Dual-Responsive Methotrexate-Human Serum Albumin Complex-Encapsulated Liposomes for Targeted and Enhanced Atherosclerosis Therapy DOI Creative Commons
Xueqin Wang, Xiaodong Chen, Huiping Ji

et al.

International Journal of Nanomedicine, Journal Year: 2025, Volume and Issue: Volume 20, P. 2305 - 2322

Published: Feb. 1, 2025

In plaque sites of atherosclerosis (AS), the physiological barrier caused by thick fiber cap due to overmigration vascular smooth muscle cells (VSMCs) prevents efficient drug delivery damaged macrophages. How ensure precise targeted drugs and their on-demand release dysfunctional under fibrous are feasible solutions enhance AS treatment. A small complex methotrexate (MTX)-human serum albumin (HSA) with strong, penetration ability was encapsulated in a cholesterol hemisuccinate (CHEM) prepared pH-sensitive liposome, modifying ROS-responsive PEG2000-TK-DSPE (PTD), termed PTD/Lipo/MTX-HSA. PTD/Lipo/MTX-HSA can achieve targeting response plaques environments AS. The designed formulation accelerated small-sized MTX-HSA excess ROS acidic pH conditions, it better penetrated macrophage spheroids. Furthermore, has mouse model produce good anti-inflammatory efficacy inhibiting p65 entry into nucleus turn out inflammatory factor. Our formulations work safety mind, also highlights potential precisely on-demand-released dual-responsive smart nanoplatforms as promising therapeutic options penetrate deeper for effective treatment

Language: Английский

Single-cell and spatial analysis reveals the interaction between ITLN1+ foam cells and SPP1+ macrophages in atherosclerosis DOI Creative Commons
Minghao Yin, Shanshan Wang, Ruidan Zhang

et al.

Frontiers in Cardiovascular Medicine, Journal Year: 2025, Volume and Issue: 12

Published: Feb. 13, 2025

Introduction Cardiovascular disease (CVD) caused by atherosclerosis (AS) remains the leading cause of mortality in developed countries. Understanding cellular heterogeneity within inflammatory microenvironment is crucial for advancing management strategies. This study investigates regulatory functions distinct cell populations AS pathogenesis, focusing on interaction between vascular smooth muscle (VSMC)-derived ITLN1 + foam cells and SPP1 FABP5 macrophages. Methods We employed single-cell RNA sequencing to characterize plaques. Correlation analyses CellChat package were utilized elucidate intercellular communication networks among various types. The functional roles key subsets macrophages VSMCs assessed using Gene Ontology (GO) Kyoto Encyclopedia Genes Genomes (KEGG) pathway analyses. Pseudotime trajectory analysis was conducted explore dynamics VSMC differentiation. Additionally, spatial transcriptomics used demonstrate physical interactions different subpopulations. Results identified significant infiltration macrophage clusters AS, with being highly enriched These associated lipid transport, storage, migration pathways. A subset derived from exhibited robust expression markers metabolism-related genes. indicated that represent a terminal stage differentiation, characterized elevated genes linked synthesis progression. Spatial revealed macrophages, mediated MIF-(CD74 CD44) SPP1-CD44 ligand-receptor axes. Discussion Our findings underscore critical crosstalk promoting accumulation Targeting this cell-cell may offer new therapeutic avenues managing atherosclerosis. Further validation these mechanisms necessary develop effective immunotherapeutic strategies against AS.

Language: Английский

Citations

0

Dual-Responsive Methotrexate-Human Serum Albumin Complex-Encapsulated Liposomes for Targeted and Enhanced Atherosclerosis Therapy DOI Creative Commons
Xueqin Wang, Xiaodong Chen, Huiping Ji

et al.

International Journal of Nanomedicine, Journal Year: 2025, Volume and Issue: Volume 20, P. 2305 - 2322

Published: Feb. 1, 2025

In plaque sites of atherosclerosis (AS), the physiological barrier caused by thick fiber cap due to overmigration vascular smooth muscle cells (VSMCs) prevents efficient drug delivery damaged macrophages. How ensure precise targeted drugs and their on-demand release dysfunctional under fibrous are feasible solutions enhance AS treatment. A small complex methotrexate (MTX)-human serum albumin (HSA) with strong, penetration ability was encapsulated in a cholesterol hemisuccinate (CHEM) prepared pH-sensitive liposome, modifying ROS-responsive PEG2000-TK-DSPE (PTD), termed PTD/Lipo/MTX-HSA. PTD/Lipo/MTX-HSA can achieve targeting response plaques environments AS. The designed formulation accelerated small-sized MTX-HSA excess ROS acidic pH conditions, it better penetrated macrophage spheroids. Furthermore, has mouse model produce good anti-inflammatory efficacy inhibiting p65 entry into nucleus turn out inflammatory factor. Our formulations work safety mind, also highlights potential precisely on-demand-released dual-responsive smart nanoplatforms as promising therapeutic options penetrate deeper for effective treatment

Language: Английский

Citations

0