A Focused Review on Oxidation of Hydrazones Using Hypervalent Iodine Reagents DOI Open Access
Monika Sihag, Mayank Kinger, Deepak Kumar Aneja

и другие.

ChemistrySelect, Год журнала: 2024, Номер 10(1)

Опубликована: Дек. 31, 2024

Abstract Hydrazones are described as synthetic equivalents to the carbonyl group and possess high synthon value. Herein, we compile oxidative transformation of hydrazones using ecologically economically benign hypervalent iodine reagents last decade. In this field, development C─H functionalization reactions leading formation heterocycles or functionalized is a major advancement in recent years. The properties exploited form many bioactive (pyrazole, pyrazoline, pyridazine, 1,2,4‐triazole, 1,2,3‐tiazole, 1,3,4‐oxadiazole, tetrazine, tetrazole, pyrrole) through intramolecular intermolecular C─N, C─O, N─N coupling. Functionalized also afforded via tandem cascade transfer/cyclization reactions. transfer perfluoroalkyl, sulfoximidoyl, aryl, halogen groups achieved donors oxidants combination with other group‐donating agents. Togni reagent preferred choice for trifluoromethyl donation, without metal catalyst. Moreover, rearrangement such acyl migration diazotization achieved.

Язык: Английский

Crystal Structure, Hirshfeld Surface Analysis, and Computational Insights into Phenoxyacetohydrazones: Hydrogen-Bonded Dimers and p-Stacking Interactions. DOI

Camila Capelini,

Samir A. Carvalho, Camilo Henrique da Silva Lima

и другие.

Journal of Molecular Structure, Год журнала: 2025, Номер 1333, С. 141752 - 141752

Опубликована: Фев. 16, 2025

Язык: Английский

Процитировано

0

Photo- and Electro-chemical Strategies for Indazole Synthesis DOI Creative Commons
Binbin Huang

Tetrahedron Chem, Год журнала: 2024, Номер unknown, С. 100116 - 100116

Опубликована: Дек. 1, 2024

The indazole core is prevalently found in the structures of bioactive molecules, demonstrating promising potential medicinal chemistry and drug discovery, which therefore has attracted sustained attention from synthetic community. Over recent decades, significant progress been achieved both organic photocatalysis electrosynthesis, offering novel approaches for efficient sustainable synthesis various functionalized indazoles. This mini-review highlights emerging methodological advancements photo-/electro-chemical two common forms indazole, namely 1H- 2H-indazoles, are classified by specific intramolecular bond formation patterns: (1) C-C formation, (2) C-N (3) N-N formation. reaction conditions, representative scopes, mechanistic understandings these protocols emphasized, to elucidate advantages limitations current strategies, with an aim inspire future innovations that may address challenges modern synthesis.Graphical abstractTo create your abstract, type over instructions template box below. Fonts or abstract dimensions should not be changed altered.

Язык: Английский

Процитировано

1

A Focused Review on Oxidation of Hydrazones Using Hypervalent Iodine Reagents DOI Open Access
Monika Sihag, Mayank Kinger, Deepak Kumar Aneja

и другие.

ChemistrySelect, Год журнала: 2024, Номер 10(1)

Опубликована: Дек. 31, 2024

Abstract Hydrazones are described as synthetic equivalents to the carbonyl group and possess high synthon value. Herein, we compile oxidative transformation of hydrazones using ecologically economically benign hypervalent iodine reagents last decade. In this field, development C─H functionalization reactions leading formation heterocycles or functionalized is a major advancement in recent years. The properties exploited form many bioactive (pyrazole, pyrazoline, pyridazine, 1,2,4‐triazole, 1,2,3‐tiazole, 1,3,4‐oxadiazole, tetrazine, tetrazole, pyrrole) through intramolecular intermolecular C─N, C─O, N─N coupling. Functionalized also afforded via tandem cascade transfer/cyclization reactions. transfer perfluoroalkyl, sulfoximidoyl, aryl, halogen groups achieved donors oxidants combination with other group‐donating agents. Togni reagent preferred choice for trifluoromethyl donation, without metal catalyst. Moreover, rearrangement such acyl migration diazotization achieved.

Язык: Английский

Процитировано

1