Continuous Flow Synthesis of Five‐Membered N‐Heterocycles by Ynone System DOI Open Access
Tamilselvan Duraisamy,

Vijay Thavasianandam Seenivasan,

Li‐Yu Wang

и другие.

Asian Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Окт. 18, 2024

Abstract In this study, we devised a practical and effective method for synthesizing ynones from terminal alkynes anhydride utilizing continuous flow apparatus at ambient temperature. Moreover, coupled the with hydrazines, hydroxylamine hydrochloride to synthesize pyrazole isoxazole derivatives. This protocol's unique characteristics include metal‐free approach, mild reaction conditions, short residence time, wide range of functional group tolerance. Sustainable strategies are most useful affordable than conventional benchtop approaches.

Язык: Английский

Exploring structure, molecular interactions, optical and thermal properties of Bis(2-Aminopyrimidinium) selenate monohydrate: A combined experimental and theoretical study DOI

V. Vijayalakshmi,

N. Sivakumar,

V. Ali Alsulmi

и другие.

Optical Materials, Год журнала: 2024, Номер 152, С. 115539 - 115539

Опубликована: Май 21, 2024

Язык: Английский

Процитировано

12

Current strategies in design and synthesis of antifungals hybrid and chimeric diazine derivatives DOI Creative Commons
Dumitrela Diaconu,

Marius Savu,

Catalina Ionica Ciobanu

и другие.

Bioorganic & Medicinal Chemistry, Год журнала: 2025, Номер 119, С. 118069 - 118069

Опубликована: Янв. 13, 2025

Язык: Английский

Процитировано

1

Pyrimidines: A New Versatile Molecule in the Drug Development Field, Scope, and Future Aspects DOI Creative Commons
Katharigatta N. Venugopala, Vinuta Kamat

Pharmaceuticals, Год журнала: 2024, Номер 17(10), С. 1258 - 1258

Опубликована: Сен. 24, 2024

Pyrimidine is a moiety that occurs in living organisms and has variety of significant biological properties pharmacology. Due to the easy handling synthesis, easily available precursor, less duration for reaction, not many technical skills are needed. All these factors attract chemists focus more on pyrimidines. Apart from synthesis applications pyrimidines, medicinal have gathered explore pyrimidine scaffolds due their interesting targeting various binding sites. This review delves into diverse activities compounds derived during year 2024. We attempted growing significance derivatives provide new path designing potent molecules.

Язык: Английский

Процитировано

3

Recent advancements of pyrimidine chemistry thriving deeper into drug discovery DOI
Glanish Jude Martis,

O Sneha,

Rajkumar Bhat D

и другие.

Synthetic Communications, Год журнала: 2025, Номер unknown, С. 1 - 29

Опубликована: Апрель 3, 2025

Язык: Английский

Процитировано

0

Evaluation of anticancer potential of diorganotin(IV) complexes derived from 4-nitro-3-methylbenzhydrazide: Synthesis, spectral and single crystal analysis DOI

Shikha Poonia,

Sonika Asija, Kashmiri Lal

и другие.

Journal of Molecular Structure, Год журнала: 2025, Номер unknown, С. 142361 - 142361

Опубликована: Апрель 1, 2025

Язык: Английский

Процитировано

0

The futuristic applications of transition metal dichalcogenides for cancer therapy DOI
Shouvik Kumar Nandy,

Sattwik Das,

Sadanand Pandey

и другие.

Luminescence, Год журнала: 2024, Номер 39(5)

Опубликована: Май 1, 2024

Abstract The second‐most common cause of death resulting from genetic mutations in DNA sequences is cancer. difficulty the field anticancer research application traditional methods, which also affects normal cells. Mutations, replication alterations, and chromosomal abnormalities have a direct impact on effectiveness drugs at different stages. Presently, therapeutic techniques utilize nanotechnology, transition metal dichalcogenides (TMDCs), robotics. TMDCs are being increasingly employed tumor therapy biosensing applications due to their biocompatibility, adjustable bandgap, versatile functionality, exceptional photoelectric properties, wide range applications. This study reports advancement nanoplatforms based that specifically engineered for responsive intelligent cancer therapy. article offers thorough examination current challenges, future possibilities theranostic using TMDCs, recent progress employing Currently, there significant interest two‐dimensional (2D) nanomaterials as ultrathin unique physicochemical properties. These materials attracted attention various fields, including biomedicine. Due inherent ability absorb near‐infrared light exceptionally large surface area, efforts made prepare multifunctional 2D TMDCs.

Язык: Английский

Процитировано

1

New thiadiazolopyrimidine-ornamented pyrazoles as prospective anticancer candidates via suppressing VEGFR-2/PI3K/Akt signaling pathway: Synthesis, characterization, in-silico, and in-vitro studies DOI
Maha M. Salem, Marian N. Gerges,

Hayam A. Abd El Salam

и другие.

International Journal of Biological Macromolecules, Год журнала: 2024, Номер unknown, С. 138735 - 138735

Опубликована: Дек. 1, 2024

Язык: Английский

Процитировано

0

Design, synthesis, α-amylase and glucose diffusion inhibition, and molecular docking studies of new indenopyrazolones bearing benzothiazole derivatives DOI
Ravinder Punia, Satbir Mor,

Suchita Sindhu

и другие.

Bioorganic & Medicinal Chemistry Letters, Год журнала: 2024, Номер 103, С. 129692 - 129692

Опубликована: Март 5, 2024

Язык: Английский

Процитировано

0

Continuous Flow Synthesis of Five‐Membered N‐Heterocycles by Ynone System DOI Open Access
Tamilselvan Duraisamy,

Vijay Thavasianandam Seenivasan,

Li‐Yu Wang

и другие.

Asian Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Окт. 18, 2024

Abstract In this study, we devised a practical and effective method for synthesizing ynones from terminal alkynes anhydride utilizing continuous flow apparatus at ambient temperature. Moreover, coupled the with hydrazines, hydroxylamine hydrochloride to synthesize pyrazole isoxazole derivatives. This protocol's unique characteristics include metal‐free approach, mild reaction conditions, short residence time, wide range of functional group tolerance. Sustainable strategies are most useful affordable than conventional benchtop approaches.

Язык: Английский

Процитировано

0