Metformin Impairs Linsitinib Anti-Tumor Effect on Ovarian Cancer Cell Lines DOI Open Access
Diana Luísa Almeida-Nunes, João P. N. Silva, Mariana Nunes

et al.

International Journal of Molecular Sciences, Journal Year: 2024, Volume and Issue: 25(22), P. 11935 - 11935

Published: Nov. 6, 2024

Ovarian cancer (OC) remains one of the leading causes cancer-related mortality among women. Targeting insulin-like growth factor 1 (IGF-1) signaling pathway has emerged as a promising therapeutic strategy. Linsitinib, an IGF-1 receptor (IGF-1R) inhibitor, shown potential in disrupting this pathway. Additionally, metformin, commonly used treatment type 2 diabetes, been studied for its anti-cancer properties due to ability inhibit metabolic pathways that intersect with signaling, making it candidate combination therapy treatments. This study explores effects linsitinib and metformin on OVCAR3 cells by suppression siRNA-mediated

Language: Английский

P-cadherin overexpression is associated with early transformation of the Fallopian tube epithelium and aggressiveness of tubo-ovarian high-grade serous carcinoma DOI Creative Commons
R. Canário, Ana Sofia Ribeiro, Inês Morgado

et al.

Virchows Archiv, Journal Year: 2025, Volume and Issue: unknown

Published: May 5, 2025

Abstract Tubo-ovarian high-grade serous carcinoma (HGSC) with proficient homologous recombination (HR) DNA repair (HRP) accounts for approximately 50% of cases and is associated platinum-resistance poor prognosis. We hypothesize that the acquisition hybrid phenotypes displaying both epithelial mesenchymal (E/M) features may be involved in malignant transformation tumour dissemination this subgroup. Therefore, we analysed, by digital pathology, expression prognostic significance 3 classic cadherins (E-cadherin, marker; N-cadherin, P-cadherin, candidate marker E/M) 577 formalin-fixed paraffin-embedded human samples representing putative stepwise carcinogenesis Fallopian tube epithelium (FTE). observed a non-canonical N-to-P-cadherin switch along carcinogenic progression, statistically significant overexpression P-cadherin pre-malignant samples, compared to control FTE. Interestingly, was most pronounced precursor lesions HGSC cells from ascites. Tumours high were significantly worse overall survival, especially subgroup without BRCA1/2 mutations. Transient knock-down resulted vitro reduction functional E/M hallmarks, namely decreased anoikis resistance, reduced collective migration invasion representative platinum-resistant HRP cell line. Taken together, our results suggest an early event activation HRP-HGSC, further supporting adhesion molecule as promising biomarker

Language: Английский

Citations

0

Metformin Impairs Linsitinib Anti-Tumor Effect on Ovarian Cancer Cell Lines DOI Open Access
Diana Luísa Almeida-Nunes, João P. N. Silva, Mariana Nunes

et al.

International Journal of Molecular Sciences, Journal Year: 2024, Volume and Issue: 25(22), P. 11935 - 11935

Published: Nov. 6, 2024

Ovarian cancer (OC) remains one of the leading causes cancer-related mortality among women. Targeting insulin-like growth factor 1 (IGF-1) signaling pathway has emerged as a promising therapeutic strategy. Linsitinib, an IGF-1 receptor (IGF-1R) inhibitor, shown potential in disrupting this pathway. Additionally, metformin, commonly used treatment type 2 diabetes, been studied for its anti-cancer properties due to ability inhibit metabolic pathways that intersect with signaling, making it candidate combination therapy treatments. This study explores effects linsitinib and metformin on OVCAR3 cells by suppression siRNA-mediated

Language: Английский

Citations

0