Access to syn α‐Amino‐β‐Hydroxyesters by N‐H Insertion on O‐Protected α‐Diazo‐β‐Hydroxyesters. DOI Creative Commons

Thomas Defuentes,

Jérôme Lhoste, Catherine Gaulon‐Nourry

и другие.

Asian Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Ноя. 13, 2024

Abstract The N−H insertion reaction is a versatile method for creating C−N bonds under mild conditions, providing in particular an efficient access to both natural and non‐natural α‐amino acid derivatives. In this field, the direct on α‐diazo‐β‐hydroxyesters has not yet been investigated constitutes significant challenge, due competitive migration processes. We report herein first insertions O ‐protected α‐diazo‐β‐aryl‐β‐hydroxyesters, enabling synthesize wide range of α‐amino‐β‐hydroxyesters by tuning nature amine aryl substituent. Overall, 28 products have isolated, with moderate good yields most cases, diastereoisomeric ratios up 8.0 : 1 favor syn diastereoisomer.

Язык: Английский

Visible Light-Induced Reactions of Diazo Compounds and Their Precursors DOI
Ziyan Zhang, Vladimir Gevorgyan

Chemical Reviews, Год журнала: 2024, Номер 124(11), С. 7214 - 7261

Опубликована: Май 16, 2024

In recent years, visible light-induced reactions of diazo compounds have attracted increasing attention in organic synthesis, leading to improvement existing reactions, as well the discovery unprecedented transformations. Thus, photochemical or photocatalytic generation both carbenes and radicals provide milder tools toward these key intermediates for many valuable However, vast majority transformations represent new reactivity modes compounds, which are achieved by decomposition photoredox catalysis. particular, use a redox-active photocatalysts opens avenue plethora radical reactions. The application methods led inaccessible classical associated with metal carbenes. most cases, act sources but can also serve acceptors. Importantly, described processes operate under mild, practical conditions. This Review describes this subfield compound chemistry, particularly focusing on advancements.

Язык: Английский

Процитировано

60

General Ir-Catalyzed N–H Insertions of Diazomalonates into Aliphatic and Aromatic Amines DOI Creative Commons

Zhong Zhuang,

Céline Besnard, Jérôme Lacour

и другие.

Organic Letters, Год журнала: 2024, Номер 26(5), С. 983 - 987

Опубликована: Янв. 26, 2024

A general N–H insertion reactivity of acceptor–acceptor diazo malonate reagents is reported using [Ir(cod)Cl]2 as catalyst. large range amines, primary and secondary, aliphatic aromatic, possible. Mild temperatures, perfect substrate/reactant stoichiometry, good functional group compatibility render the process particularly attractive for (late-stage) functionalization amines.

Язык: Английский

Процитировано

5

Visible-light-driven Synthesis of Benzoxepine Derivatives from Aromatic Diazo Compounds DOI

Xiuyuan Duan,

Guojun Zheng

Tetrahedron, Год журнала: 2025, Номер unknown, С. 134620 - 134620

Опубликована: Март 1, 2025

Язык: Английский

Процитировано

0

Axis-to-Center Chirality Transfer Reactions of Phosphates with a Binaphthyl Group and Their Congeners: New Synthetic Routes to P-Chirogenic Organophosphorus Compounds DOI
Toshiaki Murai

Chemistry Letters, Год журнала: 2023, Номер 52(9), С. 703 - 714

Опубликована: Июль 31, 2023

Abstract Novel synthetic methods for P-chirogenic four-coordinate pentadentate organophosphorus compounds are described. The pathways commenced with the use of phosphates bearing a binaphthyl group and their congeners. These underwent reactions fluoride ion, metal hydroxides, alkoxides, Grignard reagents, resulting in transfer axial chirality from to central phosphorus atom. As result, products incorporating were obtained. substitution these newly formed alkoxides reagents led formation phosphates, phosphonates, phosphinates, some sulfur isologues.

Язык: Английский

Процитировано

8

Synthesis of a versatile 1H-indene-3-carboxylate scaffold enabled by visible-light promoted Wolff rearrangement of 1-diazonaphthalen-2(1H)-ones DOI
Xin Yue, Ying Zhou, Yan Zhang

и другие.

Chemical Communications, Год журнала: 2023, Номер 59(42), С. 6363 - 6366

Опубликована: Янв. 1, 2023

Herein, we have developed a sequential visible-light-promoted Wolff rearrangement of 1-diazonaphthalen-2(1H)-ones, followed by capturing the in situ generated ketene intermediates with various alcohols, producing diverse 1H-indene-3-carboxylates moderate to good yields under mild reaction conditions. The broad substrate scope, high functional group tolerance, and robust conditions make resulting derivative versatile platform for synthesis plenty bioactive molecules.

Язык: Английский

Процитировано

4

Access to syn α‐Amino‐β‐Hydroxyesters by N‐H Insertion on O‐Protected α‐Diazo‐β‐Hydroxyesters. DOI Creative Commons

Thomas Defuentes,

Jérôme Lhoste, Catherine Gaulon‐Nourry

и другие.

Asian Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Ноя. 13, 2024

Abstract The N−H insertion reaction is a versatile method for creating C−N bonds under mild conditions, providing in particular an efficient access to both natural and non‐natural α‐amino acid derivatives. In this field, the direct on α‐diazo‐β‐hydroxyesters has not yet been investigated constitutes significant challenge, due competitive migration processes. We report herein first insertions O ‐protected α‐diazo‐β‐aryl‐β‐hydroxyesters, enabling synthesize wide range of α‐amino‐β‐hydroxyesters by tuning nature amine aryl substituent. Overall, 28 products have isolated, with moderate good yields most cases, diastereoisomeric ratios up 8.0 : 1 favor syn diastereoisomer.

Язык: Английский

Процитировано

0