The Emerging Roles of the Stress Epigenetic Reader LEDGF/p75 in Cancer Biology and Therapy Resistance: Mechanisms and Targeting Opportunities DOI Open Access
Greisha L. Ortiz-Hernández,

Evelyn S. Sanchez-Hernández,

Pedro T. Ochoa

и другие.

Cancers, Год журнала: 2024, Номер 16(23), С. 3957 - 3957

Опубликована: Ноя. 26, 2024

The lens epithelium derived growth factor of 75 kD (LEDGF/p75) is a transcription co-activator and epigenetic reader that has emerged as stress oncoprotein in multiple human cancers. Growing evidence indicates it promotes tumor cell survival against certain therapeutic drugs. amino (N)-terminal region LEDGF/p75 contains PWWP domain reads methylated histone marks, critical for recognizing transcriptionally active chromatin sites. Its carboxyl (C)-terminus an integrase binding (IBD) serves the site HIV-1 oncogenic factors. Acting hubs protein-protein interactions, both domains facilitate tethering factors regulators to regulate mRNA splicing, promote DNA repair, enhance expression cancer-related genes contribute aggressiveness chemoresistance. This review summarizes our current knowledge emerging roles cancer biology therapy resistance discusses its potential novel oncotherapeutic target combinatorial treatments.

Язык: Английский

Oxidative-Stress-Mediated Epigenetic Dysregulation in Spermatogenesis: Implications for Male Infertility and Offspring Health DOI Open Access
Aris Kaltsas,

Eleftheria Markou,

Maria-Anna Kyrgiafini

и другие.

Genes, Год журнала: 2025, Номер 16(1), С. 93 - 93

Опубликована: Янв. 17, 2025

Male reproductive health is governed by an intricate interplay of genetic, epigenetic, and environmental factors. Epigenetic mechanisms—encompassing DNA methylation, histone modifications, non-coding RNA activity—are crucial both for spermatogenesis sperm maturation. However, oxidative stress, driven excessive reactive oxygen species, disrupts these processes, leading to impaired function male infertility. This disruption extends epigenetic resulting in abnormal gene expression chromatin remodeling that compromise genomic integrity fertilization potential. Importantly, oxidative-stress-induced alterations can be inherited, affecting the fertility offspring future generations. review investigates how stress influences regulation reproduction modifying RNAs, ultimately compromising spermatogenesis. Additionally, it discusses transgenerational implications disruptions their potential role hereditary infertility disease predisposition. Understanding mechanisms vital developing therapeutic strategies mitigate damage restore homeostasis germline. By integrating insights from molecular, clinical, research, this work emphasizes need targeted interventions enhance prevent adverse outcomes progeny. Furthermore, elucidating dose–response relationships between changes remains a critical research priority, informing personalized diagnostics interventions. In context, studies should adopt standardized markers damage, robust clinical trials, multi-omic approaches capture complexity Such rigorous investigations will reduce risk disorders optimize outcomes.

Язык: Английский

Процитировано

1

Lyophilized and Oven-Dried Manilkara zapota Extracts: Characterization and In Vitro, In Vivo, and In Silico Analyses DOI Creative Commons

María Fernanda Rivas-Gastélum,

Patricia Ariadna Galindo-Castillo,

Juan Esparza-Sánchez

и другие.

Plants, Год журнала: 2025, Номер 14(2), С. 216 - 216

Опубликована: Янв. 14, 2025

In this work, extracts from the pulp, peel, and seed of Manilkara zapota were obtained via lyophilization oven drying. Bromatological analyses performed to investigate variabilities in nutritional content fruits after nine post-harvest days. The phytochemical was assessed by gas chromatography flame ionization detector (GC-FID), their biological performance studied using vitro antibacterial antioxidant assays (DPPH ABTS) vivo toxicity models. Molecular docking implemented evaluate interaction between polar compounds chicozapote with receptors involved pathogenesis bacterial strains. Results revealed that water or soluble solids did not vary post-harvest. It demonstrated oven-drying approaches influenced insoluble, total dietary fiber digestible carbohydrates among samples. According GC-FID analysis, it observed methods also altered myristic pentadecanoic acids extracts. noted activities weak due MIC (>1000 μg/mL) IC50 (>2000 values. Still, poor against Artemia salina nauplii. silico evaluation unveiled M. possess a high binding affinity towards DNA gyrase B cultured This study expands scientific evidence regarding influence distinct extraction on nutraceutical native importance considering additional enhance bioactivities.

Язык: Английский

Процитировано

0

Predictive Value of STC2 Gene Expression in Chemotherapy Response in Breast Cancer DOI Creative Commons
Juan P. Muñoz, Nicolás Lampe

Pharmaceuticals, Год журнала: 2025, Номер 18(2), С. 235 - 235

Опубликована: Фев. 8, 2025

Background: Breast cancer is the most commonly diagnosed among women, and resistance to chemotherapy presents a significant challenge in its treatment. Stanniocalcin-2 (STC2), glycoprotein involved calcium homeostasis cellular stress responses, frequently overexpressed various human cancers. Despite critical role adaptation stress, potential of STC2 as biomarker for predicting response has not been evaluated. This study aimed assess predictive breast cancer. Methods: We utilized publicly available databases characterize expression patients relapse-free survival (RFS). Moreover, we evaluated treatment responses subjected chemotherapy, correlating their outcomes with levels determine biomarker. Finally, cell lines following exposure doxorubicin (Dox), primary anthracycline used they were contrasted dataset. Results: The analysis showed that significantly luminal A cancer, where it linked genetic amplifications. High was associated improved RFS ER-positive but correlated worse ER-negative cases. Furthermore, grade II patients, higher better response, while poorer response. downregulation observed Dox Conclusions: These findings suggest serves patients.

Язык: Английский

Процитировано

0

The Emerging Roles of the Stress Epigenetic Reader LEDGF/p75 in Cancer Biology and Therapy Resistance: Mechanisms and Targeting Opportunities DOI Open Access
Greisha L. Ortiz-Hernández,

Evelyn S. Sanchez-Hernández,

Pedro T. Ochoa

и другие.

Cancers, Год журнала: 2024, Номер 16(23), С. 3957 - 3957

Опубликована: Ноя. 26, 2024

The lens epithelium derived growth factor of 75 kD (LEDGF/p75) is a transcription co-activator and epigenetic reader that has emerged as stress oncoprotein in multiple human cancers. Growing evidence indicates it promotes tumor cell survival against certain therapeutic drugs. amino (N)-terminal region LEDGF/p75 contains PWWP domain reads methylated histone marks, critical for recognizing transcriptionally active chromatin sites. Its carboxyl (C)-terminus an integrase binding (IBD) serves the site HIV-1 oncogenic factors. Acting hubs protein-protein interactions, both domains facilitate tethering factors regulators to regulate mRNA splicing, promote DNA repair, enhance expression cancer-related genes contribute aggressiveness chemoresistance. This review summarizes our current knowledge emerging roles cancer biology therapy resistance discusses its potential novel oncotherapeutic target combinatorial treatments.

Язык: Английский

Процитировано

0