Improving the Anti-Tumor Effect of Indoleamine 2,3-Dioxygenase Inhibitor CY1-4 by CY1-4 Nano-Skeleton Drug Delivery System DOI Creative Commons
Hui Li,

Jun-Wei Liu,

Jingru Wang

и другие.

Journal of Functional Biomaterials, Год журнала: 2024, Номер 15(12), С. 372 - 372

Опубликована: Дек. 9, 2024

CY1-4, 9-nitropyridine [2',3':4,5] pyrimido [1,2-α] indole -5,11- dione, is an indoleamine 2,3-dioxygenase (IDO) inhibitor and a poorly water-soluble substance. It very important to increase the solubility of CY1-4 improve its bioavailability therapeutic effect. In this study, mesoporous silica nano-skeleton carrier material Sylysia was selected as load then drug delivery system (MSNM@CY1-4) prepared by coating hydrophilic polymer Hydroxypropyl methylcellulose (HPMC) lipid Distearoylphosphatidyl-ethanolamine-poly(ethylene glycol)

Язык: Английский

Exercise-induced adaptations in the kynurenine pathway: implications for health and disease management DOI Creative Commons
Marcus Vinícius dos Santos Rangel, Karynne Grutter Lopes, Xuebin Qin

и другие.

Frontiers in Sports and Active Living, Год журнала: 2025, Номер 7

Опубликована: Март 6, 2025

Background Tryptophan (TRP) metabolism through the kynurenine (KYN) pathway is influenced by inflammatory mediators, generating metabolites that regulate immune and responses. Exercise has been proposed as a modulator of this pathway, but its role in health benefits chronic disease management remains unclear. Objective This systematic review examines exercise-induced adaptations KYN their potential implications for management. Additionally, we identify key methodological considerations future research. Methods A structured search PubMed/Medline, Web Science, Scopus was conducted up to October 2024 clinical trials investigating effects exercise training on pathway. Results Of 2,795 articles initially found, 13 involving 592 participants met inclusion criteria. Most studies reported particularly cancer survivors. These appeared be intensity duration. However, several limitations were noted, no included patients with metabolic or cardiovascular diseases. Conclusions Here, show modulates both healthy diseased populations, highlighting prevention further randomized-controlled are needed clarify mechanisms applications, Systematic Review Registration https://www.crd.york.ac.uk/PROSPERO/view/CRD42022351481 , PROSPERO (CRD42022351481).

Язык: Английский

Процитировано

0

Exploring the Mechanism of Action of Honeybran‐Fried Cimicifuga Rhizoma in the Treatment of IBS‐D Based on Metabolomics and Network Pharmacology DOI Open Access
Jingchuan Zhu,

Yuxuan Zou,

Yao Wu

и другие.

Biomedical Chromatography, Год журнала: 2025, Номер 39(5)

Опубликована: Март 24, 2025

ABSTRACT Honeybran‐fried Cimicifuga Rhizoma (HBCR) is often used to treat prolonged diarrhea and prolapse of the anus, uterine prolapse, gastric ptosis caused by spleen qi deficiency inability elevate qi, thus lowering middle qi. Rats were divided randomly into four groups. Fecal samples rats in each group subjected metabolomics analysis. We identified chemical components HBCR using liquid chromatography–tandem mass spectrometry. predicted potential active key targets network pharmacology construct a “drug–potential ingredient–target–disease” network. The screened differential metabolites analysis combined pathway Pharmacodynamic indices showed that had good therapeutic effect upon IBS‐D. Metabolomics revealed 26 treatment IBS‐D HBCR. A total 69 identified, 32 296 screened. Combination for joint may be affected metabolism linoleic acid, retinol, arachidonic tryptophan. significant effects with

Язык: Английский

Процитировано

0

Peripheral Kynurenine Pathway Metabolites in Patients with Psoriasis DOI Open Access
Anna Stepaniuk, Anna Baran, Justyna Magdalena Hermanowicz

и другие.

International Journal of Molecular Sciences, Год журнала: 2025, Номер 26(7), С. 3139 - 3139

Опубликована: Март 28, 2025

Psoriasis is a systemic disease affecting 2-3% of the general population. Tryptophan (TRP) an amino acid metabolized in kynurenine pathway (KP). The aim this study was to assess pathway's metabolites serum and urine psoriatic patients explore possible interplay with disease's pathogenesis its comorbidities. involved 60 plaque psoriasis 30 healthy volunteers matched for gender, age, BMI. Serum samples were taken from participants tested TRP, indoleamine 2,3-dioxygenase (IDO), 2,3-tryptophan dioxygenase (TDO), (KYN), kynurenic (KYNA), quinolinic (QUIN), numerous laboratory parameters. Correlations between metabolites' levels clinical, parameters depression occurrence statistically evaluated. Concentrations tryptophan, acid, significantly higher among (p < 0.05 p 0.001, 0.001 respectively). A significant stimulation suggests role chronic inflammation or Further research needed discover whether increase KP indicator compensatory mechanism psoriasis.

Язык: Английский

Процитировано

0

Kynurenine Pathway in Epilepsy: Unraveling Its Role in Glutamate Excitotoxicity, GABAergic Dysregulation, Neuroinflammation, and Mitochondrial Dysfunction DOI
Manpreet Kaur,

Pratyush Porel,

Ronak Y. Patel

и другие.

Neurotoxicity Research, Год журнала: 2025, Номер 43(2)

Опубликована: Март 28, 2025

Язык: Английский

Процитировано

0

Improving the Anti-Tumor Effect of Indoleamine 2,3-Dioxygenase Inhibitor CY1-4 by CY1-4 Nano-Skeleton Drug Delivery System DOI Creative Commons
Hui Li,

Jun-Wei Liu,

Jingru Wang

и другие.

Journal of Functional Biomaterials, Год журнала: 2024, Номер 15(12), С. 372 - 372

Опубликована: Дек. 9, 2024

CY1-4, 9-nitropyridine [2',3':4,5] pyrimido [1,2-α] indole -5,11- dione, is an indoleamine 2,3-dioxygenase (IDO) inhibitor and a poorly water-soluble substance. It very important to increase the solubility of CY1-4 improve its bioavailability therapeutic effect. In this study, mesoporous silica nano-skeleton carrier material Sylysia was selected as load then drug delivery system (MSNM@CY1-4) prepared by coating hydrophilic polymer Hydroxypropyl methylcellulose (HPMC) lipid Distearoylphosphatidyl-ethanolamine-poly(ethylene glycol)

Язык: Английский

Процитировано

0