Construction of Spiro[pyrrolidine-azlactone] via [2 + 3] Cycloaddition of Alkylidene Azlactone with Trifluoromethylated Imine DOI

Lesong Li,

Xia Wang, Yang Wang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Ноя. 13, 2024

A Ag-catalyzed [2 + 3] cycloaddition of alkylidene azlactones with trifluoromethylated imines has been documented, providing spiro[pyrrolidine-azlactones] bearing four adjacent stereogenic centers good yields and excellent diastereoselectivities. Catalytic asymmetric also developed enantioselectivities. Further gram-scale preparation synthetic transformation to pyrrolidine derivative showed the practicality applicability this reaction.

Язык: Английский

Dehydrogenation of Aromatic Alcohols, Aldehydes, and Ketones Catalyzed by Cu(I) Complexes DOI
Yangyang Shen, Xiaobin Li,

Fei Chen

и другие.

The Journal of Organic Chemistry, Год журнала: 2025, Номер unknown

Опубликована: Фев. 11, 2025

Herein, we report that binuclear copper complexes used as dehydrogenative catalysts, combined with oxygen an oxidant and 2,2,6,6-tetramethylpiperidinyl-1-oxide (TEMPO) additive, are capable of effectively catalyzing the successive dehydrogenation aromatic propanols to produce α,β-unsaturated aldehydes. This method has advantages high efficiency, simple operation, oxidant. The reaction mechanism continuous was investigated by in situ infrared spectroscopy control experiments. process suggested phenylpropanol first oxidized arylpropanals then underwent α,β-selective carbonyl group yield protocol provides insights into design synthesis efficient catalysts for preparation aldehydes propanols.

Язык: Английский

Процитировано

0

Photoinduced Site-Selective Alkylation Enabling Synthesis of C-3-Alkylated Quinoxalinone on DNA DOI

Kyeong Seop Kim,

Junseok Ra,

Madala Hari Babu

и другие.

Organic Letters, Год журнала: 2025, Номер unknown

Опубликована: Апрель 30, 2025

A mild and biocompatible strategy for the site-selective alkylation of quinoxalinones via photoinduced dehydrogenative has been developed. This protocol enables functionalization both unprotected quinoxalinone nonreactive dihydroquinoxalinone under DNA-compatible conditions. The optimized reaction proceeds efficiently while tolerating a diverse range alkyl donors from various radical precursors. Given its simplicity DNA compatibility, this methodology offers platform construction DNA-encoded libraries incorporating privileged scaffold.

Язык: Английский

Процитировано

0

Enhanced catalytic performance for aerobic dehydrogenation of N-heterocycles over bimetallic CoOX-CeO2 catalysts derived from Ce-based MOFs DOI
Zhixian Wang,

Ruibi Zhao,

Wenjing Li

и другие.

Molecular Catalysis, Год журнала: 2024, Номер 567, С. 114450 - 114450

Опубликована: Авг. 15, 2024

Язык: Английский

Процитировано

0

Efficient CuOAc/DMAP/DEAD‐Catalyzed Aerobic Oxidative Synthesis of Quinazolines DOI
Yue Ji,

Ze‐Lin Dang,

Menglong Niu

и другие.

ChemistrySelect, Год журнала: 2024, Номер 9(39)

Опубликована: Окт. 1, 2024

Abstract Efficient approaches toward the synthesis of quinazolines and dihydroisoquinolines have been developed through copper‐catalyzed aerobic oxidative dehydrogenation N ‐heterocycles. The was achieved azodicarboxylate esters‐mediated amines. Azodicarboxylate esters could be regenerated from corresponding hydrazodicarboxylate esters, which made this catalytic process more efficient reactive.

Язык: Английский

Процитировано

0

Construction of Spiro[pyrrolidine-azlactone] via [2 + 3] Cycloaddition of Alkylidene Azlactone with Trifluoromethylated Imine DOI

Lesong Li,

Xia Wang, Yang Wang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер unknown

Опубликована: Ноя. 13, 2024

A Ag-catalyzed [2 + 3] cycloaddition of alkylidene azlactones with trifluoromethylated imines has been documented, providing spiro[pyrrolidine-azlactones] bearing four adjacent stereogenic centers good yields and excellent diastereoselectivities. Catalytic asymmetric also developed enantioselectivities. Further gram-scale preparation synthetic transformation to pyrrolidine derivative showed the practicality applicability this reaction.

Язык: Английский

Процитировано

0