The need for inhaled phosphodiesterase inhibitors in chronic obstructive pulmonary disease DOI
Mario Cazzola, Luigino Calzetta, Paola Rogliani

и другие.

Expert Review of Clinical Pharmacology, Год журнала: 2024, Номер unknown

Опубликована: Дек. 3, 2024

Introduction The therapeutic implications of phosphodiesterase (PDE) inhibitors have attracted interest because PDEs are regarded as an intracellular target to be exploited for advancements in the treatment COPD. At present, only approved approach COPD with PDE is use oral PDE4 inhibitor. However, this not widely employed, primarily due narrow index associated inhibitors, which considerably restricts permissible dosage. inhalation route represents a viable alternative improving inhibitors.

Язык: Английский

Ensifentrine for COPD DOI
Rajat Suri, Sanjay Ramakrishnan

CHEST Journal, Год журнала: 2025, Номер 167(2), С. 305 - 306

Опубликована: Фев. 1, 2025

Язык: Английский

Процитировано

0

Ensifentrine vs placebo for chronic obstructive pulmonary disease: a systematic review and meta-analysis of randomized clinical trials DOI
Giulia Carvalhal,

Gonzalo Alberto Peralta-Jiménez,

M. Mora

и другие.

Expert Review of Respiratory Medicine, Год журнала: 2025, Номер unknown

Опубликована: Апрель 19, 2025

To evaluate the efficacy and safety of ensifentrine in chronic obstructive pulmonary disease (COPD). We searched electronic databases registries until 25 January 2025, for randomized clinical trials (RCTs) comparing vs placebo patients with COPD. Primary outcomes include forced expiratory volume one second (FEV₁) area under curve (AUC), peak FEV₁, morning trough FEV₁. Ten RCTs involving 2,589 were included. Compared placebo, improved FEV₁ AUC by 104.24 ml (95% CI, 74.03 to 133.44; moderate certainty) on day 1 90.37 54.94 125.81; at study end. Ensifentrine increased 140.99 107.48 174.5; 118.98 final assessment 86.49 151.47; certainty). 42.15 19.87 64.43; high Dose-response analysis showed a bell-shaped all outcomes. did not significantly differ from adverse events or improvements COPD symptoms quality life. lung function Larger are needed integrate this bronchodilator benefit patient-centered CRD42024571928.

Язык: Английский

Процитировано

0

The need for inhaled phosphodiesterase inhibitors in chronic obstructive pulmonary disease DOI
Mario Cazzola, Luigino Calzetta, Paola Rogliani

и другие.

Expert Review of Clinical Pharmacology, Год журнала: 2024, Номер unknown

Опубликована: Дек. 3, 2024

Introduction The therapeutic implications of phosphodiesterase (PDE) inhibitors have attracted interest because PDEs are regarded as an intracellular target to be exploited for advancements in the treatment COPD. At present, only approved approach COPD with PDE is use oral PDE4 inhibitor. However, this not widely employed, primarily due narrow index associated inhibitors, which considerably restricts permissible dosage. inhalation route represents a viable alternative improving inhibitors.

Язык: Английский

Процитировано

2