Advances in Psychedelic Therapeutics: Novel Prodrugs and Derivatives for Enhanced Mental Health Treatment DOI Creative Commons
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Год журнала: 2024, Номер 15(12), С. 2071 - 2073

Опубликована: Ноя. 11, 2024

Recent innovations in psychedelic research have led to the development of novel compounds designed enhance therapeutic potential psilocin and related tryptamines. This Patent Highlight reviews three essential patents that focus on improving stability, bioavailability, efficacy these for treating mental health disorders such as depression, anxiety, substance use disorders. The compounds─4-pivaloyloxy-N-methyltryptammonium chloride, alkyl quaternary ammonium tryptamines, 4-pivaloyloxy-N-methyltryptammonium derivatives─represent significant advancements field psychedelic-assisted therapy. These offer new hope more reliable effective treatments, particularly addressing limitations associated with traditional psychedelics. findings from preclinical studies support play a vital role treatment neurological

Язык: Английский

Psilocybin-assisted psychotherapy for Parkinson's disease without depression: A case-report DOI Creative Commons
Vanessa Fleury,

Emilie Tomkova,

Sabina Catalano Chiuvé

и другие.

Journal of Parkinson s Disease, Год журнала: 2025, Номер unknown

Опубликована: Фев. 2, 2025

Background Psychedelic assisted psychotherapy (PAP) can improve treatment-resistant depression. Its usefulness in Parkinson's disease (PD) is unknown. PD patients may have problems adjusting to their chronic progressive neurological disease. A change from emotional avoidance acceptance has been reported following psilocybin administration with Objective To report for the first time effect of a patient. Methods non-depressed 43-year-old female 2-year history presented difficulty PD, anxious ruminations and pessimism. The patient declined an increase dopaminergic medication or introduction anxiolytic. Therapeutic education was not beneficial. received four sessions high-dose PAP within one year. Neurological psychiatric assessments were performed before at year follow-up using qualitative interviews quantitative assessment motor status, dispositional optimism, depression, anxiety, apathy, well-being. Results well tolerated. It significantly improved patient's overall pessimistic outlook on her future decreased worries about potential handicap due PD. Her general well-being improved, as all psychometric scores except apathy scale. Motor status remained unchanged. Better allowed accept pharmacological treatment adjustment. Conclusions could be safe useful pessimism difficulties accepting by promoting profound decentration habitual thoughts emotions, improving mood acceptance. Randomized, controlled studies are needed confirm this result.

Язык: Английский

Процитировано

0

Exploring novel therapeutic strategies: Could psychedelic perspectives offer promising solutions for Alzheimer’s disease comorbidities? DOI Creative Commons

Michael Davidson,

Gabriela Dumitrița Stanciu, Jonathan Rabinowitz

и другие.

Dialogues in Clinical Neuroscience, Год журнала: 2025, Номер 27(1), С. 1 - 12

Опубликована: Март 19, 2025

The increasing prevalence of dementia within an ageing global population, combined with prolonged life expectancy, accentuates Alzheimer's disease (AD) as a multifaceted healthcare challenge. This challenge is further compounded by the limited therapeutic options currently available. Addressing intricacies AD management, mitigation comorbidities has emerged pivotal facet treatment. Comorbid conditions, such neurobehavioral symptoms, play role in shaping clinical course, and outcomes this pathology; highlighting importance comprehensive care approaches for affected individuals. Exploration psychedelic compounds psychiatric palliative settings recently uncovered promising potential, enhancing neuroplasticity, emotional processing connection. These effects are particularly relevant context AD, where therapy offers hope not only mitigating core symptoms but also addressing array associated condition. integration method chance to significantly enhance provided those navigating intricate landscape AD. Therefore, current paper reviews link between more frequent additional health conditions that may coexist dementia, explores potential these concurrent conditions.

Язык: Английский

Процитировано

0

Mushrooms, Microdosing, and Mental Illness: The Effect of Psilocybin on Neurotransmitters, Neuroinflammation, and Neuroplasticity DOI Creative Commons
Daniel A Kinderlehrer

Neuropsychiatric Disease and Treatment, Год журнала: 2025, Номер Volume 21, С. 141 - 155

Опубликована: Янв. 1, 2025

The incidence of mental health disorders is increasing worldwide. While there are multiple factors contributing to this problem, neuroinflammation underlies a significant subset psychiatric conditions, particularly major depressive and anxiety disorders. Anti-inflammatory interventions have demonstrated benefit in these conditions. Psilocin, the active ingredient mushrooms Psilocybe genus, both potent serotonin agonist anti-inflammatory agent, increases neuroplasticity, decreases overactivity default mode network. Studies using hallucinogenic doses psilocin under supervision therapist/guide consistently benefits individuals with depression end-of-life anxiety. Microdosing psilocybin sub-hallucinogenic has also mood disorders, may offer safe, less expensive, more available alternative full for as well other medical conditions which inflammation principal pathophysiology.

Язык: Английский

Процитировано

0

Exploring psilocybin’s role in mental health and palliative medicine: a path to improved well-being DOI

Maria-Alejandra Umbacia,

Marta León, Jose-Manuel Quintero

и другие.

Expert Opinion on Emerging Drugs, Год журнала: 2025, Номер unknown

Опубликована: Апрель 3, 2025

Although long known for their psychoactive effects, psychedelic drugs have only recently been investigated medicinal use. Psilocybin has attracted the greatest interest with studies suggesting that it may be a useful agent in psychiatry and palliative care. Clinical trials included psilocybin were searched PubMed, Embase, ClinicalTrials.gov, demonstrating adult care are medical fields show treatment. is powerful drug needs to used caution but benefit some patients, including when other options failed. It best evidenced treatment resistant depression care, where patients usually treated specialist centers. novel mechanism of action, targeting 5HT2A receptor, can rapid onset action. There many questions regarding its use remain clarified, efficacy indications role as adjunctive psychotherapy. The psychoactive, or effects well documented, clinical importance disputed.

Язык: Английский

Процитировано

0

Advancements in Neurotechnology: Pioneering Brain Monitoring and Stimulation for Enhanced Treatment and Understanding DOI Creative Commons
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Год журнала: 2024, Номер 16(1), С. 20 - 22

Опубликована: Дек. 18, 2024

This Patent Highlight explores recent innovations in neuroscience and neurotechnology, particularly brain monitoring stimulation. It examines four essential patents: novel psychoplastogens for neuronal growth, techniques transferring emotional states, advanced systems self-guided neural diagnostics treatment. The discussion extends to deep stimulation (DBS) motor memory disorders, enhanced function through electroencephalography (EEG), the role of artificial intelligence personalizing treatment strategies. These advancements represent a pivotal development introducing innovative methodologies elucidating neurological mechanisms, addressing psychiatric augmenting cognitive function.

Язык: Английский

Процитировано

0

Advances in Psychoactive Alkaloid Delivery, Ergoline Analogues, and Serotonin Receptor Modulation for Enhanced Therapeutic Outcomes DOI Creative Commons
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Год журнала: 2024, Номер 16(1), С. 26 - 28

Опубликована: Дек. 18, 2024

Recent advancements in pharmaceutical research have focused on developing novel psychoactive compounds and receptor modulators that enhance therapeutic outcomes while minimizing adverse effects. This Patent Highlight examines three innovative approaches: (1) transmucosal delivery of dephosphorylated alkaloids, (2) nonhallucinogenic serotonin modulators, (3) ergoline analogues designed for treating neurological disorders. These innovations offer breakthroughs drug delivery, targeting, structural modifications, aiming to address challenges the treatment mood disorders, diseases, chronic pain improving bioavailability reducing side effects hallucinogenic properties.

Язык: Английский

Процитировано

0

Advances in Psychedelic Therapeutics: Novel Prodrugs and Derivatives for Enhanced Mental Health Treatment DOI Creative Commons
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Год журнала: 2024, Номер 15(12), С. 2071 - 2073

Опубликована: Ноя. 11, 2024

Recent innovations in psychedelic research have led to the development of novel compounds designed enhance therapeutic potential psilocin and related tryptamines. This Patent Highlight reviews three essential patents that focus on improving stability, bioavailability, efficacy these for treating mental health disorders such as depression, anxiety, substance use disorders. The compounds─4-pivaloyloxy-N-methyltryptammonium chloride, alkyl quaternary ammonium tryptamines, 4-pivaloyloxy-N-methyltryptammonium derivatives─represent significant advancements field psychedelic-assisted therapy. These offer new hope more reliable effective treatments, particularly addressing limitations associated with traditional psychedelics. findings from preclinical studies support play a vital role treatment neurological

Язык: Английский

Процитировано

0