Innovative Solid Lipid Nanoparticle-Enriched Hydrogels for Enhanced Topical Delivery of L-Glutathione: A Novel Approach to Anti-Ageing DOI Creative Commons
Mengyang Liu, Manisha Sharma, Guo‐Liang Lu

и другие.

Pharmaceutics, Год журнала: 2024, Номер 17(1), С. 4 - 4

Опубликована: Дек. 24, 2024

Background: Skin ageing, driven predominantly by oxidative stress from reactive oxygen species (ROS) induced environmental factors like ultraviolet A (UVA) radiation, accounts for approximately 80% of extrinsic skin damage. L-glutathione (GSH), a potent antioxidant, holds promise in combating UVA-induced stress. However, its instability and limited penetration through the stratum corneum hinder topical application. This study introduces novel solid lipid nanoparticle (SLN)-enriched hydrogel designed to enhance GSH stability, penetration, sustained release anti-ageing applications. Methods: GSH-loaded SLNs were prepared via double-emulsion technique optimized using factorial design. These incorporated into 1-3% (w/v) Carbopol hydrogels produce semi-solid formulation. The hydrogel's characteristics, including morphology, mechanical rheological properties, drug release, antioxidant activity, cytotoxicity, evaluated. Results: SEM FTIR confirmed uniform dispersion within hydrogel. formulation exhibited desirable gel strength (5.1 ± 0.5 g), spreadability (33.6 1.9 g·s), pseudoplasticity, elasticity. In vitro studies revealed biphasic profile, with over 72 h 70% cumulative release. significantly improved capacity, protecting human fibroblasts enhancing cell viability. Stability indicated that 4 °C was optimal storage three months. Notably, enhanced 3.7-fold. Conclusions: SLN-enriched effectively improves delivery efficacy, providing promising platform other bioactive compounds similar challenges.

Язык: Английский

Hair Longevity—Evidence for a Multifactorial Holistic Approach to Managing Hair Aging Changes DOI Open Access
Gillian E. Westgate,

Daniela Grohmann,

Manuel Sáez Moya

и другие.

Journal of Clinical Medicine, Год журнала: 2025, Номер 14(6), С. 1894 - 1894

Опубликована: Март 11, 2025

Loss of hair density—hair thinning and balding— is typically referred to as male female pattern alopecia. Causes include genetic predisposition links the impact dihydrotestosterone on follicle dermal papilla, which are characterized by an increase in number vellus follicles. Links chronological aging unclear. Proven treatments remain few still targeting tested those experiencing classical loss. The way changes with aging, especially women, can be considered having a much broader scope. Trends managing density, length, fiber quality now mostly cocktail approaches—whether topical, injected, or oral—recognizing that solutions more likely require multifactorial strategy. This review examines evidence for holistic approach addressing unwanted loss, includes nutrition, lifestyle, stress management, scalp care, well co-morbidities other health concerns. We discuss strengths limitations clinical study design investigate efficacy using approaches. propose this strategy will contribute emerging concept longevity follicle, scalp, targeted maintaining anagen most appropriate route achieving healthy aging. Finally, we problem facing patients consumers regarding quantity misinformation how it influences choosing from fast-growing market bypass pharmaceutical thinning.

Язык: Английский

Процитировано

0

Unveiling a novel in-vitro model of skin inflammaging DOI Creative Commons
Ying Xu, Yue Liu,

Jun‐Xiang Li

и другие.

Frontiers in Medicine, Год журнала: 2025, Номер 12

Опубликована: Март 28, 2025

Sensitive skin is characterized by a disrupted barrier, making it prone to reacting external stimuli, including UV exposure, air pollution, and cosmetic allergens. tends react with oxidative stress factors that could further lead inflammation subsequently result in inflammaging. However, there are almost no existing inflammaging models specifically for sensitive skin, highlighting the need develop method screening anti-inflammaging ingredients products. An vitro macrophage-fibroblast model was established evaluate effects of ingredients. The M1 phenotype aging-associated gene expression were assessed using qPCR validate model. RNA sequencing used elucidate mechanisms two validated A novel in-vitro developed applying supernatant macrophage culture medium induce cellular senescence fibroblast cells, facilitating In this model, supramolecular bakuchiol promote collagen COL1A1 COL3A3 production inhibit inflammatory enhancing transcription anti-inflammatory genes (PTX3, ADAM33, PDLIM1), while Terminalia chebula extract inhibits cell reducing MAP4K2 accumulation factor CCL3.

Язык: Английский

Процитировано

0

Promoting collagen synthesis: a viable strategy to combat skin ageing DOI Creative Commons
Shan Wang, Feifan Li,

Xi-long Feng

и другие.

Journal of Enzyme Inhibition and Medicinal Chemistry, Год журнала: 2025, Номер 40(1)

Опубликована: Апрель 11, 2025

Skin ageing is a complex physiological process primarily characterised by the deepening of wrinkles and sagging skin. Collagen essential for maintaining skin elasticity firmness. As ages, it experiences structural functional changes in collagen, including decrease collagen synthesis an increase hydrolysis. Thus, promoting represents practical strategy mitigating ageing. This review systematically described functions, classifications biosynthesis as well its role Additionally, major signalling pathways targets associated with were also discussed. More importantly, provided detailed summary natural products synthesis-promoting effects highlighted small molecule compounds potential anti-ageing activity, especially PPARδ agonists. The relevant content offers lead development anti-skin therapies.

Язык: Английский

Процитировано

0

Patients With Rosacea Exhibit Lower Minimal Erythema Doses to Both UVA and UVB DOI
Rong Wei, Xiaolin Wang,

Wen-Ting Lei

и другие.

Photodermatology Photoimmunology & Photomedicine, Год журнала: 2025, Номер 41(3)

Опубликована: Апрель 14, 2025

ABSTRACT Background Rosacea, a prevalent chronic inflammatory skin condition primarily affecting the central facial convexities, is categorized into four clinical subtypes: erythematotelangiectatic rosacea (ETR), papulopustular (PPR), phymatous (PhR), ocular (OR). While ultraviolet (UV) radiation recognized as risk factor for rosacea, differential sensitivity to UVA and/or UVB between healthy individuals and patients remains ambiguous. Methods This study comprised 70 diagnosed with 100 controls. The minimal erythema doses (MED‐UVA MED‐UVB) were ascertained using an SUV‐2000 solar UV simulator. A comparative analysis was conducted on MED‐UVA MED‐UVB results patient group control group, well among varying subtypes. Furthermore, correlation MED values in factors such age, type, antinuclear antibodies (ANA), Clinical Erythema Assessment (CEA) scale evaluated. Results In comparison demonstrated significantly lower ( p < 0.05) ≤ 0.001) values. However, no significant differences observed > subtypes of specifically ETR PPR. Conclusion Patients demonstrate decreased dose both UVB, suggesting heightened radiation. Consequently, it advisable minimize sun exposure order mitigate or prevent exacerbation condition.

Язык: Английский

Процитировано

0

Exploring the Evolution of Senotherapeutics Across Generations: A New Era in Human Dermal Fibroblast Senotherapy DOI Open Access

Samila Farokhimanesh

Journal of Skin and Stem Cell, Год журнала: 2025, Номер 12(1)

Опубликована: Март 28, 2025

Background: The skin, as the body’s largest organ, plays a crucial role in systemic physiological processes. Dysfunction often driven by cellular senescence, accelerates skin aging and contributes to aging. accumulation of senescent cells secretion senescence-associated secretory phenotype (SASP) factors are central mechanisms underlying aging, particularly affecting dermal fibroblasts, which key producers collagen elastin. Given these challenges, senotherapy has emerged promising strategy mitigate specifically targeting cells. Objectives: present study evaluates therapeutic potential advanced senotherapeutics critical for maintaining structure function. It highlights integration cutting-edge technologies, including targeted nanoparticles, chimeric antigen receptor T (CAR-T) cells, artificial intelligence, gene editing, address cell heterogeneity improve outcomes. Methods: Various senotherapeutics, senolytic agents eliminating senomorphic modulating SASP, were assessed. Advanced technologies such CAR-T editing evaluated their ability enhance specificity reduce off-target effects. focused on efficacy fibroblasts inflammatory markers associated with SASP. Preclinical vitro models used test approaches. Results: demonstrated significant improvements selectively while minimizing These therapies effectively modulated leading reduced an enhanced environment health. By addressing challenges heterogeneity, approaches showcased superior precision compared earlier generations, emphasizing mitigating both Conclusions: findings highlight its implications. Through precise effective modulation offer transformative improving health combating broader age-related challenges. incorporation marks advancement pursuit innovative anti-aging solutions.

Язык: Английский

Процитировано

0

Innovative Solid Lipid Nanoparticle-Enriched Hydrogels for Enhanced Topical Delivery of L-Glutathione: A Novel Approach to Anti-Ageing DOI Creative Commons
Mengyang Liu, Manisha Sharma, Guo‐Liang Lu

и другие.

Pharmaceutics, Год журнала: 2024, Номер 17(1), С. 4 - 4

Опубликована: Дек. 24, 2024

Background: Skin ageing, driven predominantly by oxidative stress from reactive oxygen species (ROS) induced environmental factors like ultraviolet A (UVA) radiation, accounts for approximately 80% of extrinsic skin damage. L-glutathione (GSH), a potent antioxidant, holds promise in combating UVA-induced stress. However, its instability and limited penetration through the stratum corneum hinder topical application. This study introduces novel solid lipid nanoparticle (SLN)-enriched hydrogel designed to enhance GSH stability, penetration, sustained release anti-ageing applications. Methods: GSH-loaded SLNs were prepared via double-emulsion technique optimized using factorial design. These incorporated into 1-3% (w/v) Carbopol hydrogels produce semi-solid formulation. The hydrogel's characteristics, including morphology, mechanical rheological properties, drug release, antioxidant activity, cytotoxicity, evaluated. Results: SEM FTIR confirmed uniform dispersion within hydrogel. formulation exhibited desirable gel strength (5.1 ± 0.5 g), spreadability (33.6 1.9 g·s), pseudoplasticity, elasticity. In vitro studies revealed biphasic profile, with over 72 h 70% cumulative release. significantly improved capacity, protecting human fibroblasts enhancing cell viability. Stability indicated that 4 °C was optimal storage three months. Notably, enhanced 3.7-fold. Conclusions: SLN-enriched effectively improves delivery efficacy, providing promising platform other bioactive compounds similar challenges.

Язык: Английский

Процитировано

1