Bioinspired Synthesis of Phelligridin Analogues via Ru-Catalyzed C–H Activation/[4 + 2] Annulation of Aryl Imidates with Heteroaromatic Iodonium Ylides DOI

Mingdian Liang,

Si-Jing Huang,

Dongyang Zhang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Дек. 16, 2024

The first Ru(II)-catalyzed C–H activation/[4 + 2] annulation of aryl imidates with heteroaromatic iodonium ylides is reported. Our approach features the utilization a commercially available ruthenium catalyst, providing one-step construction phelligridin analogues from easily and nonpreactivated starting materials. developed methodology successfully employed for total synthesis A, significantly streamlining previous multistep synthesis. potential this further demonstrated through modular core structure C/D.

Язык: Английский

Iodonium(III) Ylide: An Iodoalkylation Reagent with Aryne DOI
Weigang Xu, Pengfei Li,

Yuerong Li

и другие.

The Journal of Organic Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Фев. 5, 2025

A tandem Hexadehydro-Diels–Alder (HDDA)/[2 + 2] cycloaddition/aryl migration reaction of iodonium ylide with tetrayne is described, in which served as a unique double bond and reacted aryne to form four-membered iodonium(III) cycle, then converted iodoarene after aryl group from iodine adjacent carbon. This strategy allows the efficient construction fully substituted compounds.

Язык: Английский

Процитировано

0

Rh-Catalyzed Coupling of Cyclic 1,3-Dicarbonyl-Derived Iodonium Ylides with Cyclopropanols DOI

Zongye Wang,

Mingxuan Liang,

Dongyang Zhang

и другие.

Organic Letters, Год журнала: 2025, Номер unknown

Опубликована: Апрель 10, 2025

Herein, we report a modular α-monoalkylation of cyclic 1,3-dicarbonyls with cyclopropyl alcohols through iodonium ylide strategy. This approach is general, base-free, operationally simple, and suitable for various medically important (hetero)cyclic 1,3-dicarbonyls. A wide range alcohols, easily prepared from feedstock chemicals, can serve as complement alkylating agents. Importantly, the newly formed carbonyl groups in resulting products provide versatile platform numerous synthetic applications.

Язык: Английский

Процитировано

0

Tunable Rh(III)-Catalyzed C(sp2)–H Bond Functionalization of Aryl Imidates with Cyclic 1,3-Diones: Strategic Use of Directing Groups DOI

E Junnan,

Luohe Wang,

Jing Zeng

и другие.

Organic Letters, Год журнала: 2024, Номер 26(37), С. 7885 - 7890

Опубликована: Сен. 6, 2024

A tunable Rh(III)-catalyzed C(sp

Язык: Английский

Процитировано

1

Cyclic Iodonium Ylide Unlocked Pd-Catalyzed α-Acyloxylation of Cyclic 1,3-Dicarbonyls with Carboxylic Acids DOI
Huanping Xie,

Borong Su,

H. -L. Cui

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Дек. 10, 2024

To date, a general approach for the direct α-acyloxylation of cyclic 1,3-dicarbonyls remains challenging. Herein, we report Pd-catalyzed 1,3-dicarbonyl-derived hypervalent iodine compounds with highly abundant carboxylic acids. Our utilizes commercially available Pd(OAc)

Язык: Английский

Процитировано

1

Bioinspired Synthesis of Phelligridin Analogues via Ru-Catalyzed C–H Activation/[4 + 2] Annulation of Aryl Imidates with Heteroaromatic Iodonium Ylides DOI

Mingdian Liang,

Si-Jing Huang,

Dongyang Zhang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Дек. 16, 2024

The first Ru(II)-catalyzed C–H activation/[4 + 2] annulation of aryl imidates with heteroaromatic iodonium ylides is reported. Our approach features the utilization a commercially available ruthenium catalyst, providing one-step construction phelligridin analogues from easily and nonpreactivated starting materials. developed methodology successfully employed for total synthesis A, significantly streamlining previous multistep synthesis. potential this further demonstrated through modular core structure C/D.

Язык: Английский

Процитировано

0