An exploratory study of the safety profile and neurocognitive function after single doses of mitragynine in humans DOI Creative Commons
Elisabeth Prevete, Eef L. Theunissen, Kim P. C. Kuypers

и другие.

Psychopharmacology, Год журнала: 2024, Номер unknown

Опубликована: Дек. 26, 2024

Despite the growing scientific interest on mitragynine, primary alkaloid in kratom (Mitragyna Speciosa), there is a lack of clinical trials humans. This phase 1 study aimed to evaluate mitragynine's safety profile and acute effects subjective drug experience, neurocognition, pain tolerance. A placebo-controlled, single-blind, within-subjects was conducted two parts. In part A, eight healthy human volunteers received placebo three doses mitragynine (5, 10, 20 mg) sequential dosing scheme, separate days. B, second group seven 40 mg mitragynine. Vital signs, neurocognitive function, tolerance were measured at regular intervals for 7 h after administration. Overall, did not affect most outcome measures any dose. Yet, lowest dose (5 increased ratings arousal attention, accuracy sustained attention task, motor inhibition. The highest (40 amnesia produced mild psychopathological symptoms. Mitragynine significantly vital only mild, transient side reported. present suggests that low (5–10 may cause feelings stimulation enhance while inhibitory distress. up well tolerated this group.

Язык: Английский

Kratom safety and toxicology in the public health context: research needs to better inform regulation DOI Creative Commons
Jack E. Henningfield, Oliver Grundmann, Marilyn A. Huestis

и другие.

Frontiers in Pharmacology, Год журнала: 2024, Номер 15

Опубликована: Июнь 3, 2024

Although kratom use has been part of life for centuries in Southeast Asia, the availability and United States (US) increased substantially since early 2000s when there was little information on pharmacology, patterns, effects, all critical to guiding regulation policy. Here we provide a synthesis research with several hundred English-language papers published past 5 years drawing from basic research, epidemiological surveillance data, recent clinical research. This review available literature aims an integrated update regarding our current understanding kratom’s benefits, risks, epidemiology, which may inform States-based regulation. Recent indicates are likely million past-year consumers, though estimates vary widely. Even without precise prevalence is no longer niche, millions adults using it myriad reasons. Despite its botanical origins coffee tree family polypharmacy, popularly characterized as opioid presumed opioid-system-based risks addiction or overdose. Neuropharmacology, toxicology, epidemiology studies show that more accurately substance diverse complex pharmacology. Taken together work reviewed here provides foundation future scientific studies, well guide ongoing efforts regulate kratom. also informs much-needed federal oversight, including by Food Drug Administration. We conclude recommendations priorities needed address policy knowledge gaps around this increasingly used product.

Язык: Английский

Процитировано

11

Chemical Analysis and Alkaloid Intake for Kratom Products Available in the United States DOI
Abhisheak Sharma, Kirsten E. Smith, Michelle A. Kuntz

и другие.

Drug Testing and Analysis, Год журнала: 2025, Номер unknown

Опубликована: Май 16, 2025

ABSTRACT Previously, we used ecological momentary assessment (EMA) to evaluate motivations and temporal patterns of kratom use for 15 days among US adult consumers ( N = 357). Here present the content analyses products during that nationwide study, with quantification 10 alkaloids. The samples 341) were primarily whole‐leaf products, not extracts, similar each other in their alkaloid composition, closely matching chromatographic‐mass spectrometry fingerprint expected Mitragyna speciosa leaf material. We found no evidence adulteration illicit or prescription drugs. With participants' self‐reported data on amount per use, calculated mitragynine intake use: mean 31.3 mg median 25.4 (range 2.0–205.9 mg). frequency, day, it ranged from 78.3 134.6 (mean) 50.8 101.6 (median). This is most comprehensive analysis date. coupling self‐report product sample‐analysis quantify daily foundational designing controlled clinical trials healthy volunteers. These findings products' chemical composition consumption can also inform clinicians, policymakers, consumers, particularly

Язык: Английский

Процитировано

0

Controversies in Assessment, Diagnosis, and Treatment of Kratom Use Disorder DOI Creative Commons
Kirsten E. Smith, David H. Epstein, Stephanie T. Weiss

и другие.

Current Psychiatry Reports, Год журнала: 2024, Номер 26(9), С. 487 - 496

Опубликована: Авг. 13, 2024

We apply the Diagnostic and Statistical Manual of Mental Disorders Fifth Edition (DSM-5) criteria for substance use disorders (SUDs) to herbal product kratom. Similarities differences between kratom disorder (KUD) other SUDs are explored, along with assessment, diagnostic, therapeutic recommendations KUD.

Язык: Английский

Процитировано

2

An exploratory study of the safety profile and neurocognitive function after single doses of mitragynine in humans DOI Creative Commons
Elisabeth Prevete, Eef L. Theunissen, Kim P. C. Kuypers

и другие.

Psychopharmacology, Год журнала: 2024, Номер unknown

Опубликована: Дек. 26, 2024

Despite the growing scientific interest on mitragynine, primary alkaloid in kratom (Mitragyna Speciosa), there is a lack of clinical trials humans. This phase 1 study aimed to evaluate mitragynine's safety profile and acute effects subjective drug experience, neurocognition, pain tolerance. A placebo-controlled, single-blind, within-subjects was conducted two parts. In part A, eight healthy human volunteers received placebo three doses mitragynine (5, 10, 20 mg) sequential dosing scheme, separate days. B, second group seven 40 mg mitragynine. Vital signs, neurocognitive function, tolerance were measured at regular intervals for 7 h after administration. Overall, did not affect most outcome measures any dose. Yet, lowest dose (5 increased ratings arousal attention, accuracy sustained attention task, motor inhibition. The highest (40 amnesia produced mild psychopathological symptoms. Mitragynine significantly vital only mild, transient side reported. present suggests that low (5–10 may cause feelings stimulation enhance while inhibitory distress. up well tolerated this group.

Язык: Английский

Процитировано

0