The Application of Response Surface Methodology (RSM) In the Computational Optimization of Sustained Release (SR) For Phenothiazine Derivative Matrix Tablet DOI Open Access
Shiva Kant Thakur, Rahul Pal,

Devanand Jha

и другие.

Journal of Pharmaceutical Research International, Год журнала: 2023, Номер 35(35), С. 13 - 27

Опубликована: Дек. 28, 2023

Introduction: This study explores the use of Response Surface Methodology (RSM), a statistical optimization technique, to optimize SR properties prochlorperazine maleate (PCM) matrix tablets. PCM is phenothiazine derivative used for treating schizophrenia, nausea, and vomiting. Sustained-release formulations offer extended drug delivery, potentially improving patient compliance reducing side effects. RSM helps identify optimal combinations critical formulation factors influencing release, such as polymer type concentration, filler type, drug/polymer ratio. The likely involves designing experiments based on chosen designs (e.g., Box-Behnken) with varying factor levels. Formulate tablets different combinations. Evaluating release profiles each tablet formulation. Analyzing data using software build mathematical models relating identifying that maximize desired characteristics. Objective: ongoing research purpose improve advancement sustained containing Phenothiazine loaded matrix. achieved by utilizing DoE computational method statistically validate Methodology: Basically two methods involved in direct compression; simple efficient where all dry ingredients are blended directly compressed into Results: obtained outcomes closely matched anticipated values derived from experimental setup. enhanced demonstrated prolonged uniform discharge over span 6 hours. Conclusion: Based 23 FD, response surface methodology was successfully develop current application. corresponding contour plots 3D represent important variables optimisation process.

Язык: Английский

The Comprehensive Review: Exploring Future Potential of Nasopulmonary Drug Delivery Systems for Nasal Route Drug Administration DOI Open Access
Rahul Pal, Prachi Pandey,

Manju Koli

и другие.

Journal of Drug Delivery and Therapeutics, Год журнала: 2024, Номер 14(3), С. 126 - 136

Опубликована: Март 15, 2024

This comprehensive review aims to explore the future potential of nasopulmonary drug delivery systems for administration drugs through nasal route. Nasal has gained significant attention due its numerous advantages, including rapid absorption, avoidance first-pass metabolism, and non-invasive administration. provides an overview anatomy physiology, highlighting factors influencing absorption bioavailability. Additionally, it discusses various types systems, such as sprays, powders, gels, along with their advantages limitations. Furthermore, delves into challenges associated delivery, mucociliary clearance, irritation, formulation issues. The applications in treatment diseases, allergies, respiratory disorders, systemic conditions, are also discussed. Finally, concludes outlook on prospects emphasising need further research development optimise efficacy safety. Keywords: pulmonary; spray; mucosa; gels; drops; approaches; route; delivery.

Язык: Английский

Процитировано

8

An Updated Comprehensive Review on Novel Drug Delivery Systems (NDDS) In the Pharmaceuticals DOI Open Access

Vinay Kumar Rao Khadam,

Ravindra Pal Singh, Deepak Prajapati

и другие.

Asian Journal of Pharmaceutical Research and Development, Год журнала: 2024, Номер 12(1), С. 55 - 64

Опубликована: Фев. 15, 2024

The field of pharmaceutical sciences has witnessed a paradigm shift with the advent Novel Drug Delivery Systems (NDDS), which aim to enhance therapeutic efficacy, reduce side effects, and improve patient compliance. This comprehensive review explores latest advancements innovations in NDDS, encompassing diverse range delivery platforms strategies.(NDDs are transforming landscape treatment, offering unparalleled potential for enhanced improved bioavailability, controlled release, targeted delivery, stability. highlighting recent addressing key challenges. Prominent NDDS include liposomes, nanoparticles, micelles, polymeric drug conjugates, monoclonal antibodies, implants, patches. Each system possesses unique properties applications, tailored specific drugs needs. Recent breakthroughs nanocarriers, gene therapy vectors, 3D-printed personalized dosage forms pushing boundaries innovation. main highlights present firstly basics on NDDs, several approaches nano carriers their preparation methods example. middle version discuss techniques NDDs lastly marketed formulation particular carrier.

Язык: Английский

Процитировано

4

Nanoparticles (NPs) Based Drug Delivery System: An Inspiring Therapeutic Strategy for Cancer Therapy and Their Future Prospects DOI Open Access

I. Dutta,

Atibur Rahaman,

S.D. Singh

и другие.

Journal of Drug Delivery and Therapeutics, Год журнала: 2025, Номер 15(4), С. 133 - 143

Опубликована: Апрель 15, 2025

Nanoparticles (NPs)-based drug delivery systems (DDs) have emerged as a promising strategy for cancer therapy, offering targeted, controlled, and efficient while minimizing systemic toxicity. Their unique physicochemical properties, including high surface area, tunable size, enhanced permeability, enable precise tumor targeting through passive, active, stimuli-responsive mechanisms. The various nanocarriers such liposomes, polymeric NPs, dendrimers, metallic NPs been extensively explored chemotherapy, gene immunotherapy, theranostic applications. ability of to overcome multidrug resistance (MDR), enhance bioavailability, facilitate combination therapies has significantly improved treatment outcomes. Despite the remarkable advancements, challenges biocompatibility, large-scale production, regulatory approval remain critical hurdles. Future research will focus on personalized nanomedicine, smart multifunctional nanocarriers, gene-editing nanoparticle systems, green nanotechnology safer more effective treatments. continuous evolution in therapy holds immense potential transform oncology, paving way patient-specific, minimally invasive, highly modalities. This review article focuses lipid-based, polymeric, inorganic nanoparticles system their applications therapy. current limitations future perspectives nanoparticle-based DDS are also discussed. Keywords: Drug delivery, Nanocarriers, NDDS, Sustained, Targeted

Язык: Английский

Процитировано

0

A Traditional Review: The Utilization of Nutraceutical as a Traditional Cure for the Modern World at Current Prospectus for Multiple Health Conditions DOI Open Access
Prachi Pandey, Rahul Pal,

Manju Koli

и другие.

Journal of Drug Delivery and Therapeutics, Год журнала: 2024, Номер 14(3), С. 154 - 163

Опубликована: Март 15, 2024

Nutraceuticals refer to food products that have a positive impact on the well-being of individuals. This category includes dietary supplements, herbal products, probiotics, and prebiotics, as well medical foods designed for disease prevention treatment. The nutraceutical market is witnessing substantial growth worldwide, primarily due growing awareness among consumers about connection between diet health. Additionally, there rising demand functional supplements. As prioritize preventive healthcare, they are increasingly looking provide targeted health benefits beyond basic nutrition. rise this trend can be attributed various factors, including aging population, healthcare expenses, preference natural organic ingredients. Nutraceuticals, major force in industry, offer numerous beneficial effects with minimal undesirable impacts, thus attracting more consumer interest. increasing shift towards treatments, along disposable income outlook pharmaceutical sector, has contributed expanding India. However, challenges such lack regulation awareness, high pricing, marketing, distribution issues need addressed. Nutraceutical seeing flowing development chiefly United States, India, European nations. review article focuses providing concise overview nutraceuticals, categorizing them, discussing their significant roles conditions. it delves into present future status nutraceuticals global scale. Keywords: traditional cure; nutraceuticals; remedy; prebiotics; probiotics; regulatory compliance; supplementary diets;

Язык: Английский

Процитировано

2

The diverse marketed formulations of advanced nano drug carrier vehicles (and CVS) in different biomedical treatments: a complete descriptive review DOI Open Access
Rahul Pal, Prachi Pandey,

Vinay Kumar Rao Khadam

и другие.

Deleted Journal, Год журнала: 2024, Номер 15(2), С. 1 - 18

Опубликована: Апрель 30, 2024

The field of pharmaceutical science and drug delivery has seen a remarkable transformation in recent years, marked by the emergence diverse advanced approaches development Novel Drug Delivery Systems (NDDs) their associated carriers.Nanocarriers are tiny particles that can be used to deliver drugs body.They typically less than 100 nanometres diameter, which is about 1,000 times smaller width human hair.NDDs play pivotal role enhancing therapeutic efficacy, safety, patient compliance pharmaceuticals.The research community increasingly focused on creating novel systems address limitations conventional administration methods.The diversification these notable, reflecting interdisciplinary nature sciences.NDDs specific sites body, control rate release, protect from degradation.Carriers an important NDDs.The main highlights review articles focus nano carriers including niosome, liposome, aquasome, nanoparticles (NPs) phytosomes with marketed available different products specified disease targeting.1.

Язык: Английский

Процитировано

2

The Comprehensive Review: Internet Protocol (IP) Address a Primer for Digital Connectivity DOI Open Access

Mayank Kumar Tiwari,

Rahul Pal,

Riya Singh

и другие.

Asian Journal of Research in Computer Science, Год журнала: 2024, Номер 17(8), С. 34 - 45

Опубликована: Июль 16, 2024

The Internet Protocol (IP) is the rule book that governs how data addressed and routed across networks on internet. Think of it as postal system for digital world. This addressing allows routers, mail carriers, to efficiently transfer packets between devices until they reach their destination. It ensures reaches right place by assigning addresses enabling efficient routing. IP also encompasses various protocols services, such ICMP (Internet Control Message Protocol) error reporting diagnostics, DHCP (Dynamic Host Configuration automatic address assignment. Additionally, can be configured support different transmission modes, including uni-cast, multicast, broadcast, catering diverse communication requirements. Adopting technology has been researched developed commercially offers military a cost-effective method implementation. systems enable forces share common network supports voice, video, sharing. systematic review article initially highlighted basics lastly brief discussion regards gram format, NAT, IPv4, IPV6 fragmentation, CIDR, TCP UDP individually.

Язык: Английский

Процитировано

1

Coating Tablets, Compositions, Recent Advancement and Current Status: A Comprehensive Review DOI Open Access

Raj Kumar Mandal,

Paarth Saini,

Rahul Pal

и другие.

Journal of Drug Delivery and Therapeutics, Год журнала: 2024, Номер 14(10), С. 182 - 195

Опубликована: Окт. 15, 2024

Conventional Tablets are solid oral dosage forms that contain an active pharmaceutical ingredient (API) along with excipients. These tablets typically prepared through direct compression, wet granulation, or dry granulation. They designed to disintegrate and release the API in a controlled immediate manner, depending on formulation. Tablet coating is vital process technology, improve therapeutic efficacy, patient compliance, stability of forms. This comprehensive review explores key aspects tablet coating, including types, compositions, recent advancements. Coating materials such as polymers, plasticizers, pigments discussed detail, their roles controlling drug release, masking taste, enhancing aesthetic appeal. The advancements focus innovative techniques like film coatings, enteric application nanotechnology precision functionality. Additionally, current status analyzed terms regulatory compliance industry trends. highlights future potential personalized smart environmentally friendly approaches, showcasing evolving landscape technologies/pans modern manufacturing development. Keywords: Table coating; form; enteric; pans; formulation; advancement; polymers

Язык: Английский

Процитировано

1

The Application of Response Surface Methodology (RSM) In the Computational Optimization of Sustained Release (SR) For Phenothiazine Derivative Matrix Tablet DOI Open Access
Shiva Kant Thakur, Rahul Pal,

Devanand Jha

и другие.

Journal of Pharmaceutical Research International, Год журнала: 2023, Номер 35(35), С. 13 - 27

Опубликована: Дек. 28, 2023

Introduction: This study explores the use of Response Surface Methodology (RSM), a statistical optimization technique, to optimize SR properties prochlorperazine maleate (PCM) matrix tablets. PCM is phenothiazine derivative used for treating schizophrenia, nausea, and vomiting. Sustained-release formulations offer extended drug delivery, potentially improving patient compliance reducing side effects. RSM helps identify optimal combinations critical formulation factors influencing release, such as polymer type concentration, filler type, drug/polymer ratio. The likely involves designing experiments based on chosen designs (e.g., Box-Behnken) with varying factor levels. Formulate tablets different combinations. Evaluating release profiles each tablet formulation. Analyzing data using software build mathematical models relating identifying that maximize desired characteristics. Objective: ongoing research purpose improve advancement sustained containing Phenothiazine loaded matrix. achieved by utilizing DoE computational method statistically validate Methodology: Basically two methods involved in direct compression; simple efficient where all dry ingredients are blended directly compressed into Results: obtained outcomes closely matched anticipated values derived from experimental setup. enhanced demonstrated prolonged uniform discharge over span 6 hours. Conclusion: Based 23 FD, response surface methodology was successfully develop current application. corresponding contour plots 3D represent important variables optimisation process.

Язык: Английский

Процитировано

2