Extracellular Vesicles and PlantCrystals for Improved Bioavailability of Curcumin as a BCS Class IV Drug DOI Creative Commons

Muzn Alkhaldi,

Tehseen Sehra,

Soma Sengupta

и другие.

Molecules, Год журнала: 2024, Номер 29(24), С. 5926 - 5926

Опубликована: Дек. 16, 2024

The limited water solubility of active compounds remains a significant challenge for efficient dermal drug delivery, particularly BCS class IV drugs such as curcumin. This study aimed to enhance curcumin’s penetration using two strategies: extracellular vesicles (EVs) and plantCrystals derived from soybeans. EVs were isolated classical methods. However, containing (PCEVs) formed during the preparation through bead milling. Curcumin was either added after PCEVs formed, resulting in curcumin-added PCEVs, or soybean dispersion before milling, forming curcumin-loaded PCEVs. formulations characterized their physicochemical properties assessed efficacy quantitative dermatokinetic semi-quantitative ex vivo porcine ear models. results indicated that achieved higher compared EVs, with approximately 1.5-fold 2.7-fold increases efficacy, respectively. Additionally, showed superior depth, while curcumin remained stratum corneum. These findings suggest strategy via milling offers more effective approach than improving topical delivery like

Язык: Английский

Plant-Derived Extracellular Vesicles: Natural Nanocarriers for Biotechnological Drugs DOI Open Access
Eleonora Calzoni, Agnese Bertoldi, Gaia Cusumano

и другие.

Processes, Год журнала: 2024, Номер 12(12), С. 2938 - 2938

Опубликована: Дек. 23, 2024

Plant-derived extracellular vesicles (PDEVs) are lipid bilayer nanoparticles, naturally produced by plant cells, with sizes ranging from 50 to 500 nm. Recent studies have highlighted their great potential in the biotechnological and medical fields, due natural origin, high biocompatibility intrinsic therapeutic properties. PDEVs contain a complex biological cargo of proteins, lipids, nucleic acids secondary metabolites, including antioxidants anti-inflammatory molecules, making them ideal for biomedical applications such as drug delivery. These play key role intercellular communication gene regulation, proving be particularly promising personalized medicine. ability improve stability bioavailability, optimizing targeted release minimizing side effects. Despite some challenges, compositional variability need standardized protocols, at gunsight innovative research aimed improving loading capacity specificity. This review aims provide comprehensive overview PDEVs, exploring structure, isolation methods, functional characteristics, applications, highlighting advantages over synthetic nanoparticles animal-derived vesicles, leading an sustainable solution development new approaches.

Язык: Английский

Процитировано

4

Extracellular nanovesicles as neurotherapeutics for central nervous system disorders DOI Creative Commons

Naznin Bhom,

Khonzisizwe Somandi, Poornima Ramburrun

и другие.

Expert Opinion on Drug Delivery, Год журнала: 2024, Номер unknown

Опубликована: Дек. 7, 2024

Introduction The blood-brain barrier (BBB) is a highly selective structure that protects the central nervous system (CNS) while hindering delivery of many therapeutic agents. This presents major challenge in treating neurological disorders, such as multiple sclerosis, where effective drug to brain crucial for improving patient outcomes. Innovative strategies are urgently needed address this limitation.

Язык: Английский

Процитировано

1

Active herbal ingredients and drug delivery design for tumor therapy: a review DOI
Jing Han,

Y. Shen,

Ruiying Cao

и другие.

Chinese Journal of Natural Medicines, Год журнала: 2024, Номер 22(12), С. 1134 - 1162

Опубликована: Дек. 1, 2024

Язык: Английский

Процитировано

1

Revolutionizing Medicine: Harnessing Plant-Derived Vesicles for Therapy and Drug Transport DOI Creative Commons
Lu Li, Zhenkun Li, Xin Liu

и другие.

Heliyon, Год журнала: 2024, Номер 10(22), С. e40127 - e40127

Опубликована: Ноя. 1, 2024

Язык: Английский

Процитировано

0

Distribution and Incorporation of Extracellular Vesicles into Chondrocytes and Synoviocytes DOI Open Access
Takashi Ohtsuki,

Ikumi Sato,

Ren Takashita

и другие.

International Journal of Molecular Sciences, Год журнала: 2024, Номер 25(22), С. 11942 - 11942

Опубликована: Ноя. 6, 2024

Osteoarthritis (OA) is a chronic disease affecting over 500 million people worldwide. As the population ages and obesity rates rise, societal burden of OA increasing. Pro-inflammatory cytokines, particularly interleukin-1β, are implicated in pathogenesis OA. Recent studies suggest that crosstalk between cartilage synovium contributes to development, but mechanisms remain unclear. Extracellular vesicles (EVs) were purified from cell culture-conditioned medium via ultracentrifugation confirmed using transmission electron microscopy, nanoparticle tracking analysis, western blotting. We demonstrated EVs taken up by human synoviocytes chondrocytes vitro, while vivo experiments revealed fluorescent-labelled injected into mouse joints incorporated synoviocytes. EV uptake was significantly inhibited dynamin-mediated endocytosis inhibitors, indicating plays major role this process. Additionally, co-culture with HEK-293 cells expressing red fluorescent protein (RFP)-tagged CD9 chondrocytic line OUMS-27 transfer RFP-positive across 600-nm not 30-nm filter. These findings released joint fluid within cartilage, potentially facilitating communication synovium. The results underscore importance pathophysiology.

Язык: Английский

Процитировано

0

Extracellular Vesicles and PlantCrystals for Improved Bioavailability of Curcumin as a BCS Class IV Drug DOI Creative Commons

Muzn Alkhaldi,

Tehseen Sehra,

Soma Sengupta

и другие.

Molecules, Год журнала: 2024, Номер 29(24), С. 5926 - 5926

Опубликована: Дек. 16, 2024

The limited water solubility of active compounds remains a significant challenge for efficient dermal drug delivery, particularly BCS class IV drugs such as curcumin. This study aimed to enhance curcumin’s penetration using two strategies: extracellular vesicles (EVs) and plantCrystals derived from soybeans. EVs were isolated classical methods. However, containing (PCEVs) formed during the preparation through bead milling. Curcumin was either added after PCEVs formed, resulting in curcumin-added PCEVs, or soybean dispersion before milling, forming curcumin-loaded PCEVs. formulations characterized their physicochemical properties assessed efficacy quantitative dermatokinetic semi-quantitative ex vivo porcine ear models. results indicated that achieved higher compared EVs, with approximately 1.5-fold 2.7-fold increases efficacy, respectively. Additionally, showed superior depth, while curcumin remained stratum corneum. These findings suggest strategy via milling offers more effective approach than improving topical delivery like

Язык: Английский

Процитировано

0