A Noninvasive Nanoeyedrop Therapy for the Inhibition of Uveal Melanoma: Tetrahedral Framework Nucleic Acid–Based Bioswitchable MicroRNA Delivery System DOI
Jiang Zhou,

Yichen Yang,

Ziqi Yue

и другие.

ACS Nano, Год журнала: 2025, Номер unknown

Опубликована: Апрель 10, 2025

Uveal melanoma (UM) is the most prevalent primary intraocular malignancy, exhibiting pronounced invasive characteristics and a dismal prognosis. Conventional therapeutic modalities, including radiotherapy, laser therapy, surgery, are frequently can lead to complications, underscoring need for development of efficacious, safe, noninvasive approaches. This study investigated tetrahedral framework nucleic acid (tFNA)-based bioswitchable microRNA (miRNA) delivery system, designated BiRDS, engineered inhibition UM through use miRNA suppressors via eyedrops. The BiRDS construct exhibited structure, which was small in size, easily synthesizable, stable, biosafe, able efficiently carry miR-30a-5p into cells. Functionally, observed inhibit proliferation, migration, invasion cells while promoting apoptosis miR-30a-5p/E2F7 axis. It noteworthy that nanoeyedrops were penetrate complex ocular barrier structure reach fundus, thereby inhibiting growth xenograft model. As patient-friendly, eyedrop-based not only inhibited without enucleation eyeball but also expected improve patient compliance quality life providing safer alternative drug administration. work substantiates as potential paradigm shift local treatment early UM, facilitating its application treating other diseases therapies.

Язык: Английский

Current Understanding and Translational Prospects of Tetrahedral Framework Nucleic Acids DOI Creative Commons
Junjie Gu,

Jiale Liang,

Taoran Tian

и другие.

JACS Au, Год журнала: 2025, Номер 5(2), С. 486 - 520

Опубликована: Фев. 10, 2025

Tetrahedral framework nucleic acids (tFNAs) represent a promising advancement in acid nanotechnology due to their unique structural properties, high biocompatibility, and multifaceted biomedical applications. Constructed through one-pot annealing method, four single-stranded DNAs self-assemble into stable, three-dimensional tetrahedral nanostructures with enhanced mechanical robustness physiological stability, resisting enzymatic degradation. Their ability permeate mammalian cells without transfection agents, coupled modifiable surfaces, positions tFNAs as versatile carriers for drug gene delivery systems. The tFNA-based platforms exhibit superior therapeutic efficacy, including antioxidative anti-inflammatory effects, alongside efficient cellular uptake tissue penetration. These features underpin role precision medicine, enabling targeted of diverse agents such synthetic compounds, peptides, acids. Additionally, demonstrate significant potential regenerative immune modulation, antibacterial strategies, oncology. By addressing challenges translational integration, stand poised accelerate the development research clinical applications, fostering novel therapies enhancing outcomes across wide spectrum diseases. This Perspective thoroughly details attributes applications critically evaluates tFNAs' potential, outlining inherent implementation exploring solutions these obstacles.

Язык: Английский

Процитировано

2

A Noninvasive Nanoeyedrop Therapy for the Inhibition of Uveal Melanoma: Tetrahedral Framework Nucleic Acid–Based Bioswitchable MicroRNA Delivery System DOI
Jiang Zhou,

Yichen Yang,

Ziqi Yue

и другие.

ACS Nano, Год журнала: 2025, Номер unknown

Опубликована: Апрель 10, 2025

Uveal melanoma (UM) is the most prevalent primary intraocular malignancy, exhibiting pronounced invasive characteristics and a dismal prognosis. Conventional therapeutic modalities, including radiotherapy, laser therapy, surgery, are frequently can lead to complications, underscoring need for development of efficacious, safe, noninvasive approaches. This study investigated tetrahedral framework nucleic acid (tFNA)-based bioswitchable microRNA (miRNA) delivery system, designated BiRDS, engineered inhibition UM through use miRNA suppressors via eyedrops. The BiRDS construct exhibited structure, which was small in size, easily synthesizable, stable, biosafe, able efficiently carry miR-30a-5p into cells. Functionally, observed inhibit proliferation, migration, invasion cells while promoting apoptosis miR-30a-5p/E2F7 axis. It noteworthy that nanoeyedrops were penetrate complex ocular barrier structure reach fundus, thereby inhibiting growth xenograft model. As patient-friendly, eyedrop-based not only inhibited without enucleation eyeball but also expected improve patient compliance quality life providing safer alternative drug administration. work substantiates as potential paradigm shift local treatment early UM, facilitating its application treating other diseases therapies.

Язык: Английский

Процитировано

0