G Protein-coupled Estrogen Receptor 1 (GPER1) Regulates Expression ofSERPINE1/PAI-1 and Inhibits Tumorigenic Potential of Cervical Squamous Cell Carcinoma CellsIn Vitro DOI Open Access

LINEA RÖRIG,

SOPHIA RUCKRIEGL,

Julia Gallwas

и другие.

Cancer Genomics & Proteomics, Год журнала: 2024, Номер 22(1), С. 13 - 23

Опубликована: Дек. 27, 2024

Background/Aim: G protein-coupled estrogen receptor 1 (GPER1) appears to play a tumor-suppressive role in cervical squamous cell carcinoma (CSCC)GPER1 suppression leads significantly increased expression of serpin family E member (SERPINE1)/protein plasminogen activator inhibitor type (PAI-1). The question arises, what does SERPINE1/PAI-1 GPER1-dependent tumorigenic potential CSCC. Materials and Methods: SiHa C33A CSCC cells were treated with GPER1 agonist G1 or antagonist G36. was suppressed by RNAi success confirmed RT-qPCR. Protein PAI-1 quantified Western blot. Viability analyzed using resazurin assay, while migration investigated gap closure. Colony tumor sphere formation used test clonogenicity. Results: After treatment, viability remained unchanged. Cell dose-dependently reduced. formed fewer smaller colonies as well spheroids. Furthermore, treatment led decreased SERPINE1/PAI-1, blockade G36 resulted expression. RNAi, unaffected; however, formed, spheroids developed. unaffected. Conclusion: Activation reduces clonogenicity suppresses SERPINE1/PAI-1. Suppression potential. may be suitable target for However, not appear the decisive factor GPER1-regulated migration.

Язык: Английский

Unveiling the role of ASPP1 in cancer progression: pan-cancer bioinformatics and experimental validation in colorectal cancer DOI Creative Commons
Keyuan Xiao, Xiang Li, Ihsan Ullah

и другие.

Frontiers in Oncology, Год журнала: 2025, Номер 14

Опубликована: Янв. 2, 2025

The Apoptosis-Stimulating Protein of P53 (ASPP) family contributes to apoptosis regulation and tumor suppression, with ASPP1 influencing processes like cancer cell proliferation, invasion, migration. Its expression varies across types, suggesting a potential role in oncogenesis. This study investigates ASPP1's various cancers using comprehensive bioinformatics approach. Data were extracted from public resources, including Cancer Genome Atlas (TCGA), GTEx, the Human Atlas, analyzed via tools such as cBioPortal, GEPIA, TIMER2. Statistical network analyses performed R, Cytoscape, Hiplot. function colorectal was further explored through vitro assays, qRT-PCR, Western blotting, colony formation, Transwell, wound healing. exhibited significant variability different marked associations patient outcomes, particularly overall survival (OS) disease-specific (DSS) several types. In-depth protein-protein interaction (PPI) analysis revealed involvement progression networks. Functional enrichment linked key apoptotic signaling pathways transcriptional regulatory processes, underscoring its impact on biology. Additionally, correlates immune infiltration patterns, cancer-associated fibroblasts markers, roles response modulation. In assays lines significantly lower levels compared normal colon cells (HCM460), overexpression experiments showed reduction migration abilities. These cellular findings align predictions, highlighting suppressor metastatic traits cancer. highlights forecasting biomarker potentially other cancers. support biology, regarding proliferation potential, establishing foundation for investigation into therapeutic relevance.

Язык: Английский

Процитировано

0

Impact of the Immune Landscape in Follicular Lymphoma: Insights into Histological Transformation in the Rituximab Era DOI Open Access
Marie Beck Enemark,

Maria Fuglsang Jensen,

Maja Dam Andersen

и другие.

Cancers, Год журнала: 2024, Номер 16(20), С. 3553 - 3553

Опубликована: Окт. 21, 2024

Follicular lymphoma (FL) presents significant clinical heterogeneity, with some patients experiencing transformation into an aggressive disease, a key contributor to FL-related mortality. Based on gene expression profiles, this study aimed provide insights immunological differences associated transformation.

Язык: Английский

Процитировано

0

G Protein-coupled Estrogen Receptor 1 (GPER1) Regulates Expression ofSERPINE1/PAI-1 and Inhibits Tumorigenic Potential of Cervical Squamous Cell Carcinoma CellsIn Vitro DOI Open Access

LINEA RÖRIG,

SOPHIA RUCKRIEGL,

Julia Gallwas

и другие.

Cancer Genomics & Proteomics, Год журнала: 2024, Номер 22(1), С. 13 - 23

Опубликована: Дек. 27, 2024

Background/Aim: G protein-coupled estrogen receptor 1 (GPER1) appears to play a tumor-suppressive role in cervical squamous cell carcinoma (CSCC)GPER1 suppression leads significantly increased expression of serpin family E member (SERPINE1)/protein plasminogen activator inhibitor type (PAI-1). The question arises, what does SERPINE1/PAI-1 GPER1-dependent tumorigenic potential CSCC. Materials and Methods: SiHa C33A CSCC cells were treated with GPER1 agonist G1 or antagonist G36. was suppressed by RNAi success confirmed RT-qPCR. Protein PAI-1 quantified Western blot. Viability analyzed using resazurin assay, while migration investigated gap closure. Colony tumor sphere formation used test clonogenicity. Results: After treatment, viability remained unchanged. Cell dose-dependently reduced. formed fewer smaller colonies as well spheroids. Furthermore, treatment led decreased SERPINE1/PAI-1, blockade G36 resulted expression. RNAi, unaffected; however, formed, spheroids developed. unaffected. Conclusion: Activation reduces clonogenicity suppresses SERPINE1/PAI-1. Suppression potential. may be suitable target for However, not appear the decisive factor GPER1-regulated migration.

Язык: Английский

Процитировано

0