Industrializing yeast as a drug repurposing platform for inherited metabolic diseases DOI Creative Commons
Mathuravani A. Thevandavakkam,

Natalie E. Long,

Briannna M. Roel

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2024, Номер unknown

Опубликована: Авг. 26, 2024

Summary The development of therapies for rare diseases, particularly inherited metabolic disorders (IMDs), faces significant challenges due to the high cost and lengthy timelines involved. This study presents a yeast-based platform drug repurposing that capitalizes on remarkable similarity between yeast human cellular pathways. enables rapid, cost-effective screening potential therapeutic compounds offering quick turnaround compared traditional processes. Utilizing TargetMol library comprising ∼50% nutraceuticals, our pipeline accelerates translation promising hits into patient observational studies in as little 6 months. We demonstrate efficacy this through three case context IMDs, showcasing its uncover novel treatments reduce time expense associated with bringing patients diseases.

Язык: Английский

Dysregulation of serotonergic neurotransmission in Parkinson disease: A key duet DOI Creative Commons
Manal M. Khowdiary, Hayder M. Al‐kuraishy, Ali I. Al‐Gareeb

и другие.

European Journal of Pharmacology, Год журнала: 2025, Номер unknown, С. 177419 - 177419

Опубликована: Фев. 1, 2025

Язык: Английский

Процитировано

0

Unravelling the Proteinopathic Engagement of α-Synuclein, Tau, and Amyloid Beta in Parkinson’s Disease: Mitochondrial Collapse as a Pivotal Driver of Neurodegeneration DOI
Trilochan Sahoo, Jagdish Chand,

Amarjith Thiyyar Kandy

и другие.

Neurochemical Research, Год журнала: 2025, Номер 50(3)

Опубликована: Апрель 16, 2025

Язык: Английский

Процитировано

0

Clinical study to investigate the adjuvant role of Pentoxifylline in patients with Parkinson's disease: A randomized controlled study DOI

M O Khrieba,

Sahar K. Hegazy,

Wessam Fathi Mohammed

и другие.

International Immunopharmacology, Год журнала: 2025, Номер 156, С. 114689 - 114689

Опубликована: Апрель 19, 2025

Язык: Английский

Процитировано

0

Cyclin‐dependent kinase 5 (CDK5) inhibitors in Parkinson disease DOI Creative Commons
Mohammed Alrouji,

Haydar M. Al‐kuraishy,

Ali I. Al‐Gareeb

и другие.

Journal of Cellular and Molecular Medicine, Год журнала: 2024, Номер 28(11)

Опубликована: Июнь 1, 2024

Abstract Cyclin‐dependent kinase 5 (Cdk5) is a protein expressed in postmitotic neurons the central nervous system (CNS). Cdk5 activated by p35 and p39 which are neuron regulatory subunits. Cdk5/p35 complex calpain protease to form has neuroprotective effect regulating synaptic plasticity memory functions. However, exaggerated implicated different types of neurodegenerative diseases including Parkinson disease (PD). Therefore, modulation signalling may mitigate PD neuropathology. aim present review was discuss critical role pathogenesis PD, how inhibitors effectual management PD. In conclusion, overactivated involved development neurodegeneration, Cdk5/calpain such as statins, metformin, fenofibrates rosiglitazone can attenuate progression

Язык: Английский

Процитировано

3

Industrializing yeast as a drug repurposing platform for inherited metabolic diseases DOI Creative Commons
Mathuravani A. Thevandavakkam,

Natalie E. Long,

Briannna M. Roel

и другие.

bioRxiv (Cold Spring Harbor Laboratory), Год журнала: 2024, Номер unknown

Опубликована: Авг. 26, 2024

Summary The development of therapies for rare diseases, particularly inherited metabolic disorders (IMDs), faces significant challenges due to the high cost and lengthy timelines involved. This study presents a yeast-based platform drug repurposing that capitalizes on remarkable similarity between yeast human cellular pathways. enables rapid, cost-effective screening potential therapeutic compounds offering quick turnaround compared traditional processes. Utilizing TargetMol library comprising ∼50% nutraceuticals, our pipeline accelerates translation promising hits into patient observational studies in as little 6 months. We demonstrate efficacy this through three case context IMDs, showcasing its uncover novel treatments reduce time expense associated with bringing patients diseases.

Язык: Английский

Процитировано

0