Synthesis and Evaluation of Polymer-Drug Conjugates as Potential Antioxidants and Cholinesterase Inhibitors for Neurodegenerative Diseases DOI Creative Commons
Nuruddin Mahadik, Gemma A. Barron, Paul Kong Thoo Lin

и другие.

Chemistry of Materials, Год журнала: 2024, Номер 36(21), С. 10514 - 10527

Опубликована: Окт. 23, 2024

Polymer-drug conjugates (PDCs) may offer improved water-solubility and in vitro activity of potential antioxidant cholinesterase (ChE) inhibitor drugs compared to the alone. Conjugation these water-soluble polymers could increase their therapeutic efficacy. Vanillin was conjugated poly(allylamine hydrochloride) (NM10 NM15) naphthalimidohexylamine (HEXNAP) poly(acrylic acid) (N5 N10). The inhibitory activities novel PDCs were evaluated with those respective starting materials. Additionally, silico molecular modeling studies conducted explore mechanisms conjugates. NM15 (unadjusted adjusted value) showed significantly enhanced (p ≤ 0.0001) vanillin. value N5 HEXNAP against acetylcholinesterase (AChE) butyrylcholinesterase (BuChE) 0.0001). Kinetic revealed that a competitive interacted active sites human enzymes. identified as lead based on activity, respectively. Overall, this work demonstrates use treatment options for neurodegenerative diseases.

Язык: Английский

Polymer–drug and polymer–protein conjugated nanocarriers: Design, drug delivery, imaging, therapy, and clinical applications DOI
Haochen Guo, Peng Mi

Wiley Interdisciplinary Reviews Nanomedicine and Nanobiotechnology, Год журнала: 2024, Номер 16(4)

Опубликована: Июль 1, 2024

Polymer-drug conjugates and polymer-protein have been pivotal in the realm of drug delivery systems for over half a century. These polymeric drugs are characterized by conjugation therapeutic molecules or functional moieties to polymers, enabling range benefits including extended circulation times, targeted delivery, controlled release, decreased immunogenicity. This review delves into recent advancements challenges clinical translations preclinical studies polymer-drug conjugates. The design principles functionalization strategies crucial development these were explored followed structural properties characteristics various polymer carriers. also identifies significant obstacles translation provides insights directions their future development. article is categorized under: Therapeutic Approaches Drug Discovery > Nanomedicine Oncologic Disease.

Язык: Английский

Процитировано

4

Hydroxyapatite–polymer nanocomposites for drug delivery applications: A mini review DOI Creative Commons

Farnaz Behmagham,

Shahad Mohammed Dhiaa,

Abbas Hameed Abdul Hussein

и другие.

European Journal of Medicinal Chemistry Reports, Год журнала: 2024, Номер unknown, С. 100231 - 100231

Опубликована: Окт. 1, 2024

Язык: Английский

Процитировано

4

Clinical Applications of Targeted Nanomaterials DOI Creative Commons

Ankesh Kumar,

SK Shahvej,

Pankaj Yadav

и другие.

Pharmaceutics, Год журнала: 2025, Номер 17(3), С. 379 - 379

Опубликована: Март 17, 2025

Targeted nanomaterials are at the forefront of advancements in nanomedicine due to their unique and versatile properties. These include nanoscale size, shape, surface chemistry, mechanical flexibility, fluorescence, optical behavior, magnetic electronic characteristics, as well biocompatibility biodegradability. attributes enable application across diverse fields, including drug delivery. This review explores fundamental characteristics emphasizes importance clinical applications. It further delves into methodologies for nanoparticle programming alongside discussions on trials case studies. We discussed some promising nanomaterials, such polymeric nanoparticles, carbon-based metallic role biomedical underscores significant translating applications highlights potential these innovative approaches revolutionizing medical field.

Язык: Английский

Процитировано

0

Synthesis and Evaluation of Polymer-Drug Conjugates as Potential Antioxidants and Cholinesterase Inhibitors for Neurodegenerative Diseases DOI Creative Commons
Nuruddin Mahadik, Gemma A. Barron, Paul Kong Thoo Lin

и другие.

Chemistry of Materials, Год журнала: 2024, Номер 36(21), С. 10514 - 10527

Опубликована: Окт. 23, 2024

Polymer-drug conjugates (PDCs) may offer improved water-solubility and in vitro activity of potential antioxidant cholinesterase (ChE) inhibitor drugs compared to the alone. Conjugation these water-soluble polymers could increase their therapeutic efficacy. Vanillin was conjugated poly(allylamine hydrochloride) (NM10 NM15) naphthalimidohexylamine (HEXNAP) poly(acrylic acid) (N5 N10). The inhibitory activities novel PDCs were evaluated with those respective starting materials. Additionally, silico molecular modeling studies conducted explore mechanisms conjugates. NM15 (unadjusted adjusted value) showed significantly enhanced (p ≤ 0.0001) vanillin. value N5 HEXNAP against acetylcholinesterase (AChE) butyrylcholinesterase (BuChE) 0.0001). Kinetic revealed that a competitive interacted active sites human enzymes. identified as lead based on activity, respectively. Overall, this work demonstrates use treatment options for neurodegenerative diseases.

Язык: Английский

Процитировано

0