Substrate-Controlled Electrochemical Reaction of 2-Alkynylbenzamides, Inorganic Sulfites, and Alcohols DOI
Xiaoman Wang, Shanshan Feng, Jiarui Han

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(22), С. 16873 - 16882

Опубликована: Ноя. 6, 2024

Isoindolones constitute a dominant structural class in synthetic and medicinal chemistry. In this research, an electrochemical reaction involving 2-alkynylbenzamides, inorganic sulfites, alcohols was first established to provide sulfonyl ester-substituted 3-hydroxyisoindolinone derivatives moderate good yields with excellent functional group tolerance. When bulky aryl-substituted 2-alkynylbenzamides are utilized as substrates, 3-alkylideneisoindolinones can be selectively generated chemoselectivity. Alkoxysulfonyl radicals derived from the anodic oxidation of sulfite involved transformation.

Язык: Английский

Electrochemical Synthesis of Alkenylsulfonates from Alkynes, NaHSO3 and Alcohols DOI
Xiaoman Wang, Qianqian Chen,

Jinhang Zhou

и другие.

Chinese Journal of Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Ноя. 7, 2024

Comprehensive Summary Alkenylsulfonates are commonly encountered in medicinal chemistry, polymer and organic synthesis. In this research, an electrochemical reaction involving alkynes, NaHSO 3 , alcohols has been developed. This method yields functionalized alkenylsulfonates good with broad functional group tolerance. Mechanism studies indicate that anodic oxidation of inorganic sulfite, radical insertion process, HAT process involved transformation.

Язык: Английский

Процитировано

2

Manganaelectro-Catalyzed Cyclization of o-Aminoarylketones with Ammonia: An Approach to 1,2-Dihydroquinazolines DOI

Qiang Zhong,

Pei-Long Wang, Hui Gao

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Сен. 12, 2024

A manganaelectro-catalyzed cyclization reaction of 2-aminoarylketones with simple alcohols and ammonia under mild conditions is reported for the first time. The cooperative catalysis effectively enhances oxidation primary into aldehydes, thus enabling synthesis substituted 1,2-dihydroquinazolines in good to excellent yields. In addition, utilities this method are highlighted construction biologically active molecules that would otherwise be difficult access through a traditional method.

Язык: Английский

Процитировано

1

Substrate-Controlled Electrochemical Reaction of 2-Alkynylbenzamides, Inorganic Sulfites, and Alcohols DOI
Xiaoman Wang, Shanshan Feng, Jiarui Han

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(22), С. 16873 - 16882

Опубликована: Ноя. 6, 2024

Isoindolones constitute a dominant structural class in synthetic and medicinal chemistry. In this research, an electrochemical reaction involving 2-alkynylbenzamides, inorganic sulfites, alcohols was first established to provide sulfonyl ester-substituted 3-hydroxyisoindolinone derivatives moderate good yields with excellent functional group tolerance. When bulky aryl-substituted 2-alkynylbenzamides are utilized as substrates, 3-alkylideneisoindolinones can be selectively generated chemoselectivity. Alkoxysulfonyl radicals derived from the anodic oxidation of sulfite involved transformation.

Язык: Английский

Процитировано

1