Development and Characterization of Tannic Acid‐Modified PVA‐κCarrageenan Gel for Sustained Release of Lidocaine DOI
Anita Marlina, Misni Misran, Sun Theo Constan Lotebulo Ndruru

и другие.

ChemistrySelect, Год журнала: 2024, Номер 9(37)

Опубликована: Сен. 27, 2024

Abstract PVA‐κcarrageenan (κCar) gel is widely used in the pharmaceutical field for transdermal drug delivery, enhancing stability and bioavailability. This study aims to modify PVA‐κCar by introducing tannic acid. Lidocaine was as a model incorporation into novel gel. The matrix mixed with acid prior freeze– thaw cycle create composite. physicochemical features of this were evaluated using FTIR, XRD, thermal analysis, SEM. presence has reduced from 84 around 70 °C. content acid‐modified 34.6% (A) 52.1% (B). addition substantially increased viscosity. Cytotoxicity analysis showed that did not affect viability HCT colon cancer cells. encapsulation efficiency lidocaine 13 ± 0.2% 12 0.5% (B), while loading 0.96 0.01 0.91 0.02 In vitro release modified exhibited sustained mechanism phosphate‐buffered saline solution. These findings indicate possesses advantageous characteristics carrier.

Язык: Английский

Waste-to-resource: Extraction and transformation of aquatic biomaterials for regenerative medicine DOI

Huaqi Cao,

Yuanjin Zeng,

Xueyu Yuan

и другие.

Biomaterials Advances, Год журнала: 2024, Номер 166, С. 214023 - 214023

Опубликована: Сен. 1, 2024

Язык: Английский

Процитировано

2

Chitosan-ricobendazole complex: Synthesis, characterization and anthelmintic activity DOI
А.В. Блинов, Владимир Оробец, Elena Kastarnova

и другие.

International Journal of Biological Macromolecules, Год журнала: 2024, Номер 280, С. 135572 - 135572

Опубликована: Сен. 11, 2024

Язык: Английский

Процитировано

1

Incorporation of Capecitabine Into Extended Chain of N‐Acylated Chitosan Carrier DOI Creative Commons
Anita Marlina, Misni Misran, Witta Kartika Restu

и другие.

Advances in Polymer Technology, Год журнала: 2024, Номер 2024(1)

Опубликована: Янв. 1, 2024

Enhancing the hydrophobicity of chitosan through acylation enables encapsulation water‐insoluble drugs within polymeric carrier cores. In this study, hydrophobically modified was synthesized by reacting low‐molecular‐weight with acyl chloride (C18–C24) using an agitation method under mild conditions. The structure acylated analyzed FTIR and 1 H‐NMR spectroscopy. degree substitution (DS) varied between 56% 69% for different long‐chain N‐acylated chitosan, N‐stearoyl (ChC18) exhibiting highest DS. incorporation capecitabine (CAP) into extended increased particle size decreased zeta potential. N‐lignoceroyl (ChC24) exhibited potential value −27 mV 0.2 mg CAP, indicating that most group stable in suspension. Transmission electron microscope images revealed all particles were spherical, sizes ranging from 100 to 200 nm, existed as stand‐alone entities, excellent stability loading CAP but did not alter shape, except ChC24, which agglomeration. SEM individual arrangement CAP‐ChC18 made it more than other chitosan. contrast, formation clusters CAP‐ChC24 can be attributed strong hydrophobic interactions. X‐ray photoelectron spectroscopy results show there is no nitrogen atom ChC18, means oriented inward bound stearoyl via van der Waals forces. At drug weight‐to‐carrier ratios, efficiency (EE) varying lengths ranged 85% 97%. (DL) capacity EE amount increased. However, length significantly affect DL EE, even when carrier‐to‐drug ratio consistently maintained. Sustained release observed CAP‐loaded a significant influence chain on Consequently, possesses enormous delivery system CAP.

Язык: Английский

Процитировано

1

Development and Characterization of Tannic Acid‐Modified PVA‐κCarrageenan Gel for Sustained Release of Lidocaine DOI
Anita Marlina, Misni Misran, Sun Theo Constan Lotebulo Ndruru

и другие.

ChemistrySelect, Год журнала: 2024, Номер 9(37)

Опубликована: Сен. 27, 2024

Abstract PVA‐κcarrageenan (κCar) gel is widely used in the pharmaceutical field for transdermal drug delivery, enhancing stability and bioavailability. This study aims to modify PVA‐κCar by introducing tannic acid. Lidocaine was as a model incorporation into novel gel. The matrix mixed with acid prior freeze– thaw cycle create composite. physicochemical features of this were evaluated using FTIR, XRD, thermal analysis, SEM. presence has reduced from 84 around 70 °C. content acid‐modified 34.6% (A) 52.1% (B). addition substantially increased viscosity. Cytotoxicity analysis showed that did not affect viability HCT colon cancer cells. encapsulation efficiency lidocaine 13 ± 0.2% 12 0.5% (B), while loading 0.96 0.01 0.91 0.02 In vitro release modified exhibited sustained mechanism phosphate‐buffered saline solution. These findings indicate possesses advantageous characteristics carrier.

Язык: Английский

Процитировано

0