Synthesis, Properties, and Biological Activity of Benzothiadiazine DOI
Navnath T. Hatvate, Rutuja Rambhau Ukhade, Hemantkumar N. Akolkar

и другие.

Advances in bioinformatics and biomedical engineering book series, Год журнала: 2024, Номер unknown, С. 317 - 346

Опубликована: Ноя. 27, 2024

Heterocyclic compounds are ubiquitous in biologically active compounds, including many drugs. Benzothiadiazine is a class of sulphur and nitrogen-containing heterocyclic comprised benzene ring fused with thiadiazine. rings appear marketed drugs, such as bendroflumethiazide, chlorothiazide, cyclothiazide, hydrochlorothiazide, diazoxide, which popularly known for their diuretic activity. The has diverse pharmacological activity, anti-cancer, antifungal, antimicrobial, anthelmintic, hypolipidaemic, antidiabetic This chapter focuses on the chemistry, synthetic methods, bioactivity different benzothiadiazine. Furthermore, updates patents clinical trials have also been summarized present chapter.

Язык: Английский

Recent advances in meglumine catalyzed organic synthesis: A comprehensive review DOI

Dharti R. Bhandari,

Urvi J. Khengar,

Rajesh H. Vekariya

и другие.

Synthetic Communications, Год журнала: 2024, Номер 54(16), С. 1285 - 1310

Опубликована: Авг. 1, 2024

Meglumine, an amino sugar alcohol compound, has recently emerged as a promising catalyst in various organic transformations due to its unique properties. This review provides comprehensive overview of the applications meglumine synthesis, highlighting their efficiency, versatility, and mechanistic insights. Key examples reactions catalyzed by meglumine, including aldol condensation, Michael addition, Mannich reaction, other one-pot multicomponent condensation reaction are discussed along with pathways synthetic strategies. Additionally, recent advancements future perspectives field explored.

Язык: Английский

Процитировано

1

An efficient, green and solvent-free three-component synthesis of 2,4,6-triarylpyridines utilizing ZSM-5 as a heterogeneous catalyst DOI
Navnath T. Hatvate, Juhi Gupta

Synthetic Communications, Год журнала: 2024, Номер unknown, С. 1 - 11

Опубликована: Сен. 12, 2024

Язык: Английский

Процитировано

1

Synthesis of Isoxazol-5-One Derivatives Catalyzed by Amine-Functionalized Cellulose DOI Creative Commons

Sanaz Gharehassanlou,

Hamzeh Kiyani

Organics, Год журнала: 2024, Номер 5(4), С. 378 - 394

Опубликована: Окт. 12, 2024

In this contribution, propylamine-functionalized cellulose (Cell-Pr-NH2) was employed as the catalyst in three-component reaction between hydroxylamine hydrochloride and various types of aryl/heteroaryl aldehydes, ethyl acetoacetate/ethyl 4-chloroacetoacetate, or 3-oxohexanoate. The result these experiments formation 3,4-disubstituted isoxazol-5(4H)-one heterocycles. desired five-membered heterocyclic compounds were obtained good to high yields at room temperature. investigation different solvents led us conclusion that water is best solvent perform current one-pot, reactions. Attempts find optimal loading clearly showed 14 mg cell-Pr-NH2 seems be sufficient carry out This method has highlighted some principles green chemistry including less waste generation, atom economy, use an environmentally friendly solvent, energy saving. Purification without chromatographic methods, mild conditions, simple work-up, low-cost medium, saving time, obtainable precursors are other notable features one-pot fashion.

Язык: Английский

Процитировано

1

Synthesis, Properties, and Biological Activity of Benzothiadiazine DOI
Navnath T. Hatvate, Rutuja Rambhau Ukhade, Hemantkumar N. Akolkar

и другие.

Advances in bioinformatics and biomedical engineering book series, Год журнала: 2024, Номер unknown, С. 317 - 346

Опубликована: Ноя. 27, 2024

Heterocyclic compounds are ubiquitous in biologically active compounds, including many drugs. Benzothiadiazine is a class of sulphur and nitrogen-containing heterocyclic comprised benzene ring fused with thiadiazine. rings appear marketed drugs, such as bendroflumethiazide, chlorothiazide, cyclothiazide, hydrochlorothiazide, diazoxide, which popularly known for their diuretic activity. The has diverse pharmacological activity, anti-cancer, antifungal, antimicrobial, anthelmintic, hypolipidaemic, antidiabetic This chapter focuses on the chemistry, synthetic methods, bioactivity different benzothiadiazine. Furthermore, updates patents clinical trials have also been summarized present chapter.

Язык: Английский

Процитировано

0