The Future of Electro-organic Synthesis in Drug Discovery and Early Development DOI Creative Commons
Hamish R. Stephen, Johannes L. Röckl

ACS Organic & Inorganic Au, Год журнала: 2024, Номер 4(6), С. 571 - 578

Опубликована: Ноя. 16, 2024

Electro-organic chemistry presents a promising frontier in drug discovery and early development, facilitating novel reactivity aligned with green principles. Despite this, electrochemistry is not widely used as synthesis manufacturing tool or development. This overview seeks to identify key areas that require additional research make synthetic more accessible chemists development provide potential solutions. includes expanding the reaction scope, simplifying rapid scale-up, developing electrode materials, improving knowledge transfer aid reproducibility increase awareness of electrochemistry. The integration electro-organic into holds enable efficient, sustainable routes toward future medicines faster than ever.

Язык: Английский

Recent advances on electrochemical generation of sulfonyl radical triggered cyclization of alkene/alkynes DOI

Jiaqing Shao,

Jiang Liu, Haibo Mei

и другие.

Tetrahedron, Год журнала: 2025, Номер 173, С. 134467 - 134467

Опубликована: Янв. 12, 2025

Язык: Английский

Процитировано

1

Flow Electroreductive Nickel‐Catalyzed Cyclopropanation of Alkenes Using gem‐Dichloroalkanes DOI Creative Commons
Morgan Regnier, Clara Vega, Dimitris I. Ioannou

и другие.

Angewandte Chemie International Edition, Год журнала: 2025, Номер unknown

Опубликована: Янв. 31, 2025

Abstract Cyclopropanes are valuable motifs in organic synthesis, widely featured pharmaceuticals and functional materials. Herein, we report an efficient electrochemical methodology for the cyclopropanation of alkenes, leveraging a nickel‐catalyzed process continuous‐flow. The developed protocol demonstrates broad substrate scope, accommodating both electron‐rich electron‐poor alkenes with high group tolerance. Beyond dichloromethane as feedstock methylene source, enables synthesis methylated, deuterated, chloro‐substituted cyclopropanes. Mechanistic investigations suggest electro‐generation nickel carbene key intermediate. Notably, reaction operates under ambient conditions, tolerates air moisture, achieves scalability through continuous‐flow technology, offering straightforward route to multi‐gram quantities enhanced throughput.

Язык: Английский

Процитировано

0

Tunable selective electrochemical selenization of tetrahydroquinolines with diselenides DOI

Lan-Xi Zong,

Yu‐Fang Tan,

Yu-Hao Yang

и другие.

Green Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Янв. 1, 2025

An electrochemical method for selenylating tetrahydroquinolines with diselenides is presented. By tuning reaction conditions, C-3 selenylated quinolines and C-6 can be selectively synthesized excellent outcomes.

Язык: Английский

Процитировано

0

A Scalable Flow Electrolysis of Heterogeneous Mixtures Using a Rotating Cylinder Electrode Reactor: Access to a Chiral Iminophosphorane DOI

Felix Xu,

Longrui Chen, Dan Lehnherr

и другие.

Organic Process Research & Development, Год журнала: 2025, Номер unknown

Опубликована: Фев. 27, 2025

We report the application of rotating cylinder electrode (RCE) reactors for electrolysis heterogeneous reactions in batch and recirculating flow. A scalable method synthesis an N-cyano iminophosphorane ligand RCE reactor is also reported. In development this process, a graphite felt attached to inner impervious was used as anode, outer stainless steel wall cathode. The reaction first evaluated using small optimize spinning rate, supporting electrolyte, current density. optimal condition then scaled up medium-sized with modifications adapt it flow process. electrosynthesis demonstrated 100 g scale, impact temperature investigated. Finally, operationally simple direct crystallization water antisolvent provided chiral 74% isolated yield on scale from commercially available (S)-BINAP bis(trimethylsilyl)carbodiimide.

Язык: Английский

Процитировано

0

Microfluidic Technology: A New Strategy for Controllable Synthesis of Metal Nanomaterials DOI Creative Commons
Dongtang Zhang, Shuang Jia, Jin Zhao

и другие.

ChemElectroChem, Год журнала: 2025, Номер unknown

Опубликована: Март 7, 2025

Abstract Microfluidic technology has exhibited remarkable potential and significance in the precise preparation of multifunctional nanomaterials. Thanks to its small reaction volume superior hydrodynamic control, this emerged as an essential tool for synthesizing nanomaterials with precisely tunable microstructures morphologies. This paper reviews latest advancements controllable synthesis metal nano‐electrocatalysts utilizing microfluidic technology. Firstly, it systematically elucidates fundamental principles distinctive parameter control strategies. Subsequently, delves deeply into mechanism enhancement process nanoparticles environment. Through analysis specific cases, extensive application prospects advantages system have been further elucidated. Finally, summarizes looks forward challenges future development directions that faces nano‐electrocatalysts. review aims provide valuable insights morphology design technological innovation electrocatalysts.

Язык: Английский

Процитировано

0

Feed and Bleed Operating Mode for Electrochemical Flow Cells: Challenges, Solutions and Practical Insights DOI Creative Commons
Jonas Baessler, Malte Wehner, Mojtaba Mohseni

и другие.

ChemElectroChem, Год журнала: 2025, Номер unknown

Опубликована: Март 29, 2025

Abstract Electrochemical processes offer promising routes to defossilize the chemical industry by integrating low‐carbon electricity. However, bridging gap between lab‐scale experimental studies and pilot‐scale industrial applications is still challenging: Lab‐scale electrochemical flow cells typically operate in batch or single‐pass mode, with each mode facing limitations regarding steady‐state operation at industrially relevant conditions. This work introduces “feed bleed” operating continuous exchange of a recirculated electrolyte stream, which enables versatile operation. The compared We develop mathematical model for validate experimentally. Additionally, this 3D‐printed phase separator coupled separate gas from liquid stream. Batch, single‐pass, are demonstrated methanol oxidation formate 200 mA/cm 2 25 cm cell. provides an comparison concerning product/reactant concentration, conversion, Faraday efficiency. highlights characteristics electrosynthesis chemicals, showcasing unique feed bleed industrially‐relevant conditions high product concentration.

Язык: Английский

Процитировано

0

Electrochemical Access to Difluoromethyl Groups: An Overview of Scope, Mechanisms, and Challenges DOI
Seonyoung Kim, Hyunwoo Kim

ACS Catalysis, Год журнала: 2025, Номер unknown, С. 6826 - 6851

Опубликована: Апрель 14, 2025

Язык: Английский

Процитировано

0

Nitrogen-Based Organofluorine Functional Molecules: Synthesis and Applications DOI
Shuai Liu, Jun Zhou, Lu Yu

и другие.

Chemical Reviews, Год журнала: 2025, Номер unknown

Опубликована: Апрель 22, 2025

Fluorine and nitrogen form a successful partnership in organic synthesis, medicinal chemistry, material sciences. Although fluorine-nitrogen chemistry has long rich history, this field received increasing interest made remarkable progress over the past two decades, driven by recent advancements transition metal organocatalysis photochemistry. This review, emphasizing contributions from 2015 to 2023, aims update state of art synthesis applications nitrogen-based organofluorine functional molecules chemistry. In dedicated sections, we first focus on fluorine-containing reagents organized according type groups attached nitrogen, including N-F, N-RF, N-SRF, N-ORF. review also covers nitrogen-linked building blocks, catalysts, pharmaceuticals, agrochemicals, underlining these components' broad applicability growing importance modern

Язык: Английский

Процитировано

0

The Future of Electro-organic Synthesis in Drug Discovery and Early Development DOI Creative Commons
Hamish R. Stephen, Johannes L. Röckl

ACS Organic & Inorganic Au, Год журнала: 2024, Номер 4(6), С. 571 - 578

Опубликована: Ноя. 16, 2024

Electro-organic chemistry presents a promising frontier in drug discovery and early development, facilitating novel reactivity aligned with green principles. Despite this, electrochemistry is not widely used as synthesis manufacturing tool or development. This overview seeks to identify key areas that require additional research make synthetic more accessible chemists development provide potential solutions. includes expanding the reaction scope, simplifying rapid scale-up, developing electrode materials, improving knowledge transfer aid reproducibility increase awareness of electrochemistry. The integration electro-organic into holds enable efficient, sustainable routes toward future medicines faster than ever.

Язык: Английский

Процитировано

0