Annulative Coupling of β‐Ketosulfoxonium Ylides and β‐Ketothioamides: Access to Thiazolines and Thiazolidin‐4‐Ones DOI

Rahul Kumar Saini,

Satyendra Kumar Pandey

Advanced Synthesis & Catalysis, Год журнала: 2024, Номер 366(19), С. 4073 - 4077

Опубликована: Июль 3, 2024

Abstract A catalyst‐ and additive‐free one‐step protocol for synthesizing thiazolines thiazolidin‐4‐ones, utilizing the annulative coupling between β‐ketosulfoxonium ylides β‐ketothioamides has been described. The dual functionalization of through S‐alkylation intramolecular N‐cyclization leads to generation both C−S C−N bonds. developed synthetic methods facilitate synthesis diverse functionalized thiazolidin‐4‐one derivatives, validated large‐scale reactions.

Язык: Английский

Direct C−H Sulfuration: Synthesis of Disulfides, Dithiocarbamates, Xanthates, Thiocarbamates and Thiocarbonates DOI
Qiao Sun, Yuan Xu,

Liu Yang

и другие.

Chemistry - An Asian Journal, Год журнала: 2024, Номер 19(9)

Опубликована: Фев. 29, 2024

Abstract In light of the important biological activities and widespread applications organic disulfides, dithiocarbamates, xanthates, thiocarbamates thiocarbonates, continual persuit efficient methods for their synthesis remains crucial. Traditionally, preparation such compounds heavily relied on intricate multi‐step syntheses use highly prefunctionalized starting materials. Over past two decades, direct sulfuration C−H bonds has evolved into a straightforward, atom‐ step‐economical method organosulfur compounds. This review aims to provide an up‐to‐date discussion disulfuration, dithiocarbamation, xanthylation, thiocarbamation thiocarbonation, with special focus describing scopes mechanistic aspects. Moreover, synthetic limitations some these methodologies, along key unsolved challenges be addressed in future are also discussed. The majority examples covered this accomplished via metal‐free, photochemical or electrochemical approaches, which alignment overraching objectives green sustainable chemistry. comprehensive consolidate recent advancements, providing valuable insights dynamic landscape strategies crucial classes

Язык: Английский

Процитировано

4

Catalyst/Metal/Solvent-Free Markovnikov Hydrothiolation of Unactivated Alkenes with Dithiocarbamic Acids DOI
Azim Ziyaei Halimehjani, Ziya Dağalan,

Zahra Marjani

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(8), С. 5353 - 5362

Опубликована: Апрель 2, 2024

Catalyst-free Markovnikov-selective hydrothiolation of unactivated alkenes still remains a great challenge. Herein, we develop catalyst/metal/solvent-free methodology for the Markovnikov with in situ prepared dithiocarbamic acids, providing wide array alkyl dithiocarbamates. A variety terminal, internal, cyclic, and acyclic were applied successfully this protocol. This three-component thiol–ene reaction can be considered as new family click reactions.

Язык: Английский

Процитировано

3

High-efficient green catalytic conversion for waste CS2 by non-noble metal cage-based MOFs: An access to high-valued thiazolidine-2-thione DOI

Wenyu Ding,

Xinyu Tang,

Sheng Chih Jin

и другие.

Green Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Янв. 1, 2024

High-efficiency non-noble cage-based MOFs catalyst for CS 2 waste green disposal through catalytic conversion into high-value thiazolidine-2-thione.

Язык: Английский

Процитировано

3

Electro-Oxidative Three-Component Synthesis of 3,5-Disubstituted-1,2,4-Thiadiazoles from Amines, Amidines, and CS2 DOI
Peng‐Fei Huang, Ying Peng,

Jia-Le Fu

и другие.

The Journal of Organic Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Март 29, 2025

1,2,4-Thiadiazoles, a significant class of heterocyclic compounds, are widely found in biologically active molecules. Herein, we report green electrochemical three-component reaction amines, amidines, and CS2 for the effective synthesis 3,5-disubstituted-1,2,4-thiadiazoles under metal- oxidant-free conditions. Both aliphatic aryl amines well-tolerated at room temperature simple undivided cell. A series 1,2,4-thiadiazoles prepared with excellent functional groups.

Язык: Английский

Процитировано

0

Lithium Bromide-Promoted Formal C(sp3)–H Bond Insertion Reactions of β-Carbonyl Esters with Sulfoxonium Ylides to Synthesize 1,4-Dicarbonyl Compounds DOI

Hailin Guo,

Yuhao Ding,

Jing-Wen Fan

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(10), С. 6974 - 6986

Опубликована: Май 4, 2024

A LiBr-promoted formal C(sp3)–H bond insertion reaction between β-carbonyl esters and sulfoxonium ylides is established. This practical has a wide range of substrate scope for both to give variety 1,4-dicarbonyl compounds with 43–94% yields. The features transition-metal-free conditions exclusive C-alkylation chemselectivity. use bench-stable overcomes previous methods that require transition metal as catalysts unstable diazo or toxic haloketones alkylation reagents.

Язык: Английский

Процитировано

2

Annulative coupling of sulfoxonium ylides with 2‑amino(thio)phenols: Easy access to 2-acyl benzox(thio)azoles DOI

Trayambek Nath Chaubey,

Paran J. Borpatra, Satyendra Kumar Pandey

и другие.

Organic & Biomolecular Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Янв. 1, 2024

A novel elemental sulfur-mediated approach for the synthesis of 2-acyl benzothiazoles and benzoxazole derivatives via annulative coupling sulfoxonium ylides with 2-aminobenzenethiol 2-aminophenol derivatives, respectively, is described.

Язык: Английский

Процитировано

1

Base-mediated synthesis of cyclic dithiocarbamates from 1-amino-3-chloropropan-2-ol derivatives and carbon disulfide DOI
Yasunori Toda,

Masaya Iwasaki,

Hiroyuki Suga

и другие.

Organic & Biomolecular Chemistry, Год журнала: 2023, Номер 21(31), С. 6293 - 6297

Опубликована: Янв. 1, 2023

An efficient method for the preparation of six-membered cyclic dithiocarbamates is described, in which triethylamine effectively promotes reaction 1-amino-3-chloropropan-2-ol derivatives with carbon disulfide. On basis experimental and theoretical studies, a mechanism proposed to explain difference between present our previously reported dioxide fixation.

Язык: Английский

Процитировано

2

Sc(OTf)3-catalyzed diastereoselective [4 + 2] cycloaddition reaction of 3-benzylideneindoline-2-thiones with alkylidene malonates DOI
Xuelong Wang, Junyi Zeng, Yi Yang

и другие.

Tetrahedron Letters, Год журнала: 2023, Номер 135, С. 154886 - 154886

Опубликована: Дек. 13, 2023

Язык: Английский

Процитировано

2

Annulative Coupling of β‐Ketosulfoxonium Ylides and β‐Ketothioamides: Access to Thiazolines and Thiazolidin‐4‐Ones DOI

Rahul Kumar Saini,

Satyendra Kumar Pandey

Advanced Synthesis & Catalysis, Год журнала: 2024, Номер 366(19), С. 4073 - 4077

Опубликована: Июль 3, 2024

Abstract A catalyst‐ and additive‐free one‐step protocol for synthesizing thiazolines thiazolidin‐4‐ones, utilizing the annulative coupling between β‐ketosulfoxonium ylides β‐ketothioamides has been described. The dual functionalization of through S‐alkylation intramolecular N‐cyclization leads to generation both C−S C−N bonds. developed synthetic methods facilitate synthesis diverse functionalized thiazolidin‐4‐one derivatives, validated large‐scale reactions.

Язык: Английский

Процитировано

0