Layer-by-Layer Biopolymer-Coated Deformable Liposomes–In Situ Gel: A Hybrid Strategy for Enhanced Ocular Delivery of Itraconazole: In Vitro and In Vivo Appraisal DOI Creative Commons

Mohamed M. Badran,

Areej Alsubaie,

Mounir M. Salem‐Bekhit

и другие.

Gels, Год журнала: 2024, Номер 11(1), С. 19 - 19

Опубликована: Дек. 31, 2024

Itraconazole (ITZ) is a potent antifungal agent. Its oral administration associated with systemic toxicity, and its efficacy in ocular formulations limited. This study aims to enhance ITZ’s permeation by loading it into deformable liposomes (DLs) based on Tween 80 (T) or Poloxamer 188 (P). Moreover, ITZ was loaded biopolymer-coated DLs augment availability. ITZ-loaded were coated hyaluronic acid (HA-DLs), chitosan (CS-DLs), layer-by-layer coating (CS/HA-DLs). These further laden pH-sensitive situ gels provide hybrid system intensify their adhesion properties. The prepared successfully vesicle sizes nonorange (<200 nm). zeta potential values of DLS negative before shifted high negativity HA positivity CS CS/HA bilayer coating. variations indicate successful coatings. optimized A EE% achieved DLs-T: 89% (CS/HA-DLs-T), 86% (CS-DLs-T), 85% (HA-DLs-T), 79% (HA-DLs-T). Therefore, DLs-T incorporated gels, displaying optimal gelling capacity viscosity. release rate from the DLs-laden slower than that observed uncoated DLs-gel. CS/HA-DLs-T laden-in showed highest ex vivo transcorneal permeability efficacy. data suggest layer-by-layer-CS/HA-DLs-T presents hopeful strategy for delivery ITZ, offering promising approach managing fungal infections.

Язык: Английский

Novel Strategies for Preventing Fungal Infections—Outline DOI Creative Commons

Damilola Janet Agbadamashi,

Claire Price

Pathogens, Год журнала: 2025, Номер 14(2), С. 126 - 126

Опубликована: Фев. 1, 2025

Fungal infections are a significant global health challenge, causing approximately 3.8 million deaths annually, with immunocompromised populations particularly at risk. Traditional antifungal therapies, including azoles, echinocandins, and polyenes, face limitations due to rising resistance, toxicity, inadequate treatment options. This review explores innovative strategies for preventing managing fungal infections, such as vaccines, peptides, nanotechnology, probiotics, immunotherapy. Vaccines offer promising avenues long-term protection, despite difficulties in their development complexity immune evasion mechanisms. Antifungal peptides provide novel class of agents broad-spectrum activity reduced resistance risk, whilst nanotechnology enables targeted, effective drug delivery systems. Probiotics show potential vulvovaginal candidiasis, by maintaining microbial balance. Immunotherapy leverages system modulation enhance defenses, omics technologies deliver comprehensive insights into biology, paving the way therapeutic vaccine targets. While these approaches hold immense promise, challenges cost, accessibility, translational barriers remain. A coordinated effort among researchers, clinicians, policymakers is critical advancing addressing burden effectively.

Язык: Английский

Процитировано

1

Combination of Machine Learning and COSMO-RS Thermodynamic Model in Predicting Solubility Parameters of Coformers in Production of Cocrystals for Enhanced Drug Solubility DOI
Wael A. Mahdi, Ahmad J. Obaidullah

Chemometrics and Intelligent Laboratory Systems, Год журнала: 2024, Номер 253, С. 105219 - 105219

Опубликована: Авг. 23, 2024

Язык: Английский

Процитировано

4

An exploration of the ocular mysteries linking nanoparticles to the patho-therapeutic effects against keratitis DOI Creative Commons

Siying Qu,

Shuihua Zheng,

Saleh Muhammad

и другие.

Journal of Nanobiotechnology, Год журнала: 2025, Номер 23(1)

Опубликована: Март 6, 2025

Microbial keratitis, a sight-threatening corneal infection, remains significant global health concern. Conventional therapies using antimicrobial agents often suffers from limitations such as poor drug penetration, side effects, and occurrence of resistance, with prognosis. Novel treatment techniques, their unique properties targeted delivery capabilities, offers promising solution to overcome these challenges. This review delves into timely update the state-of-the-art advance therapeutics for keratitis treatment. The diverse microbial origins including viral, bacterial, fungal infections, exploring complex pathogenic mechanisms, followed by resistance mechanisms in pathogens are reviewed briefly. Importantly, emerging therapeutic techniques piezodynamic therapy, photothermal photodynamic nanoenzyme metal ion therapy summarized this showcasing potential traditional treatments. challenges future directions nanotechnology-based approaches discussed, focusing on safety, targeting strategies, combination therapies. aims inspire researchers revolutionize accelerate development functional materials different

Язык: Английский

Процитировано

0

Advances in Nanoparticles in Targeted Drug Delivery- A Review DOI Creative Commons
Safiul Islam, Md Mir Shakib Ahmed, Mohammad Aminul Islam

и другие.

Results in Surfaces and Interfaces, Год журнала: 2025, Номер unknown, С. 100529 - 100529

Опубликована: Апрель 1, 2025

Язык: Английский

Процитировано

0

Anti-fungal peptides: an emerging category with enthralling therapeutic prospects in the treatment of candidiasis DOI
Jyoti Sankar Prusty, Ashwini Kumar, Awanish Kumar

и другие.

Critical Reviews in Microbiology, Год журнала: 2024, Номер unknown, С. 1 - 37

Опубликована: Окт. 23, 2024

infections, particularly invasive candidiasis, pose a serious global health threat.

Язык: Английский

Процитировано

0

Layer-by-Layer Biopolymer-Coated Deformable Liposomes–In Situ Gel: A Hybrid Strategy for Enhanced Ocular Delivery of Itraconazole: In Vitro and In Vivo Appraisal DOI Creative Commons

Mohamed M. Badran,

Areej Alsubaie,

Mounir M. Salem‐Bekhit

и другие.

Gels, Год журнала: 2024, Номер 11(1), С. 19 - 19

Опубликована: Дек. 31, 2024

Itraconazole (ITZ) is a potent antifungal agent. Its oral administration associated with systemic toxicity, and its efficacy in ocular formulations limited. This study aims to enhance ITZ’s permeation by loading it into deformable liposomes (DLs) based on Tween 80 (T) or Poloxamer 188 (P). Moreover, ITZ was loaded biopolymer-coated DLs augment availability. ITZ-loaded were coated hyaluronic acid (HA-DLs), chitosan (CS-DLs), layer-by-layer coating (CS/HA-DLs). These further laden pH-sensitive situ gels provide hybrid system intensify their adhesion properties. The prepared successfully vesicle sizes nonorange (<200 nm). zeta potential values of DLS negative before shifted high negativity HA positivity CS CS/HA bilayer coating. variations indicate successful coatings. optimized A EE% achieved DLs-T: 89% (CS/HA-DLs-T), 86% (CS-DLs-T), 85% (HA-DLs-T), 79% (HA-DLs-T). Therefore, DLs-T incorporated gels, displaying optimal gelling capacity viscosity. release rate from the DLs-laden slower than that observed uncoated DLs-gel. CS/HA-DLs-T laden-in showed highest ex vivo transcorneal permeability efficacy. data suggest layer-by-layer-CS/HA-DLs-T presents hopeful strategy for delivery ITZ, offering promising approach managing fungal infections.

Язык: Английский

Процитировано

0