Double Duty: SGLT2 Inhibitors as Cardioprotective and Anticancer Allies DOI Creative Commons
Linda Piras,

Michela Zuccanti,

Giacomo Tini

и другие.

Hearts, Год журнала: 2024, Номер 5(4), С. 529 - 546

Опубликована: Ноя. 1, 2024

Sodium glucose cotransporter-2 inhibitors (SGLT2i), originally developed for type II diabetes mellitus, have recently been approved the treatment of heart failure in both diabetic and non-diabetic patients due to their significant cardiovascular benefits. Beyond established role management, current research is exploring potential applications SGLT2 field cardio-oncology. This interest driven by dual possible benefits: cardioprotection against adverse effects antitumor therapies inherent properties. Patients affected cancer often face challenge managing toxicity induced antineoplastic treatments. shown promise mitigating toxicities, thereby enhancing health these patients. Additionally, emerging evidence suggests that may possess direct effects, further contributing therapeutic oncology. review aims provide a comprehensive overview molecular mechanisms through which exert cardioprotective effects. Furthermore, we will examine body supporting use cardio-oncology setting.

Язык: Английский

Atherosclerosis and the Bidirectional Relationship Between Cancer and Cardiovascular Disease: From Bench to Bedside, Part 2 Management DOI Open Access

Giuseppina Gallucci,

Mario Larocca, Alessandro Navazio

и другие.

International Journal of Molecular Sciences, Год журнала: 2025, Номер 26(1), С. 334 - 334

Опубликована: Янв. 2, 2025

The first part of this review highlighted the evolving landscape atherosclerosis, noting emerging cardiometabolic risk factors, growing impact exposomes, and social determinants health. prominent role atherosclerosis in bidirectional relationship between cardiovascular disease cancer was also discussed. In second part, we examine complex interplay multimorbid cardio-oncologic patients, harmful environments that lend a “syndemic” nature to these chronic diseases. We summarize management strategies targeting disordered factors mitigate explore molecular mechanisms enabling more tailored therapies. Importantly, emphasize early interception through multifactorial interventions detect subclinical signs (via biomarkers imaging) treat modifiable prevent clinical events. A concerted preventive effort—referred by some as “preventome”—is essential reduce burden atherosclerosis-driven diseases, shifting from mere proactive promotion “chronic health”.

Язык: Английский

Процитировано

1

SGLT2 inhibitors for prevention and management of cancer treatment-related cardiovascular toxicity: a review of potential mechanisms and clinical insights DOI Creative Commons

Carl Simela,

John M. Walker, Arjun K. Ghosh

и другие.

Cardio-Oncology, Год журнала: 2025, Номер 11(1)

Опубликована: Фев. 11, 2025

Abstract More evidence-based strategies are needed for preventing and managing cancer treatment-related cardiovascular toxicity (CTR-CVT). Owing to the growing body of evidence supporting their cardioprotective role in several cardiac injury scenarios, sodium-glucose cotransporter 2 inhibitors (SGLT2i) may be beneficial treating CTR-CVT. In October 2024, a search was conducted PubMed database review full studies investigating SGLT2i against We identified 44 published/pre-print 3 ongoing randomised controlled trial across eight types treatment (anthracyclines, platinum-containing therapy, immune checkpoint inhibitors, HER2-targeted therapies, kinase androgen deprivation multiple myeloma therapies 5-fluorouracil). Most used animal models focussed on primary prevention. 43 found some effect CTR-CVT, which cases included ejection fraction decline aberrations electrophysiological parameters. Some also observed effects mortality. A central triad anti-inflammatory, anti-oxidative anti-apoptotic mechanisms likely underlie SGLT2i-mediated cardioprotection Overall, this research suggests that promising candidate CTR-CVT either as monotherapy or combination with other drugs. However, literature is limited no prospective trials prevention management exist most existing human retrospective data based diabetic populations. Future work must focus addressing these limitations current literature.

Язык: Английский

Процитировано

0

Cardioprotective Effects of Dapagliflozin and Trimetazidine on Doxorubicin-Induced Cardiotoxicity in Streptozotocin-Induced Type 1 Diabetic Rats via Endoplasmic Reticulum Stress DOI Open Access
Muhammed Mürsel Öğütveren, Ömer Şatıroğlu, Zülkar Özden

и другие.

Journal of Clinical Medicine, Год журнала: 2025, Номер 14(4), С. 1315 - 1315

Опубликована: Фев. 16, 2025

Background/Objectives: Diabetic cardiomyopathy is a distinct myocardial dysfunction characterized by structural and functional changes in the heart that occur diabetic patients independently of coronary artery disease or hypertension. It closely associated with oxidative stress, inflammation, mitochondrial dysfunction, endoplasmic reticulum (ER) contributes to progressive cardiac damage. This study aimed evaluate cardioprotective effects dapagliflozin (DAPA) trimetazidine (TMZ) rat model doxorubicin-induced streptozotocin-induced diabetes, focusing on their potential mechanisms related ER stress. Methods: A total 48 Sprague Dawley rats aged 6-8 weeks were randomly distributed equally into six cages. The diabetes was induced intraperitoneal administration streptozotocin (STZ) blood glucose levels above 250 mg/dL considered diabetic. For those cardiotoxicity injection 5 mg/kg/week doxorubicin (DOXO) for 4 weeks. After cumulative dose 20 mg/kg doxorubicin, week break given, followed TMZ (10 mg/kg) and/or DAPA treatment groups. Results: STZ caused significant degeneration cardiomyocytes. With addition DOXO (STZ + DOXO), cardiomyocyte became more severe. When groups histopathologically evaluated based parameters degenerative cardiomyocytes, vascular congestion, edema, it shown both DAPA, whether applied alone combination, reduced damage tissue. Both damage, combination provided lowest level through stress pathway reducing GRP 78 CHOP positivity. Conclusions: reduce have protective against diabetic-induced cardiotoxicity. Combination therapy found be effective than alleviating appears carry cell individuals diabetes.

Язык: Английский

Процитировано

0

Effects of empagliflozin and dapagliflozin on serum humanin, MOTS-c levels, nitrosative stress, and ferroptosis parameters in diabetic patients with heart failure DOI

Hatice Asil,

Abdullah T. Demiryürek, İrfan Veysel Düzen

и другие.

European Journal of Pharmacology, Год журнала: 2024, Номер 982, С. 176934 - 176934

Опубликована: Авг. 23, 2024

Язык: Английский

Процитировано

2

SNX3 Promotes Doxorubicin-Induced Cardiomyopathy by Regulating GPX4-Mediated Ferroptosis DOI Creative Commons
Shuai Huang,

Fan Zou,

Hao Zhou

и другие.

International Journal of Medical Sciences, Год журнала: 2024, Номер 21(9), С. 1629 - 1639

Опубликована: Янв. 1, 2024

The complete molecular mechanism underlying doxorubicin-induced cardiomyopathy remains incompletely elucidated. In this investigation, we engineered mice with cardiomyocyte-specific

Язык: Английский

Процитировано

0

Glucagon-like Peptide 1 Receptor Agonists in Cardio-Oncology: Pathophysiology of Cardiometabolic Outcomes in Cancer Patients DOI Open Access
Vincenzo Quagliariello,

Maria Laura Canale,

Irma Bisceglia

и другие.

International Journal of Molecular Sciences, Год журнала: 2024, Номер 25(20), С. 11299 - 11299

Опубликована: Окт. 21, 2024

Cancer patients, especially long cancer survivors, are exposed to several cardio-metabolic diseases, including diabetes, heart failure, and atherosclerosis, which increase their risk of cardiovascular mortality. Therapy with glucagon-like peptide 1 (GLP1) receptor agonists demonstrated beneficial effects, atherosclerosis failure prevention. Cardiovascular outcome trials (CVOTs) suggest that GLP-1 RA could exert cardiorenal benefits systemic anti-inflammatory effects in patients type-2 diabetes through the activation cAMP PI3K/AkT pathways inhibition NLRP-3 MyD88. In this narrative review, we highlight biochemical properties a deep analysis clinical preclinical evidence primary prevention cardiomyopathies. The overall picture review encourages study as potential strategy against atherosclerosis.

Язык: Английский

Процитировано

0

Bibliometric and visual analysis of SGLT2 inhibitors in cardiovascular diseases DOI Creative Commons

Rongfang Pan,

Yuqing He,

Wan Melisandre

и другие.

Frontiers in Pharmacology, Год журнала: 2024, Номер 15

Опубликована: Окт. 30, 2024

Cardiovascular diseases (CVD) pose a significant threat to human health due their high mortality and morbidity rates. Despite advances in treatments, the prevalence impact of cardiovascular disease continue increase. Sodium-glucose transporter 2 inhibitors (SGLT2i), initially approved for treatment type diabetes, have important research value promising applications reducing CVD risk, especially heart failure (HF) atherosclerosis patients with (ASCVD). This study aims comprehensively review latest progress, trends, cutting-edge hot spots, future development directions SGLT2i field through bibliometric analysis.

Язык: Английский

Процитировано

0

Double Duty: SGLT2 Inhibitors as Cardioprotective and Anticancer Allies DOI Creative Commons
Linda Piras,

Michela Zuccanti,

Giacomo Tini

и другие.

Hearts, Год журнала: 2024, Номер 5(4), С. 529 - 546

Опубликована: Ноя. 1, 2024

Sodium glucose cotransporter-2 inhibitors (SGLT2i), originally developed for type II diabetes mellitus, have recently been approved the treatment of heart failure in both diabetic and non-diabetic patients due to their significant cardiovascular benefits. Beyond established role management, current research is exploring potential applications SGLT2 field cardio-oncology. This interest driven by dual possible benefits: cardioprotection against adverse effects antitumor therapies inherent properties. Patients affected cancer often face challenge managing toxicity induced antineoplastic treatments. shown promise mitigating toxicities, thereby enhancing health these patients. Additionally, emerging evidence suggests that may possess direct effects, further contributing therapeutic oncology. review aims provide a comprehensive overview molecular mechanisms through which exert cardioprotective effects. Furthermore, we will examine body supporting use cardio-oncology setting.

Язык: Английский

Процитировано

0