2024, Номер 18(1), С. 31 - 31

Опубликована: Дек. 30, 2024

Basal cell skin cancer (BCSC) develops when cells proliferate uncontrollably. Sonidegib (SDB) is a therapeutic option for the treatment of BCSC by inhibiting hedgehog signaling. The problems with SDB's low solubility, poor bioavailability, resistance, targeting, and first-pass action make it less effective taken orally. This investigation set out to design an intratumoral in situ pH-sensitive hydrogel SDB-invasomes (IPHS-INV) that can effectively treat improving sustainability, efficacy while also reducing its resistance undesirable side effects. Numerous S-INV formulations were developed using Box-Behnken Design Expert tested before settling on optimum formulation. An experimental 7, 12-dimethylbenzanthracene (DMBA) carcinoma rat model was used vivo studies IPHS-INV formulation after combined chitosan. Phospholipids (1.72% w/w), cholesterol (0.15% ethanol (1% v/v), cineole (1.5% v/v) shown be optimal components SDB-invasome outperformed permeation bioavailability free SDB 7.14 6 times, respectively, sustained release 57.41%. showed decrease tumor volume 99.05% reduction hypercellular tumors, indicating anti-cancer activity. maintained higher concentration targeting These findings support use as strategy BCSC.

Язык: Английский

Процитировано

0