Exploring the therapeutic potential of glucagon-like peptide 1 agonists in metabolic disorders DOI
Adrián Cortés‐Martín, Julio Plaza‐Díaz

World Journal of Gastroenterology, Journal Year: 2024, Volume and Issue: 31(4)

Published: Dec. 30, 2024

This article comments on the work by Soresi and Giannitrapani. The authors have stated that one of most novel promising treatments for metabolic dysfunction-associated steatotic liver disease (MASLD) is use glucagon-like peptide 1 receptor agonists, especially when used in combination therapy. However, despite their notable efficacy, these drugs were not initially designed to target MASLD directly. In a groundbreaking development, Food Drug Administration has recently approved resmetirom, first treatment specifically aimed at reducing fibrosis metabolic-associated steatohepatitis. Resmetirom, an orally administered, liver-directed thyroid hormone beta-selective agonist, acts directly intrahepatic pathways, enhancing its therapeutic potential marking beginning new era MASLD. Furthermore, integration lifestyle modifications into management essential component should be considered reinforced. By incorporating dietary changes regular physical exercise treatment, patients may achieve improved outcomes, need pharmacological interventions and/or improving efficacy. As complement medical therapies, factors overlooked broader strategy managing

Language: Английский

Caloric restriction and its mimetics in heart failure with preserved ejection fraction: mechanisms and therapeutic potential DOI Creative Commons

Alexander Fuerlinger,

Alina Stockner,

Simon Sedej

et al.

Cardiovascular Diabetology, Journal Year: 2025, Volume and Issue: 24(1)

Published: Jan. 18, 2025

Language: Английский

Citations

2

A Remotely Delivered, GLP-1RA-Supported Specialist Weight Management Program: 12 Month Outcomes From a Retrospective Service Evaluation (Preprint) DOI Creative Commons
Rebecca Richards, Michael Whitman, Gina Wren

et al.

Published: Feb. 14, 2025

BACKGROUND Limited access to specialist weight management services (SWMS) restricts the implementation of novel obesity pharmacotherapy in United Kingdom’s (UK) National Health Service (NHS). Remote delivery GLP-1 receptor agonist (GLP-1RA) medication with digital behavioural support could provide a scalable solution, but evidence for long-term effectiveness is limited OBJECTIVE To evaluate effectiveness, feasibility, acceptability and potential cost-effectiveness Second Nature's remotely-delivered, semaglutide-supported program over 12 months METHODS Retrospective data were extracted participants who initiated intervention between September December 2023. Primary outcome was change at months. Secondary outcomes included behavioral changes, side effects, engagement, participant experience comparative cost analysis against NHS SWMS. Descriptive statistics paired two-tailed t-tests evaluated outcomes. Content used qualitative data. RESULTS Of 341 (82.8% women; mean age 49.0 years, SD 11.1; baseline BMI 37.9 kg/m², 6.9). Participants active subscriptions (39.6%, n=135) achieved 20.0 kg (19.1%, ,P<.001) loss versus 12.4 (11.9%) inactive subscriptions. Overall, 77.7% ≥10% 61.5% ≥15%. Program engagement declined from 113 (SD 78.4) home screen views month 1 25 29.06) 12. Side effects decreased time, 69.6% reporting none by Most reported positive (34.2%) or neutral (56.7%) experiences The costs estimated 30-40% current SWMS, projecting savings £1.5m-£1.8m per 100,000 population CONCLUSIONS This evaluation suggests that remotely-delivered GLP-1RA-supported can be effective, feasible, acceptable cost-effective people living obesity. Further research within public healthcare settings needed clinical assess sustained results continuation discontinuation medication.

Language: Английский

Citations

0

Efficacy and Safety of Tirzepatide for Weight Management in Non-Diabetic Obese Individuals: A Narrative Review DOI Creative Commons
Mohammed Sallam, Johan Snygg, Sara El Ghandour

et al.

Obesities, Journal Year: 2025, Volume and Issue: 5(2), P. 26 - 26

Published: April 18, 2025

Obesity represents a global health challenge, with critical and urgent need for long-term, sustainable management strategies. Tirzepatide is novel dual glucose-dependent insulinotropic polypeptide (GIP) glucagon-like peptide-1 (GLP-1) receptor agonist. At first approved the treatment of type 2 diabetes mellitus, tirzepatide one latest clinically commercially available pharmacological options obesity management. This narrative review aimed to synthesize existing clinical evidence on efficacy safety in non-diabetic obese individuals. A comprehensive literature search was conducted using PubMed, Scopus, Web Science, ClinicalTrials.gov, Google Scholar databases identify relevant trials, meta-analyses, original studies assessing weight-loss impact from 2022 onwards. Synthesized indicated that achieved up 20.9% weight loss over 72 weeks (SURMOUNT-1), 18.4% after lifestyle intervention (SURMOUNT-3), 17.5% Chinese adults (SURMOUNT-CN), 25.3% continued 88 (SURMOUNT-4). Meta-analyses confirmed higher odds ≥5–20% versus semaglutide liraglutide, significantly reducing body mass index, waist circumference, blood pressure, atherosclerotic cardiovascular disease risk. Health-related quality life improved greater loss, gastrointestinal side effects (nausea, diarrhea, constipation) were common but mild moderate, <5% discontinuation. significant cardiometabolic benefits, individuals, further research needed long-term efficacy, safety, application.

Language: Английский

Citations

0

Exploring the therapeutic potential of glucagon-like peptide 1 agonists in metabolic disorders DOI
Adrián Cortés‐Martín, Julio Plaza‐Díaz

World Journal of Gastroenterology, Journal Year: 2024, Volume and Issue: 31(4)

Published: Dec. 30, 2024

This article comments on the work by Soresi and Giannitrapani. The authors have stated that one of most novel promising treatments for metabolic dysfunction-associated steatotic liver disease (MASLD) is use glucagon-like peptide 1 receptor agonists, especially when used in combination therapy. However, despite their notable efficacy, these drugs were not initially designed to target MASLD directly. In a groundbreaking development, Food Drug Administration has recently approved resmetirom, first treatment specifically aimed at reducing fibrosis metabolic-associated steatohepatitis. Resmetirom, an orally administered, liver-directed thyroid hormone beta-selective agonist, acts directly intrahepatic pathways, enhancing its therapeutic potential marking beginning new era MASLD. Furthermore, integration lifestyle modifications into management essential component should be considered reinforced. By incorporating dietary changes regular physical exercise treatment, patients may achieve improved outcomes, need pharmacological interventions and/or improving efficacy. As complement medical therapies, factors overlooked broader strategy managing

Language: Английский

Citations

0