The Design and Optimization of Fast-dissolving Oral Drug Delivery System (ODDS) of Valproic Acid (VLA) an Anti-epileptic Category Drug DOI Open Access

Devanand Jha,

Gagan Kumar Utwaliya,

K. Bhavya Sindhu

и другие.

Advances in Research, Год журнала: 2024, Номер 25(2), С. 152 - 166

Опубликована: Фев. 28, 2024

Objective: Develop and optimize a fast-dissolving oral drug delivery system (ODDS) for Valproic acid (VLA), an anti-epileptic drug, using Design of Experiments (DoE). Methodology: DoE, powerful tool optimizing formulations, was employed to investigate the impact various factors on dissolution rate VLA ODDS. Key studied included superdisintegrants (sodium starch glycolate, crospovidone), diluents (lactose, microcrystalline cellulose), lubricants (magnesium stearate). A Box-Behnken design used create experimental runs, at 30 minutes chosen as response variable. Results: The DoE analysis revealed significant interactions between affecting rate. formulation containing sodium lactose, low magnesium stearate concentration exhibited fastest (Q30 > 85% in 10 minutes). Conclusion: This study successfully designed optimized ODDS DoE. offered rapid release, potentially improving patient compliance therapeutic efficacy. approach demonstrates effectiveness pharmaceutical formulations enhanced performance. findings indicated that RSM effectively utilized developing valproic fast dispersible tablets, thus representing progress treatment epileptic seizures.

Язык: Английский

An Updated Comprehensive Review on Novel Drug Delivery Systems (NDDS) In the Pharmaceuticals DOI Open Access

Vinay Kumar Rao Khadam,

Ravindra Pal Singh, Deepak Prajapati

и другие.

Asian Journal of Pharmaceutical Research and Development, Год журнала: 2024, Номер 12(1), С. 55 - 64

Опубликована: Фев. 15, 2024

The field of pharmaceutical sciences has witnessed a paradigm shift with the advent Novel Drug Delivery Systems (NDDS), which aim to enhance therapeutic efficacy, reduce side effects, and improve patient compliance. This comprehensive review explores latest advancements innovations in NDDS, encompassing diverse range delivery platforms strategies.(NDDs are transforming landscape treatment, offering unparalleled potential for enhanced improved bioavailability, controlled release, targeted delivery, stability. highlighting recent addressing key challenges. Prominent NDDS include liposomes, nanoparticles, micelles, polymeric drug conjugates, monoclonal antibodies, implants, patches. Each system possesses unique properties applications, tailored specific drugs needs. Recent breakthroughs nanocarriers, gene therapy vectors, 3D-printed personalized dosage forms pushing boundaries innovation. main highlights present firstly basics on NDDs, several approaches nano carriers their preparation methods example. middle version discuss techniques NDDs lastly marketed formulation particular carrier.

Язык: Английский

Процитировано

4

The Design and Optimization of Fast-dissolving Oral Drug Delivery System (ODDS) of Valproic Acid (VLA) an Anti-epileptic Category Drug DOI Open Access

Devanand Jha,

Gagan Kumar Utwaliya,

K. Bhavya Sindhu

и другие.

Advances in Research, Год журнала: 2024, Номер 25(2), С. 152 - 166

Опубликована: Фев. 28, 2024

Objective: Develop and optimize a fast-dissolving oral drug delivery system (ODDS) for Valproic acid (VLA), an anti-epileptic drug, using Design of Experiments (DoE). Methodology: DoE, powerful tool optimizing formulations, was employed to investigate the impact various factors on dissolution rate VLA ODDS. Key studied included superdisintegrants (sodium starch glycolate, crospovidone), diluents (lactose, microcrystalline cellulose), lubricants (magnesium stearate). A Box-Behnken design used create experimental runs, at 30 minutes chosen as response variable. Results: The DoE analysis revealed significant interactions between affecting rate. formulation containing sodium lactose, low magnesium stearate concentration exhibited fastest (Q30 > 85% in 10 minutes). Conclusion: This study successfully designed optimized ODDS DoE. offered rapid release, potentially improving patient compliance therapeutic efficacy. approach demonstrates effectiveness pharmaceutical formulations enhanced performance. findings indicated that RSM effectively utilized developing valproic fast dispersible tablets, thus representing progress treatment epileptic seizures.

Язык: Английский

Процитировано

1