Metal‐Free Direct Synthesis of N‐Sulfonyl Amidines from Thioamides and Electron Deficient N‐Sulfonylamides DOI
Jigarkumar K. Vankar, Srinu Tothadi, Guddeangadi N. Gururaja

и другие.

European Journal of Organic Chemistry, Год журнала: 2024, Номер 27(45)

Опубликована: Авг. 29, 2024

Abstract A metal‐free, efficient synthesis of N ‐sulfonyl amidines has been demonstrated from easily accessible thioamides and electron‐deficient sulfonyl amides. The amidation reaction is facile at room temperature with low amide loading. illustrated various amides broad substrate scope. utility amidine validated late‐stage drug functionalization.

Язык: Английский

1,1,1,3,3,3-Hexafluoro-2-propanol (HFIP)-promoted regiospecific 1,6-hydroarylation of para-quinone methides with N-heteroarenes: Synthesis of unsymmetrical triarylmethanes DOI
Haiyan Xu,

C. K. LIANG,

Junyu Zhu

и другие.

Tetrahedron, Год журнала: 2024, Номер 158, С. 133982 - 133982

Опубликована: Апрель 7, 2024

Язык: Английский

Процитировано

2
Metal‐Free Direct Synthesis of N‐Sulfonyl Amidines from Thioamides and Electron Deficient N‐Sulfonylamides DOI
Jigarkumar K. Vankar, Srinu Tothadi, Guddeangadi N. Gururaja

и другие.

European Journal of Organic Chemistry, Год журнала: 2024, Номер 27(45)

Опубликована: Авг. 29, 2024

Abstract A metal‐free, efficient synthesis of N ‐sulfonyl amidines has been demonstrated from easily accessible thioamides and electron‐deficient sulfonyl amides. The amidation reaction is facile at room temperature with low amide loading. illustrated various amides broad substrate scope. utility amidine validated late‐stage drug functionalization.

Язык: Английский

Процитировано

0