Extracellular Vesicles and PlantCrystals for Improved Bioavailability of Curcumin as a BCS Class IV Drug DOI Creative Commons

Muzn Alkhaldi,

Tehseen Sehra,

Soma Sengupta

и другие.

Molecules, Год журнала: 2024, Номер 29(24), С. 5926 - 5926

Опубликована: Дек. 16, 2024

The limited water solubility of active compounds remains a significant challenge for efficient dermal drug delivery, particularly BCS class IV drugs such as curcumin. This study aimed to enhance curcumin’s penetration using two strategies: extracellular vesicles (EVs) and plantCrystals derived from soybeans. EVs were isolated classical methods. However, containing (PCEVs) formed during the preparation through bead milling. Curcumin was either added after PCEVs formed, resulting in curcumin-added PCEVs, or soybean dispersion before milling, forming curcumin-loaded PCEVs. formulations characterized their physicochemical properties assessed efficacy quantitative dermatokinetic semi-quantitative ex vivo porcine ear models. results indicated that achieved higher compared EVs, with approximately 1.5-fold 2.7-fold increases efficacy, respectively. Additionally, showed superior depth, while curcumin remained stratum corneum. These findings suggest strategy via milling offers more effective approach than improving topical delivery like

Язык: Английский

Plant-Derived Extracellular Vesicles: Natural Nanocarriers for Biotechnological Drugs DOI Open Access
Eleonora Calzoni, Agnese Bertoldi, Gaia Cusumano

и другие.

Processes, Год журнала: 2024, Номер 12(12), С. 2938 - 2938

Опубликована: Дек. 23, 2024

Plant-derived extracellular vesicles (PDEVs) are lipid bilayer nanoparticles, naturally produced by plant cells, with sizes ranging from 50 to 500 nm. Recent studies have highlighted their great potential in the biotechnological and medical fields, due natural origin, high biocompatibility intrinsic therapeutic properties. PDEVs contain a complex biological cargo of proteins, lipids, nucleic acids secondary metabolites, including antioxidants anti-inflammatory molecules, making them ideal for biomedical applications such as drug delivery. These play key role intercellular communication gene regulation, proving be particularly promising personalized medicine. ability improve stability bioavailability, optimizing targeted release minimizing side effects. Despite some challenges, compositional variability need standardized protocols, at gunsight innovative research aimed improving loading capacity specificity. This review aims provide comprehensive overview PDEVs, exploring structure, isolation methods, functional characteristics, applications, highlighting advantages over synthetic nanoparticles animal-derived vesicles, leading an sustainable solution development new approaches.

Язык: Английский

Процитировано

3

Engineering Strategies of Plant-Derived Exosome-Like Nanovesicles: Current Knowledge and Future Perspectives DOI Creative Commons
Yuhan Li, Yulong Wang,

Hongrui Zhao

и другие.

International Journal of Nanomedicine, Год журнала: 2024, Номер Volume 19, С. 12793 - 12815

Опубликована: Ноя. 1, 2024

Plant-derived exosome-like nanovesicles (PELNs) from edible plants, isolated by ultracentrifugation, size exclusion chromatography or other methods, were proved to contain a variety of biologically active and therapeutically specific components. Recently, investigations in the field PELN-based biomedicine have been conducted, which positioned those as promising tools for prevention treatment several diseases, with their natural origin potentially offering superior biocompatibility bioavailability. However, inadequate targeting limited therapeutic effects constrain utility clinical translation PELNs. Thus, strategies aiming at bridging gap engineering PELNs great interest. Those approaches include membrane hybridization, physical chemical surface functionalization encapsulation payloads. Herein, we provide comprehensive overview biogenesis composition, isolation purification methods characterization PELNs, well functions. Current knowledge on construction biomedical application engineered reviewed. Additionally, future directions perspectives this discussed order further enrich expand prospects

Язык: Английский

Процитировано

1

Extracellular Vesicles and PlantCrystals for Improved Bioavailability of Curcumin as a BCS Class IV Drug DOI Creative Commons

Muzn Alkhaldi,

Tehseen Sehra,

Soma Sengupta

и другие.

Molecules, Год журнала: 2024, Номер 29(24), С. 5926 - 5926

Опубликована: Дек. 16, 2024

The limited water solubility of active compounds remains a significant challenge for efficient dermal drug delivery, particularly BCS class IV drugs such as curcumin. This study aimed to enhance curcumin’s penetration using two strategies: extracellular vesicles (EVs) and plantCrystals derived from soybeans. EVs were isolated classical methods. However, containing (PCEVs) formed during the preparation through bead milling. Curcumin was either added after PCEVs formed, resulting in curcumin-added PCEVs, or soybean dispersion before milling, forming curcumin-loaded PCEVs. formulations characterized their physicochemical properties assessed efficacy quantitative dermatokinetic semi-quantitative ex vivo porcine ear models. results indicated that achieved higher compared EVs, with approximately 1.5-fold 2.7-fold increases efficacy, respectively. Additionally, showed superior depth, while curcumin remained stratum corneum. These findings suggest strategy via milling offers more effective approach than improving topical delivery like

Язык: Английский

Процитировано

0