New Insights into the Development of Donepezil-Based Hybrid and Natural Molecules as Multi-Target Drug Agents for Alzheimer’s Disease Treatment DOI Creative Commons
Violina T. Angelova, Boris Petrov Stoyanov, Rumyana Simeonova

et al.

Molecules, Journal Year: 2024, Volume and Issue: 29(22), P. 5314 - 5314

Published: Nov. 11, 2024

Alzheimer's disease (AD) involves a complex pathophysiology with multiple interconnected subpathologies, including protein aggregation, impaired neurotransmission, oxidative stress, and microglia-mediated neuroinflammation. Current treatments, which generally target single subpathology, have failed to modify the disease's progression, providing only temporary symptom relief. Multi-target drugs (MTDs) address several aggregation of pathological proteins. In this review, we cover hybrid molecules published between 2014 2024. We offer an overview strategies employed in drug design approaches that led notable improvements reduced hepatotoxicity. Our aim is insights into potential development new drugs. This highlights multi-target featuring heterocycles

Language: Английский

Mental health law in Philippines: health policy issues governing mental health promotion among Filipino older adults with serious mental illnesses DOI

Muamar O. Aldalaeen,

Rabia H. Haddad,

Talal Bani Ahmad

et al.

Mental Health and Social Inclusion, Journal Year: 2025, Volume and Issue: unknown

Published: Jan. 22, 2025

Purpose This study aims to discuss the mental health in Philippines and existing laws policies governing care among Filipino older adults with serious illnesses. Design/methodology/approach The used policy research understand issues gaps Philippine health-care system adults. deductive methods (based on testing specific hypotheses) inductive of inquiry formation general inferences), which are necessary but insufficient for theory development without retroductive reasoning. researcher believes that critical realism provides a philosophically grounded theoretical framework can be underpin into causal mechanisms such as analysis. Findings Mental is integral holistic health. commitment improve services highlighted recent legislative actions policymakers. professionals experts suggest failure address psycho-social problems population will hinder attempts increase social capital, promote human reduce poverty. Originality/value A disregard still apparent. norm continues include chronic shortage professionals, an inadequate number facilities hospitals, lack accessible equitable treatment, especially marginalized sectors, stigma, discrimination exclusion against people conditions very widespread. Some refuse even get help treatment their disorders not because high cost stigma attached disorders.

Language: Английский

Citations

1

Impact of GSK-3β and CK-1δ on Wnt signaling pathway in alzheimer disease: A dual target approach DOI
Vinita Sharma, Prabodh Chander Sharma,

Jurnal Reang

et al.

Bioorganic Chemistry, Journal Year: 2024, Volume and Issue: 147, P. 107378 - 107378

Published: April 17, 2024

Language: Английский

Citations

5

Computational Analysis of Stilbenes as Potential Multi-Targeted Therapeutics for Alzheimer’s Disease DOI Creative Commons
Seda Şirin

Osmaniye Korkut Ata Üniversitesi Fen Bilimleri Enstitüsü Dergisi, Journal Year: 2025, Volume and Issue: 8(1), P. 145 - 166

Published: Jan. 15, 2025

Purpose: The aim of this study is to compare 13 stilbenes and 5 FDA-approved drugs used in the treatment Alzheimer’s disease (AD) by ADME prediction molecular docking method. Cholinergic, amyloid, tau, oxidative stress inflammation hypotheses involved AD pathology were targeted docking. Materials Methods: SwissADME has been determine physicochemical, lipophilicity, water solubility, pharmacokinetics, drug-likeness medicinal chemistry properties (resveratrol, pterostilbene, oxyresveratrol, piceatannol, pinosylvin, isorhapontigenin, isorhapontin, astringin, piceid (polydatin), mulberroside A) (tacrine, donepezil, rivastigmine, galantamine, memantine). CBDOCK2 binding affinity target proteins (AChE, BuChE, APP, BACE, GSK-3β, CDK5, SOD, CAT, GPx, Cox-2, iNOS, IL-1β, TNF-α). Results: SWISS results showed that could be as natural products AD. indicated A best vina score (kcal/mol) followed galanthamine, resveratrol, tacrine, memantine. Conclusion: Our evaluated for using computational approaches. highlight its potential therapeutic effects on various pathology. More research needed validate these findings clinical practice.

Language: Английский

Citations

0

Gene Co-Expression Analysis Reveals Functional Differences Between Early- and Late-Onset Alzheimer’s Disease DOI Creative Commons

Abel Isaías Gutiérrez Cruz,

Guillermo de Anda‐Jáuregui, Enrique Hernández-Lemus

et al.

Current Issues in Molecular Biology, Journal Year: 2025, Volume and Issue: 47(3), P. 200 - 200

Published: March 18, 2025

The rising prevalence of Alzheimer’s disease (AD), particularly among older adults, has driven increased research into its underlying mechanisms and risk factors. Aging, genetic susceptibility, cardiovascular health are recognized contributors to AD, but how the age onset affects progression remains underexplored. This study investigates role early- versus late-onset (EOAD LOAD, respectively) in shaping trajectory cognitive decline. Leveraging data from Religious Orders Study Memory Aging Project (ROSMAP), two cohorts were established: individuals with early-onset AD those AD. Comprehensive analyses, including differential gene expression profiling, pathway enrichment, co-expression network construction, conducted identify distinct molecular signatures associated each cohort. Network modularity learning algorithms used discern inner structure networks their related functional features. Computed descriptors provided deeper insights influence at on biological

Language: Английский

Citations

0

Introduction to Alzheimer's Disease, Biomarkers, and the AI Revolution DOI
Bancha Yingngam

Advances in medical technologies and clinical practice book series, Journal Year: 2024, Volume and Issue: unknown, P. 1 - 23

Published: June 28, 2024

Alzheimer's disease (AD) is a progressive neurodegenerative that results in steady decline cognitive ability and memory function. As society ages, the need for an optimum AD management strategy becomes more important. This chapter analyzes stage-construction etiology escalating symptoms of discovered throughout this review, as well identification barrier to precise diagnosis. The artificial intelligence achieve quicker detection through machine learning, data analytics, predictive modeling also being considered. Therefore, employing AI AD-related studies novel approach enhancing patient outcomes. Proper diagnosis parallel increased probability many parameters one most difficult moments identify. However, use evaluation sensor network technologies big analysis has advanced, preventive instruments can be used. Thus, technology gives humanity hope stop or, at very least, slow down tragedy.

Language: Английский

Citations

1

Emerging Role of Medicinal Herbs on Alzheimer’s Disease and Memory Deficits DOI Creative Commons
Sadaf Naeem, Saira Saeed Khan, Yousra Shafiq

et al.

IntechOpen eBooks, Journal Year: 2024, Volume and Issue: unknown

Published: Aug. 30, 2024

Alzheimer’s disease (AD) is an age-related neurodegenerative disorder characterized by memory deficits. It associated with the presence of intracellular neurofibrillary tangles (NFTs) and extracellular amyloid beta plaques, loss neuronal subpopulations, cholinergic fibers, microglial inactivation. According to studies, from year 2000–2020, death toll attributed AD increased 146.2%, its major causes are neurodegeneration oxidative stress (OS). Currently, available treatment options limited, there no cure for disease. In Asia, such as in China India, herbal medicines have been used diseases thousands years, which has recently attracted considerable attention due development curative drugs AD. this chapter, we first summarized pathogenic factors secondly, that extensively investigated both models clinical trials. Also, specified potential targets herbs view signaling pathways implicated inflammatory pathogenesis. We consider knowledge can be favorable disease-modifying

Language: Английский

Citations

0

New Insights into the Development of Donepezil-Based Hybrid and Natural Molecules as Multi-Target Drug Agents for Alzheimer’s Disease Treatment DOI Creative Commons
Violina T. Angelova, Boris Petrov Stoyanov, Rumyana Simeonova

et al.

Molecules, Journal Year: 2024, Volume and Issue: 29(22), P. 5314 - 5314

Published: Nov. 11, 2024

Alzheimer's disease (AD) involves a complex pathophysiology with multiple interconnected subpathologies, including protein aggregation, impaired neurotransmission, oxidative stress, and microglia-mediated neuroinflammation. Current treatments, which generally target single subpathology, have failed to modify the disease's progression, providing only temporary symptom relief. Multi-target drugs (MTDs) address several aggregation of pathological proteins. In this review, we cover hybrid molecules published between 2014 2024. We offer an overview strategies employed in drug design approaches that led notable improvements reduced hepatotoxicity. Our aim is insights into potential development new drugs. This highlights multi-target featuring heterocycles

Language: Английский

Citations

0