Visible-Light-Induced Cascade Cyclization of 1-(2-(Arylethynyl)benzoyl)indoles into Sulfonated Benazepino[1,2-a]indolones

Organic Letters, Год журнала: 2024, Номер 26(50), С. 10982 - 10987

Опубликована: Дек. 10, 2024

1-(2-(Arylethynyl)benzoyl)indoles were developed as an innovative scaffold for radical cascade cyclization under visible-light and mild conditions, enabling efficient synthesis of sulfonated benazepino[1,2-

Язык: Английский

Electrochemical synthesis of γ-carbolinones via sulfonylation-triggered cyclization of indole-3-carboxamides

Organic & Biomolecular Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Дек. 5, 2024

A novel electrochemical cyclization reaction of N -acryloyl-indole-3-carboxamides has been developed, which provides a new and efficient strategy for the synthesis γ-carbolinone derivatives.

Язык: Английский

Synthesis of dithioacetals via nucleophilic substitution and their antifungal activity evaluation

Organic & Biomolecular Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Янв. 1, 2024

A novel substitution reaction of dichloromethane with thiols is developed, affording varieties dithioacetals and α-acyloxy sulfides in up to 96% yields. Moreover, the obtained exhibit excellent antifungal activity against L. theobromae .

Язык: Английский