Towards accurate, force field independent conformational ensembles of intrinsically disordered proteins DOI Creative Commons

Kaushik Borthakur,

Thomas R. Sisk, Francesco Paolo Panei

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2024, Номер unknown

Опубликована: Окт. 5, 2024

Abstract Determining accurate atomic resolution conformational ensembles of intrinsically disordered proteins (IDPs) is extremely challenging. Molecular dynamics (MD) simulations provide atomistic IDPs, but their accuracy highly dependent on the quality physical models, or force fields, used. Here, we demonstrate how to determine IDPs by integrating all-atom MD with experimental data from nuclear magnetic resonance (NMR) spectroscopy and small-angle x-ray scattering (SAXS) a simple, robust fully automated maximum entropy reweighting procedure. We that when this approach applied sufficient data, IDP derived different fields converge similar distributions. The procedure presented here facilitates integration extensive datasets enables calculation accurate, force-field independent IDPs.

Язык: Английский

Simulation-based inference of single-molecule experiments DOI Creative Commons
Lars Dingeldein, Pilar Cossio, Roberto Covino

и другие.

Current Opinion in Structural Biology, Год журнала: 2025, Номер 91, С. 102988 - 102988

Опубликована: Фев. 7, 2025

Язык: Английский

Процитировано

1

MDRefine: A Python package for refining molecular dynamics trajectories with experimental data DOI Creative Commons
Ivan Gilardoni, Valerio Piomponi, Thorben Fröhlking

и другие.

The Journal of Chemical Physics, Год журнала: 2025, Номер 162(19)

Опубликована: Май 15, 2025

Molecular dynamics (MD) simulations play a crucial role in resolving the underlying conformational of molecular systems. However, their capability to correctly reproduce and predict agreement with experiments is limited by accuracy force-field model. This can be improved refining structural ensembles or parameters. Furthermore, discrepancies experimental data due imprecise forward models, namely, functions mapping simulated structures observables. Here, we introduce MDRefine, Python package aimed at implementing refinement ensemble, force field, and/or model comparing MD-generated trajectories data. The software consists several tools that employed separately from each other combined together different ways, providing seamless interpolation between these three types refinement. We use some benchmark cases show approach superior applied refinements. MDRefine has been released as an open-source under LGPLv2+ license. Source code, documentation, examples are available https://pypi.org/project/MDRefine https://github.com/bussilab/MDRefine.

Язык: Английский

Процитировано

0

Model Selection Using Replica Averaging with Bayesian Inference of Conformational Populations DOI
Robert M. Raddi, Tim Marshall, Ge Yunhui

и другие.

Journal of Chemical Theory and Computation, Год журнала: 2025, Номер unknown

Опубликована: Июнь 2, 2025

Bayesian Inference of Conformational Populations (BICePs) is a reweighting algorithm that reconciles simulated ensembles with sparse and/or noisy observables by sampling the full posterior distribution conformational populations in presence experimental restraints. By modifying BICePs to use replica-averaging its forward model, becomes similar other MaxEnt approaches, but significant advantages (1) being able sample over uncertainties due random and systematic error, improved likelihoods deal outliers, (2) having an objective score for model selection, free energy-like quantity called score. To demonstrate power our approach, we used reweight mini-protein chignolin nine different force fields TIP3P water, using set 158 measurements (139 NOE distances, 13 chemical shifts, 6 vicinal J-coupling constants HN Hα). In all cases, reweighted favor correctly folded conformation. The score, which reports energy "turning on" along restraints, provides metric evaluate each field. For tested (A14SB, A99SB-ildn, A99, A99SBnmr1-ildn, A99SB, C22star, C27, C36, OPLS-aa), obtain results consistent previous work conventional χ2 selection small polypeptides ubiquitin (J. Chem. Theory Comput., 2012, 8, 1409-1414). These suggest powerful role future applications requiring ensemble selection.

Язык: Английский

Процитировано

0

Towards accurate, force field independent conformational ensembles of intrinsically disordered proteins DOI Creative Commons

Kaushik Borthakur,

Thomas R. Sisk, Francesco Paolo Panei

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2024, Номер unknown

Опубликована: Окт. 5, 2024

Abstract Determining accurate atomic resolution conformational ensembles of intrinsically disordered proteins (IDPs) is extremely challenging. Molecular dynamics (MD) simulations provide atomistic IDPs, but their accuracy highly dependent on the quality physical models, or force fields, used. Here, we demonstrate how to determine IDPs by integrating all-atom MD with experimental data from nuclear magnetic resonance (NMR) spectroscopy and small-angle x-ray scattering (SAXS) a simple, robust fully automated maximum entropy reweighting procedure. We that when this approach applied sufficient data, IDP derived different fields converge similar distributions. The procedure presented here facilitates integration extensive datasets enables calculation accurate, force-field independent IDPs.

Язык: Английский

Процитировано

2