
Опубликована: Май 22, 2024
We report herein our studies on the direct photoactivation of carbonyl cyclopropanes to give biradical intermediates, leading selective cleavage more substituted carbon-carbon bond. Depending substrate structure, extended alkenes were isolated or directly reacted in a photo-Nazarov process bicyclic products. Based these results, unified reductive ring-opening reaction was developed by using diphenyl disulfide as HAT reagent. By performing sequential cyclopropanation/selective ring opening reaction, we achieved CH2 insertion into alpha,beta- bond both acyclic and cyclic unsaturated compounds. Our protocol therefore provides further tool for framework-editing carbocycles, complementing recent progress "skeletal editing" strategies.
Язык: Английский