Preparation and Characterization of Tiamulin-Loaded Niosomes for Oral Bioavailability Enhancement in Mycoplasma-Infected Broilers DOI Creative Commons

Shimaa G. Abonashey,

Amr Gamal, Hatem A. F. M. Hassan

и другие.

Micro, Год журнала: 2024, Номер 4(4), С. 734 - 750

Опубликована: Ноя. 27, 2024

Mycoplasma infections pose significant challenges in the poultry industry, necessitating effective therapeutic interventions. Tiamulin, a veterinary antibiotic, has demonstrated efficacy against species. However, emergence of resistant species could dramatically reduce potential, contributing to economic losses. Optimizing tiamulin’s pharmacokinetic profile via nanocarrier incorporation enhance its potential and administration frequency, ultimately reducing strain emergence. Niosomes, type self-assembled non-ionic surfactant-based nanocarrier, have emerged as promising drug delivery system, offering improved stability, sustained release, enhanced bioavailability. In this study, niosomal nanocarriers encapsulating tiamulin were prepared, characterized assessed Mycoplasma-inoculated broilers following oral administration. Differential scanning colorimetry (DSC) confirmed alterations crystalline state components integration into structures formed during formulation procedure. Transmission electron microscopy (TEM) showed spherical nanostructure niosomes. The formulated exhibited zeta average hydrodynamic diameter −10.65 ± 1.37 mV 339.67 30.88 nm, respectively. Assessment parameters gallisepticum-infected revealed ability increase bioavailability systemic exposure, marked by significantly higher area under curve (AUC) (p < 0.01) prolonged elimination half-life (T1/2) 0.05). Enhanced residence time are crucial factors maintaining concentrations at reduced doses frequencies. This approach provides viable strategy decrease risk subtherapeutic levels, thereby mitigating development antibiotic resistance. findings presented herein offer sustainable for efficient use antibiotics medicine.

Язык: Английский

Electrospinning in Drug Delivery: Progress and Future Outlook DOI Open Access

Naimah Abdul Halim,

N. Nallusamy, Rajamani Lakshminarayanan

и другие.

Macromolecular Rapid Communications, Год журнала: 2025, Номер unknown

Опубликована: Фев. 20, 2025

Abstract There is intense research during the past few decades to design and fabricate drug delivery systems using electrospinning system. Electrospinning an efficient technique produce nanofiber materials with different dimensions morphologies by adjusting processing parameters. becoming innovative technology that promotes pursuit maintenance of human health. Herein, review discusses contribution in systems, summarising modification various system configurations effects process parameters on fibers, their application including carrier materials, loaded drugs release mechanisms illustrates medical applications. Finally, this challenges, bottlenecks, development prospects field terms scaling up for clinical use exploring potential solutions pave way establish future systems.

Язык: Английский

Процитировано

1

Synergistic Enhancement of Carboplatin Efficacy through pH-Sensitive Nanoparticles Formulated Using Naturally Derived Boswellia Extract for Colorectal Cancer Therapy DOI Creative Commons
Sherif Ashraf Fahmy, Nada K. Sedky, Hatem A. F. M. Hassan

и другие.

Pharmaceutics, Год журнала: 2024, Номер 16(10), С. 1282 - 1282

Опубликована: Сен. 30, 2024

Carboplatin (Cp) is a potent chemotherapeutic agent, but its effectiveness constrained by associated side effects. Frankincense, an oleo-gum resin from the

Язык: Английский

Процитировано

4

Nano/Micro-Enabled Modification and Innovation of Conventional Adjuvants for Next-Generation Vaccines DOI Creative Commons
Xingchi Liu,

Yang Xu,

Tao Lu

и другие.

Journal of Functional Biomaterials, Год журнала: 2025, Номер 16(5), С. 185 - 185

Опубликована: Май 19, 2025

The global spread of infectious diseases has raised public awareness vaccines, highlighting their essential role in protecting health. Among the components modern adjuvants have received increasing attention for boosting immune responses and enhancing efficacy. Recent advancements adjuvant research, particularly nanodelivery systems, paved way developing more effective safer adjuvants. This review outlines properties, progress, mechanisms FDA-approved conventional adjuvants, focusing on contributions to challenges vaccine success. Despite these advancements, still face suboptimal immunomodulatory effects, potential side limitations targeting specific pathways. Nanodelivery systems emerged as a transformative approach design, offering unique advantages such stability, enabling controlled antigen release, inducing responses. By addressing limitations, nanocarriers improve safety efficacy drive development next-generation complex diseases. also explores strategies incorporating into development, emphasizing its optimizing formulations. summarizing current recent advances, this aims provide valuable insights guiding future efforts designing innovative that meet evolving needs immunization programs.

Язык: Английский

Процитировано

0

Sustainable Nanomedicine: Enhancement of Asplatin’s Cytotoxicity In Vitro and In Vivo Using Green-Synthesized Zinc Oxide Nanoparticles Formed via Microwave-Assisted and Gambogic Acid-Mediated Processes DOI Creative Commons
Hatem A. F. M. Hassan, Nada K. Sedky, Mohamed S. Nafie

и другие.

Molecules, Год журнала: 2024, Номер 29(22), С. 5327 - 5327

Опубликована: Ноя. 12, 2024

Chemoresistance encountered using conventional chemotherapy demands novel treatment approaches. Asplatin (Asp), a platinum (IV) prodrug designed to release cisplatin and aspirin in reductive environment, has demonstrated high cytotoxicity at reduced drug resistance. Herein, we investigated the ability of green-synthesized nanocarriers enhance Asp’s efficacy. Zinc oxide nanoparticles (ZnO-NPs) were synthesized green microwave-assisted method with reducing capping agent gambogic acid (GA). These then loaded Asp, yielding Asp@ZnO-NPs. Transmission electron microscopy was utilized study morphological features ZnO-NPs. Cell viability studies conducted on MDA-MB-231 breast cancer cells Asp@ZnO-NPs significantly decrease half-maximal inhibitory concentration (IC50) (5 ± 1 µg/mL). This further flow cytometric analysis that revealed capacity increase late apoptotic fractions. Furthermore, vivo carried out solid Ehrlich carcinoma-bearing mice showed significant tumor volume reduction (156.3 7.6 mm3), compared Asp alone (202.3 8.4 mm3) untreated controls (342.6 10.3 mm3). The histopathological increased necrosis Asp@ZnO-NPs-treated group. Asp@ZnO-NPs, an eco-friendly approach, enhanced anticancer activity, offering sustainable solution for potent formulations.

Язык: Английский

Процитировано

1

Preparation and Characterization of Tiamulin-Loaded Niosomes for Oral Bioavailability Enhancement in Mycoplasma-Infected Broilers DOI Creative Commons

Shimaa G. Abonashey,

Amr Gamal, Hatem A. F. M. Hassan

и другие.

Micro, Год журнала: 2024, Номер 4(4), С. 734 - 750

Опубликована: Ноя. 27, 2024

Mycoplasma infections pose significant challenges in the poultry industry, necessitating effective therapeutic interventions. Tiamulin, a veterinary antibiotic, has demonstrated efficacy against species. However, emergence of resistant species could dramatically reduce potential, contributing to economic losses. Optimizing tiamulin’s pharmacokinetic profile via nanocarrier incorporation enhance its potential and administration frequency, ultimately reducing strain emergence. Niosomes, type self-assembled non-ionic surfactant-based nanocarrier, have emerged as promising drug delivery system, offering improved stability, sustained release, enhanced bioavailability. In this study, niosomal nanocarriers encapsulating tiamulin were prepared, characterized assessed Mycoplasma-inoculated broilers following oral administration. Differential scanning colorimetry (DSC) confirmed alterations crystalline state components integration into structures formed during formulation procedure. Transmission electron microscopy (TEM) showed spherical nanostructure niosomes. The formulated exhibited zeta average hydrodynamic diameter −10.65 ± 1.37 mV 339.67 30.88 nm, respectively. Assessment parameters gallisepticum-infected revealed ability increase bioavailability systemic exposure, marked by significantly higher area under curve (AUC) (p < 0.01) prolonged elimination half-life (T1/2) 0.05). Enhanced residence time are crucial factors maintaining concentrations at reduced doses frequencies. This approach provides viable strategy decrease risk subtherapeutic levels, thereby mitigating development antibiotic resistance. findings presented herein offer sustainable for efficient use antibiotics medicine.

Язык: Английский

Процитировано

0