Synthesis of Thiaphenanthridinones from Sulfinate Esters and 2-Borylanilines DOI Creative Commons
Keisuke Nakamura,

Minori Suzuki,

Suguru Yoshida

et al.

Organic Letters, Journal Year: 2024, Volume and Issue: 26(45), P. 9676 - 9681

Published: Nov. 6, 2024

A facile palladium-catalyzed synthesis of thiaphenanthridinones from sulfinate esters and 2-borylanilines is disclosed. Various sulfur analogs phenanthridinones were synthesized by bromide-selective cross-coupling cyclization in one step. Further transformations the obtained allowed preparing a broad range thiaphenanthridinone derivatives involving bioactive compounds.

Language: Английский

Recent advances in the synthesis and transformations of sulfinate esters DOI Creative Commons
Suguru Yoshida

Chemical Communications, Journal Year: 2025, Volume and Issue: unknown

Published: Jan. 1, 2025

Recent sulfinate esters chemistry is summarized in this feature article. Efficient methods to synthesize diverse from readily available starting materials and various modern transformations of are introduced.

Language: Английский

Citations

0

Synthesis of Thiaphenanthridinones from Sulfinate Esters and 2-Borylanilines DOI Creative Commons
Keisuke Nakamura,

Minori Suzuki,

Suguru Yoshida

et al.

Organic Letters, Journal Year: 2024, Volume and Issue: 26(45), P. 9676 - 9681

Published: Nov. 6, 2024

A facile palladium-catalyzed synthesis of thiaphenanthridinones from sulfinate esters and 2-borylanilines is disclosed. Various sulfur analogs phenanthridinones were synthesized by bromide-selective cross-coupling cyclization in one step. Further transformations the obtained allowed preparing a broad range thiaphenanthridinone derivatives involving bioactive compounds.

Language: Английский

Citations

1