I2-Mediated [3 + 3] Annulation for the Construction of Indole-Pyrimidine-Pyrazole-Fused Tetracyclic Heteroarenes DOI

Heng-Tong Qu,

Long-Sheng Zhou,

Jiaxin Yang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(20), С. 15164 - 15169

Опубликована: Окт. 7, 2024

An I2-mediated annulation of 3-aminopyrazoles with indole-3-carboxaldehydes has been demonstrated for the first time. This tandem strategy allows facile construction indole-pyrimidine-pyrazole-fused tetracyclic heteroarenes that are otherwise inaccessible by existing methods. These fused heterocycles exhibited enhanced antifungal activities against Valsa mali and Botryosphaeria dothidea compared commercial Xemium fungicide.

Язык: Английский

Electrochemical Atom Transfer Radical Addition of Polychloroalkanes to Olefins Promoted by 4,4‐Ditert‐butyl Bipyridine DOI

Fei Lian,

Fei‐Xian Luo, Meng Wang

и другие.

Chinese Journal of Chemistry, Год журнала: 2023, Номер 41(13), С. 1583 - 1588

Опубликована: Фев. 14, 2023

Comprehensive Summary A new electrochemical strategy for the atom transfer radical addition (ATRA) of polychloroalkanes across olefins has been realized by synergism paired electrolysis and halogen bonding activation. Notably, readily accessible 4,4‐di‐ tert ‐butyl bipyridine (dtbpy), acting as a acceptor, shifted reduction potential C—Cl bonds positively 110 mV. The decreased operating leads to wide substrate scope excellent functional group compatibility. diverse array terminal internal alkenes such (hetero)aryl olefins, unactive aliphatic natural products drugs‐derived were well compatible.

Язык: Английский

Процитировано

21

Recent Advances toward Electro- and Electrophotochemical 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone (DDQ)-Catalyzed C—H/C—F Bonds Functionalization DOI
Yongmei Li,

Liangbo Sun,

Kun Xu

и другие.

Chinese Journal of Organic Chemistry, Год журнала: 2025, Номер 45(2), С. 668 - 668

Опубликована: Янв. 1, 2025

Язык: Английский

Процитировано

0

Role of delocalized electrons on the doping effect in vanadia DOI Creative Commons

Ran Luo,

Sai Chen, Xin Chang

и другие.

Chem, Год журнала: 2023, Номер 9(8), С. 2255 - 2266

Опубликована: Май 12, 2023

Язык: Английский

Процитировано

8

When transition-metal catalysis meets electrosynthesis: a recent update DOI
Fei Lian, Jiuling Li, Kun Xu

и другие.

Organic & Biomolecular Chemistry, Год журнала: 2024, Номер 22(22), С. 4390 - 4419

Опубликована: Янв. 1, 2024

The merger of organic electrosynthesis with 3d transition-metal catalysis has offered huge opportunities for modern synthesis. This review summarizes the key advancements in this direction published recent two years.

Язык: Английский

Процитировано

3

Electrochemical Cobalt-Catalyzed C-H Hydroxyalkylation of N-Heteroarenes with Trifluoromethyl Ketones DOI Open Access
Huiqiao Wang,

Kun Xu

Chinese Journal of Organic Chemistry, Год журнала: 2023, Номер 43(2), С. 789 - 789

Опубликована: Янв. 1, 2023

Язык: Английский

Процитировано

4

Convergent Paired Electrolysis for the Synthesis of Pyrazolyl‐Substituted Tetrahydroisoquinolines DOI Open Access

Yanyan Kong,

Mengmeng Huang, Yabo Li

и другие.

Advanced Synthesis & Catalysis, Год журнала: 2023, Номер 365(23), С. 4198 - 4204

Опубликована: Окт. 24, 2023

Abstract A convergent paired electrolysis method for the synthesis of 1‐pyrazolyl‐substituted tetrahydroisoquinolines has been developed. The reaction proceeded without any transition metal catalyst and chemical oxidant. desired products could be isolated in high yields (80–99%) 60–80 minutes. Faradaic efficiency was 108% gram‐scale (84%) carried out. Mechanistic studies revealed that C−N bond formation process might mainly involve a nucleophilic addition reaction.

Язык: Английский

Процитировано

2

Synthetic Access to 1,3-Butadiynes via Electro-redox Cuprous-Catalyzed Dehydrogenative Csp–Csp Homocoupling of Terminal Acetylenes DOI
Murugavel Kathiresan, Chandrasekar Praveen,

Murugan Krishnan

и другие.

Synthesis, Год журнала: 2023, Номер 56(05), С. 777 - 786

Опубликована: Ноя. 8, 2023

Abstract Herein, we disclose the oxidative homocoupling of terminal alkynes under electrochemically generated cuprous catalysis. The scope this protocol was established by preparing an array structurally and electronically different 1,3-butadiyne derivatives. Good synthetic yields, functional group tolerance, oxidant-free conditions, no cross-selectivity are some intrinsic advantages methodology. developed chemistry features electro-redox formation copper acetylide, intermediate appropriate for Csp–Csp coupling step. chemical state in acetylide found to be Cu(I), as confirmed click trapping experiments, cyclic voltammetry, EPR spectroscopy, XPS. A competition reaction determine reactivity dissimilar acetylenes revealed that product ratio is rather dependent on electronic nature alkynyl substituents. To highlight value products, selected diynes were subjected diversification.

Язык: Английский

Процитировано

2

I2-Mediated [3 + 3] Annulation for the Construction of Indole-Pyrimidine-Pyrazole-Fused Tetracyclic Heteroarenes DOI

Heng-Tong Qu,

Long-Sheng Zhou,

Jiaxin Yang

и другие.

The Journal of Organic Chemistry, Год журнала: 2024, Номер 89(20), С. 15164 - 15169

Опубликована: Окт. 7, 2024

An I2-mediated annulation of 3-aminopyrazoles with indole-3-carboxaldehydes has been demonstrated for the first time. This tandem strategy allows facile construction indole-pyrimidine-pyrazole-fused tetracyclic heteroarenes that are otherwise inaccessible by existing methods. These fused heterocycles exhibited enhanced antifungal activities against Valsa mali and Botryosphaeria dothidea compared commercial Xemium fungicide.

Язык: Английский

Процитировано

0